306 related articles for article (PubMed ID: 24651228)
1. An improved design of water-soluble propofol prodrugs characterized by rapid onset of action.
Lang BC; Yang J; Wang Y; Luo Y; Kang Y; Liu J; Zhang WS
Anesth Analg; 2014 Apr; 118(4):745-54. PubMed ID: 24651228
[TBL] [Abstract][Full Text] [Related]
2. Efficacy comparison of the novel water-soluble propofol prodrug HX0969w and fospropofol in mice and rats.
Zhou Y; Yang J; Liu J; Wang Y; Zhang WS
Br J Anaesth; 2013 Nov; 111(5):825-32. PubMed ID: 23801745
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and characterization of novel quick-release propofol prodrug via lactonization.
Yang J; Yin W; Liu J; Wang Y; Zhou C; Kang Y; Zhang WS
Bioorg Med Chem Lett; 2013 Mar; 23(6):1813-6. PubMed ID: 23395634
[TBL] [Abstract][Full Text] [Related]
4. [The sedative-hypnotic effects and safety of oral administrated propofol prodrugs hx0969w and fospropofol disodiun in comparison with propofol emulsion in rats].
Wang HY; Yang J; Yin W; Yang LH; Zhang WS
Sichuan Da Xue Xue Bao Yi Xue Ban; 2015 Mar; 46(2):214-7. PubMed ID: 25924432
[TBL] [Abstract][Full Text] [Related]
5. Pharmacokinetics and pharmacodynamics of GPI 15715 or fospropofol (Aquavan injection) - a water-soluble propofol prodrug.
Fechner J; Schwilden H; Schüttler J
Handb Exp Pharmacol; 2008; (182):253-66. PubMed ID: 18175095
[TBL] [Abstract][Full Text] [Related]
6. An improved water-soluble prodrug of propofol with high molecular utilization and rapid onset of action.
Zhang W; Yang J; Fan J; Wang B; Kang Y; Liu J; Zhang W; Zhu T
Eur J Pharm Sci; 2019 Jan; 127():9-13. PubMed ID: 30290219
[TBL] [Abstract][Full Text] [Related]
7. Synthesis, in vitro and in vivo characterization of novel ethyl dioxy phosphate prodrug of propofol.
Kumpulainen H; Järvinen T; Mannila A; Leppänen J; Nevalainen T; Mäntylä A; Vepsäläinen J; Rautio J
Eur J Pharm Sci; 2008 Jul; 34(2-3):110-7. PubMed ID: 18403185
[TBL] [Abstract][Full Text] [Related]
8. Design, Synthesis, and Activity Study of Water-Soluble, Rapid-Release Propofol Prodrugs.
Liu LQ; Hong PX; Song XH; Zhou CC; Ling R; Kang Y; Qi QR; Yang J
J Med Chem; 2020 Jul; 63(14):7857-7866. PubMed ID: 32588620
[TBL] [Abstract][Full Text] [Related]
9. The preclinical pharmacological study on HX0969W, a novel water-soluble pro-drug of propofol, in rats.
Zhang Y; Jiang Y; Wang H; Wang B; Yang J; Kang Y; Chen J; Liu J; Zhang WS
PeerJ; 2020; 8():e8922. PubMed ID: 32337104
[TBL] [Abstract][Full Text] [Related]
10. Fospropofol disodium, a water-soluble prodrug of the intravenous anesthetic propofol (2,6-diisopropylphenol).
Fechner J; Ihmsen H; Jeleazcov C; Schüttler J
Expert Opin Investig Drugs; 2009 Oct; 18(10):1565-71. PubMed ID: 19758110
[TBL] [Abstract][Full Text] [Related]
11. [Fospropofol: A new prodrug of propofol].
Telletxea S; Lauzirika Z; Etxebarria A; Ortega LF
Rev Esp Anestesiol Reanim; 2012 Nov; 59(9):497-502. PubMed ID: 22748853
[TBL] [Abstract][Full Text] [Related]
12. Interactive web simulation for propofol and fospropofol, a new propofol prodrug.
Yavas S; Lizdas D; Gravenstein N; Lampotang S
Anesth Analg; 2008 Mar; 106(3):880-3, table of contents. PubMed ID: 18292434
[TBL] [Abstract][Full Text] [Related]
13. Fospropofol assay issues and impact on pharmacokinetic and pharmacodynamic evaluation.
Shah A; Mistry B; Gibiansky E; Gibiansky L
Anesth Analg; 2009 Jan; 108(1):382; author reply 382-3. PubMed ID: 19095885
[No Abstract] [Full Text] [Related]
14. Propylene glycol-linked amino acid/dipeptide diester prodrugs of oleanolic acid for PepT1-mediated transport: synthesis, intestinal permeability, and pharmacokinetics.
Cao F; Gao Y; Wang M; Fang L; Ping Q
Mol Pharm; 2013 Apr; 10(4):1378-87. PubMed ID: 23339520
[TBL] [Abstract][Full Text] [Related]
15. Pharmacokinetics and pharmacodynamics of the new propofol prodrug GPI 15715 in rats.
Schywalsky M; Ihmsen H; Tzabazis A; Fechner J; Burak E; Vornov J; Schwilden H
Eur J Anaesthesiol; 2003 Mar; 20(3):182-90. PubMed ID: 12650488
[TBL] [Abstract][Full Text] [Related]
16. New drug, fospropofol disodium: a propofol prodrug.
Welliver M; Rugari SM
AANA J; 2009 Aug; 77(4):301-8. PubMed ID: 19731849
[TBL] [Abstract][Full Text] [Related]
17. Highly water-soluble derivatives of the anesthetic agent propofol: in vitro and in vivo evaluation of cyclic amino acid esters.
Altomare C; Trapani G; Latrofa A; Serra M; Sanna E; Biggio G; Liso G
Eur J Pharm Sci; 2003 Sep; 20(1):17-26. PubMed ID: 13678789
[TBL] [Abstract][Full Text] [Related]
18. Minimum infusion rates and recovery times from different durations of continuous infusion of fospropofol, a prodrug of propofol, in rabbits: a comparison with propofol emulsion.
Li R; Zhang WS; Liu J; Tang M; Yang YY; Luo NF
Vet Anaesth Analg; 2012 Jul; 39(4):373-84. PubMed ID: 22642486
[TBL] [Abstract][Full Text] [Related]
19. Development of water-soluble prodrugs of the HIV-1 protease inhibitor KNI-727: importance of the conversion time for higher gastrointestinal absorption of prodrugs based on spontaneous chemical cleavage.
Sohma Y; Hayashi Y; Ito T; Matsumoto H; Kimura T; Kiso Y
J Med Chem; 2003 Sep; 46(19):4124-35. PubMed ID: 12954064
[TBL] [Abstract][Full Text] [Related]
20. In vitro stability and in vivo pharmacokinetic studies of a model opioid peptide, H-Tyr-D-Ala-Gly-Phe-D-Leu-OH (DADLE), and its cyclic prodrugs.
Yang JZ; Chen W; Borchardt RT
J Pharmacol Exp Ther; 2002 Nov; 303(2):840-8. PubMed ID: 12388671
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]