These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

295 related articles for article (PubMed ID: 24564570)

  • 1. Diamidine compounds for selective inhibition of protein arginine methyltransferase 1.
    Yan L; Yan C; Qian K; Su H; Kofsky-Wofford SA; Lee WC; Zhao X; Ho MC; Ivanov I; Zheng YG
    J Med Chem; 2014 Mar; 57(6):2611-22. PubMed ID: 24564570
    [TBL] [Abstract][Full Text] [Related]  

  • 2. The Development of Tetrazole Derivatives as Protein Arginine Methyltransferase I (PRMT I) Inhibitors.
    Sun Y; Wang Z; Yang H; Zhu X; Wu H; Ma L; Xu F; Hong W; Wang H
    Int J Mol Sci; 2019 Aug; 20(15):. PubMed ID: 31390828
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Design and synthesis of novel PRMT1 inhibitors and investigation of their binding preferences using molecular modelling.
    Yang H; Ouyang Y; Ma H; Cong H; Zhuang C; Lok WT; Wang Z; Zhu X; Sun Y; Hong W; Wang H
    Bioorg Med Chem Lett; 2017 Oct; 27(20):4635-4642. PubMed ID: 28927791
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Exploration of cyanine compounds as selective inhibitors of protein arginine methyltransferases: synthesis and biological evaluation.
    Hu H; Owens EA; Su H; Yan L; Levitz A; Zhao X; Henary M; Zheng YG
    J Med Chem; 2015 Feb; 58(3):1228-43. PubMed ID: 25559100
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Novel inhibitors for PRMT1 discovered by high-throughput screening using activity-based fluorescence polarization.
    Dillon MB; Bachovchin DA; Brown SJ; Finn MG; Rosen H; Cravatt BF; Mowen KA
    ACS Chem Biol; 2012 Jul; 7(7):1198-204. PubMed ID: 22506763
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Discovery of alkyl bis(oxy)dibenzimidamide derivatives as novel protein arginine methyltransferase 1 (PRMT1) inhibitors.
    Zhang WY; Lu WC; Jiang H; Lv ZB; Xie YQ; Lian FL; Liang ZJ; Jiang YX; Wang DJ; Luo C; Jin J; Ye F
    Chem Biol Drug Des; 2017 Dec; 90(6):1260-1270. PubMed ID: 28636189
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Development of Potent Type I Protein Arginine Methyltransferase (PRMT) Inhibitors of Leukemia Cell Proliferation.
    Wang C; Jiang H; Jin J; Xie Y; Chen Z; Zhang H; Lian F; Liu YC; Zhang C; Ding H; Chen S; Zhang N; Zhang Y; Jiang H; Chen K; Ye F; Yao Z; Luo C
    J Med Chem; 2017 Nov; 60(21):8888-8905. PubMed ID: 29019697
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Small molecule inhibitors that discriminate between protein arginine N-methyltransferases PRMT1 and CARM1.
    Dowden J; Pike RA; Parry RV; Hong W; Muhsen UA; Ward SG
    Org Biomol Chem; 2011 Oct; 9(22):7814-21. PubMed ID: 21952734
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Investigating the binding preferences of small molecule inhibitors of human protein arginine methyltransferase 1 using molecular modelling.
    Hong W; Li J; Laughton CA; Yap LF; Paterson IC; Wang H
    J Mol Graph Model; 2014 Jun; 51():193-202. PubMed ID: 24937176
    [TBL] [Abstract][Full Text] [Related]  

  • 10. A Pan-Inhibitor for Protein Arginine Methyltransferase Family Enzymes.
    Iyamu ID; Al-Hamashi AA; Huang R
    Biomolecules; 2021 Jun; 11(6):. PubMed ID: 34201091
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Inhibitory study of protein arginine methyltransferase 1 using a fluorescent approach.
    Feng Y; Xie N; Wu J; Yang C; Zheng YG
    Biochem Biophys Res Commun; 2009 Feb; 379(2):567-72. PubMed ID: 19121292
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Virtual screening and biological evaluation of novel small molecular inhibitors against protein arginine methyltransferase 1 (PRMT1).
    Xie Y; Zhou R; Lian F; Liu Y; Chen L; Shi Z; Zhang N; Zheng M; Shen B; Jiang H; Liang Z; Luo C
    Org Biomol Chem; 2014 Dec; 12(47):9665-73. PubMed ID: 25348815
    [TBL] [Abstract][Full Text] [Related]  

  • 13. In situ generation of a bisubstrate analogue for protein arginine methyltransferase 1.
    Osborne T; Roska RL; Rajski SR; Thompson PR
    J Am Chem Soc; 2008 Apr; 130(14):4574-5. PubMed ID: 18338885
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Structure, Function, and Activity of Small Molecule and Peptide Inhibitors of Protein Arginine Methyltransferase 1.
    Hendrickson-Rebizant T; Sudhakar SRN; Rowley MJ; Frankel A; Davie JR; Lakowski TM
    J Med Chem; 2024 Sep; 67(18):15931-15946. PubMed ID: 39250434
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Discovery of a Potent Class I Protein Arginine Methyltransferase Fragment Inhibitor.
    Ferreira de Freitas R; Eram MS; Szewczyk MM; Steuber H; Smil D; Wu H; Li F; Senisterra G; Dong A; Brown PJ; Hitchcock M; Moosmayer D; Stegmann CM; Egner U; Arrowsmith C; Barsyte-Lovejoy D; Vedadi M; Schapira M
    J Med Chem; 2016 Feb; 59(3):1176-83. PubMed ID: 26824386
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Transient Kinetics Define a Complete Kinetic Model for Protein Arginine Methyltransferase 1.
    Hu H; Luo C; Zheng YG
    J Biol Chem; 2016 Dec; 291(52):26722-26738. PubMed ID: 27834681
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and evaluation of protein arginine N-methyltransferase inhibitors designed to simultaneously occupy both substrate binding sites.
    van Haren M; van Ufford LQ; Moret EE; Martin NI
    Org Biomol Chem; 2015 Jan; 13(2):549-60. PubMed ID: 25380215
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Histone H4-based peptoids are inhibitors of protein arginine methyltransferase 1 (PRMT1).
    Mann SA; DeMart MK; May B; Causey CP; Knuckley B
    Biochem J; 2020 Aug; 477(16):2971-2980. PubMed ID: 32716034
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Protein arginine methyltransferase 1: positively charged residues in substrate peptides distal to the site of methylation are important for substrate binding and catalysis.
    Osborne TC; Obianyo O; Zhang X; Cheng X; Thompson PR
    Biochemistry; 2007 Nov; 46(46):13370-81. PubMed ID: 17960915
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Toward the development of potent and selective bisubstrate inhibitors of protein arginine methyltransferases.
    Dowden J; Hong W; Parry RV; Pike RA; Ward SG
    Bioorg Med Chem Lett; 2010 Apr; 20(7):2103-5. PubMed ID: 20219369
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 15.