194 related articles for article (PubMed ID: 24694376)
1. Synthesis and in vitro evaluation of 1,3,4-thiadiazol-2-yl urea derivatives as novel AChE inhibitors.
Xue XJ; Wang YB; Lu P; Shang HF; She JX; Xia LX; Qian H; Huang WL
Chem Pharm Bull (Tokyo); 2014; 62(6):524-7. PubMed ID: 24694376
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and biological evaluation of 1,3,4-thiadiazole analogues as novel AChE and BuChE inhibitors.
Skrzypek A; Matysiak J; Niewiadomy A; Bajda M; Szymański P
Eur J Med Chem; 2013 Apr; 62():311-9. PubMed ID: 23376249
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and anticholinesterase activities of novel 1,3,4-thiadiazole based compounds.
Skrzypek A; Matysiak J; Karpińska MM; Niewiadomy A
J Enzyme Inhib Med Chem; 2013 Aug; 28(4):816-23. PubMed ID: 22630076
[TBL] [Abstract][Full Text] [Related]
4. Potential of aryl-urea-benzofuranylthiazoles hybrids as multitasking agents in Alzheimer's disease.
Kurt BZ; Gazioglu I; Basile L; Sonmez F; Ginex T; Kucukislamoglu M; Guccione S
Eur J Med Chem; 2015 Sep; 102():80-92. PubMed ID: 26244990
[TBL] [Abstract][Full Text] [Related]
5. Exploring indole-based-thiadiazole derivatives as potent acetylcholinesterase and butyrylcholinesterase enzyme inhibitors.
Taha M; Rahim F; Uddin N; Khan IU; Iqbal N; Anouar EH; Salahuddin M; Farooq RK; Gollapalli M; Khan KM; Zafar A
Int J Biol Macromol; 2021 Oct; 188():1025-1036. PubMed ID: 34390751
[TBL] [Abstract][Full Text] [Related]
6. Antioxidant Activity, Acetylcholinesterase, and Carbonic Anhydrase Inhibitory Properties of Novel Ureas Derived from Phenethylamines.
Aksu K; Özgeriş B; Taslimi P; Naderi A; Gülçin İ; Göksu S
Arch Pharm (Weinheim); 2016 Dec; 349(12):944-954. PubMed ID: 27862205
[TBL] [Abstract][Full Text] [Related]
7. Synthesis, antioxidant and anticholinesterase activities of novel coumarylthiazole derivatives.
Kurt BZ; Gazioglu I; Sonmez F; Kucukislamoglu M
Bioorg Chem; 2015 Apr; 59():80-90. PubMed ID: 25706320
[TBL] [Abstract][Full Text] [Related]
8. Synthesis, crystal structure and biological evaluation of some novel 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazines.
Khan I; Zaib S; Ibrar A; Rama NH; Simpson J; Iqbal J
Eur J Med Chem; 2014 May; 78():167-77. PubMed ID: 24681981
[TBL] [Abstract][Full Text] [Related]
9. Design, synthesis and evaluation of new thiazole-piperazines as acetylcholinesterase inhibitors.
Yurttaş L; Kaplancıklı ZA; Özkay Y
J Enzyme Inhib Med Chem; 2013 Oct; 28(5):1040-7. PubMed ID: 22871134
[TBL] [Abstract][Full Text] [Related]
10. Active compounds from a diverse library of triazolothiadiazole and triazolothiadiazine scaffolds: synthesis, crystal structure determination, cytotoxicity, cholinesterase inhibitory activity, and binding mode analysis.
Khan I; Ibrar A; Zaib S; Ahmad S; Furtmann N; Hameed S; Simpson J; Bajorath J; Iqbal J
Bioorg Med Chem; 2014 Nov; 22(21):6163-73. PubMed ID: 25257911
[TBL] [Abstract][Full Text] [Related]
11. Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds.
Özgeriş B; Göksu S; Polat Köse L; Gülçin İ; Salmas RE; Durdagi S; Tümer F; Supuran CT
Bioorg Med Chem; 2016 May; 24(10):2318-29. PubMed ID: 27068142
[TBL] [Abstract][Full Text] [Related]
12. Design, synthesis and biological assessment of acridine derivatives containing 1,3,4-thiadiazole moiety as novel selective acetylcholinesterase inhibitors.
Lotfi S; Rahmani T; Hatami M; Pouramiri B; Kermani ET; Rezvannejad E; Mortazavi M; Fathi Hafshejani S; Askari N; Pourjamali N; Zahedifar M
Bioorg Chem; 2020 Dec; 105():104457. PubMed ID: 33339082
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and biological evaluation of tacrine-thiadiazolidinone hybrids as dual acetylcholinesterase inhibitors.
Dorronsoro I; Alonso D; Castro A; del Monte M; García-Palomero E; Martínez A
Arch Pharm (Weinheim); 2005 Jan; 338(1):18-23. PubMed ID: 15674800
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and biological evaluation of functionalized coumarins as acetylcholinesterase inhibitors.
Shen Q; Peng Q; Shao J; Liu X; Huang Z; Pu X; Ma L; Li YM; Chan AS; Gu L
Eur J Med Chem; 2005 Dec; 40(12):1307-15. PubMed ID: 16182411
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and anti-acetylcholinesterase activity of scopoletin derivatives.
Khunnawutmanotham N; Chimnoi N; Saparpakorn P; Techasakul S
Bioorg Chem; 2016 Apr; 65():137-45. PubMed ID: 26943478
[TBL] [Abstract][Full Text] [Related]
16. Synthesis, Biological Evaluation and Molecular Docking Study of Hydrazone-Containing Pyridinium Salts as Cholinesterase Inhibitors.
Parlar S; Bayraktar G; Tarikogullari AH; Alptüzün V; Erciyas E
Chem Pharm Bull (Tokyo); 2016; 64(9):1281-7. PubMed ID: 27581632
[TBL] [Abstract][Full Text] [Related]
17. Drug-1,3,4-Thiadiazole Conjugates as Novel Mixed-Type Inhibitors of Acetylcholinesterase: Synthesis, Molecular Docking, Pharmacokinetics, and ADMET Evaluation.
Ujan R; Saeed A; Channar PA; Larik FA; Abbas Q; Alajmi MF; El-Seedi HR; Rind MA; Hassan M; Raza H; Seo SY
Molecules; 2019 Feb; 24(5):. PubMed ID: 30823444
[TBL] [Abstract][Full Text] [Related]
18. Synthesis, In Vitro Biological Evaluation and In Silico Molecular Docking Studies of Indole Based Thiadiazole Derivatives as Dual Inhibitor of Acetylcholinesterase and Butyrylchloinesterase.
Khan S; Iqbal S; Taha M; Rahim F; Shah M; Ullah H; Bahadur A; Alrbyawi H; Dera AA; Alahmdi MI; Pashameah RA; Alzahrani E; Farouk AE
Molecules; 2022 Oct; 27(21):. PubMed ID: 36364195
[TBL] [Abstract][Full Text] [Related]
19. Design, synthesis and preliminary structure-activity relationship investigation of nitrogen-containing chalcone derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors: a further study based on Flavokawain B Mannich base derivatives.
Liu H; Fan H; Gao X; Huang X; Liu X; Liu L; Zhou C; Tang J; Wang Q; Liu W
J Enzyme Inhib Med Chem; 2016 Aug; 31(4):580-9. PubMed ID: 26186269
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and acetylcholinesterase inhibitory activity of Mannich base derivatives flavokawain B.
Liu HR; Huang XQ; Lou DH; Liu XJ; Liu WK; Wang QA
Bioorg Med Chem Lett; 2014 Oct; 24(19):4749-4753. PubMed ID: 25205193
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
