BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

182 related articles for article (PubMed ID: 24650641)

  • 1. Arylamino bisphosphonates: potent and selective inhibitors of the tumor-associated carbonic anhydrase XII.
    Tauro M; Loiodice F; Ceruso M; Supuran CT; Tortorella P
    Bioorg Med Chem Lett; 2014 Apr; 24(8):1941-3. PubMed ID: 24650641
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Carbonic anhydrase inhibitors: synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety.
    Sethi KK; Vullo D; Verma SM; Tanç M; Carta F; Supuran CT
    Bioorg Med Chem; 2013 Oct; 21(19):5973-82. PubMed ID: 23965175
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Dual carbonic anhydrase/matrix metalloproteinase inhibitors incorporating bisphosphonic acid moieties targeting bone tumors.
    Tauro M; Loiodice F; Ceruso M; Supuran CT; Tortorella P
    Bioorg Med Chem Lett; 2014 Jun; 24(12):2617-20. PubMed ID: 24813742
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Pyrazolylbenzo[d]imidazoles as new potent and selective inhibitors of carbonic anhydrase isoforms hCA IX and XII.
    Kumar S; Ceruso M; Tuccinardi T; Supuran CT; Sharma PK
    Bioorg Med Chem; 2016 Jul; 24(13):2907-2913. PubMed ID: 27166574
    [TBL] [Abstract][Full Text] [Related]  

  • 5. N-β-glycosyl sulfamides are selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII.
    Rodríguez OM; Maresca A; Témpera CA; Bravo RD; Colinas PA; Supuran CT
    Bioorg Med Chem Lett; 2011 Aug; 21(15):4447-50. PubMed ID: 21723123
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII--a new scaffold for designing isoform-selective inhibitors.
    Carradori S; De Monte C; D'Ascenzio M; Secci D; Celik G; Ceruso M; Vullo D; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2013 Dec; 23(24):6759-63. PubMed ID: 24189056
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis of 6-tetrazolyl-substituted sulfocoumarins acting as highly potent and selective inhibitors of the tumor-associated carbonic anhydrase isoforms IX and XII.
    Grandane A; Tanc M; Zalubovskis R; Supuran CT
    Bioorg Med Chem; 2014 Mar; 22(5):1522-8. PubMed ID: 24513186
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Metronidazole-coumarin conjugates and 3-cyano-7-hydroxy-coumarin act as isoform-selective carbonic anhydrase inhibitors.
    Bonneau A; Maresca A; Winum JY; Supuran CT
    J Enzyme Inhib Med Chem; 2013 Apr; 28(2):397-401. PubMed ID: 22299576
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Carbonic anhydrase inhibitors. Synthesis of heterocyclic 4-substituted pyridine-3-sulfonamide derivatives and their inhibition of the human cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII.
    Sławiński J; Szafrański K; Vullo D; Supuran CT
    Eur J Med Chem; 2013 Nov; 69():701-10. PubMed ID: 24095761
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Benzenesulfonamide bearing 1,2,4-triazole scaffolds as potent inhibitors of tumor associated carbonic anhydrase isoforms hCA IX and hCA XII.
    SitaRam ; Celik G; Khloya P; Vullo D; Supuran CT; Sharma PK
    Bioorg Med Chem; 2014 Mar; 22(6):1873-82. PubMed ID: 24560737
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII.
    Nocentini A; Carta F; Ceruso M; Bartolucci G; Supuran CT
    Bioorg Med Chem; 2015 Nov; 23(21):6955-66. PubMed ID: 26432607
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Dual targeting of cancer-related human matrix metalloproteinases and carbonic anhydrases by chiral N-(biarylsulfonyl)-phosphonic acids.
    Luisi G; Angelini G; Gasbarri C; Laghezza A; Agamennone M; Loiodice F; Supuran CT; Campestre C; Tortorella P
    J Enzyme Inhib Med Chem; 2017 Dec; 32(1):1260-1264. PubMed ID: 28948845
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.
    Saczewski F; Innocenti A; Sławiński J; Kornicka A; Brzozowski Z; Pomarnacka E; Scozzafava A; Temperini C; Supuran CT
    Bioorg Med Chem; 2008 Apr; 16(7):3933-40. PubMed ID: 18242998
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Novel coumarins and benzocoumarins acting as isoform-selective inhibitors against the tumor-associated carbonic anhydrase IX.
    Sharma A; Tiwari M; Supuran CT
    J Enzyme Inhib Med Chem; 2014 Apr; 29(2):292-6. PubMed ID: 23488741
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: solution and X-ray crystallographic studies.
    Bozdag M; Ferraroni M; Nuti E; Vullo D; Rossello A; Carta F; Scozzafava A; Supuran CT
    Bioorg Med Chem; 2014 Jan; 22(1):334-40. PubMed ID: 24300919
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Carbonic anhydrase inhibitors. Inhibition of the transmembrane isozyme XII with sulfonamides-a new target for the design of antitumor and antiglaucoma drugs?
    Vullo D; Innocenti A; Nishimori I; Pastorek J; Scozzafava A; Pastoreková S; Supuran CT
    Bioorg Med Chem Lett; 2005 Feb; 15(4):963-9. PubMed ID: 15686894
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Cyclic tertiary sulfamates: selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives.
    De Monte C; Carradori S; Secci D; D'Ascenzio M; Vullo D; Ceruso M; Supuran CT
    Eur J Med Chem; 2014 Sep; 84():240-6. PubMed ID: 25019479
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Structural investigations on coumarins leading to chromeno[4,3-c]pyrazol-4-ones and pyrano[4,3-c]pyrazol-4-ones: New scaffolds for the design of the tumor-associated carbonic anhydrase isoforms IX and XII.
    Bonardi A; Falsini M; Catarzi D; Varano F; Di Cesare Mannelli L; Tenci B; Ghelardini C; Angeli A; Supuran CT; Colotta V
    Eur J Med Chem; 2018 Feb; 146():47-59. PubMed ID: 29407972
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Carbonic anhydrase inhibitors. Interaction of the antiepileptic drug sulthiame with twelve mammalian isoforms: kinetic and X-ray crystallographic studies.
    Temperini C; Innocenti A; Mastrolorenzo A; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2007 Sep; 17(17):4866-72. PubMed ID: 17588751
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Attachment of carbohydrates to methoxyaryl moieties leads to highly selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII.
    Riafrecha LE; Rodríguez OM; Vullo D; Supuran CT; Colinas PA
    Bioorg Med Chem; 2014 Oct; 22(19):5308-14. PubMed ID: 25156300
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.