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15. IV. Discovery of CXCR3 antagonists substituted with heterocycles as amide surrogates: improved PK, hERG and metabolic profiles. Nair AG; Wong MK; Shu Y; Jiang Y; Jenh CH; Kim SH; Yang DY; Zeng Q; Shao Y; Zawacki LG; Duo J; McGuinness BF; Carroll CD; Hobbs DW; Shih NY; Rosenblum SB; Kozlowski JA Bioorg Med Chem Lett; 2014 Feb; 24(4):1085-8. PubMed ID: 24486132 [TBL] [Abstract][Full Text] [Related]
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