These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

89 related articles for article (PubMed ID: 24727279)

  • 21. 1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: structure-affinity/activity relationship at alpha1-adrenoceptor subtypes and at 5-HT1A receptors.
    Franchini S; Prandi A; Baraldi A; Sorbi C; Tait A; Buccioni M; Marucci G; Cilia A; Pirona L; Fossa P; Cichero E; Brasili L
    Eur J Med Chem; 2010 Sep; 45(9):3740-51. PubMed ID: 20605276
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Synthesis, alpha-adrenoceptors affinity and alpha 1-adrenoceptor antagonistic properties of some 1,4-substituted piperazine derivatives.
    Marona H; Kubacka M; Filipek B; Siwek A; Dybała M; Szneler E; Pociecha T; Gunia A; Waszkielewicz AM
    Pharmazie; 2011 Oct; 66(10):733-9. PubMed ID: 22026152
    [TBL] [Abstract][Full Text] [Related]  

  • 23. The possible mechanism of hypotensive activity of some pyrrolidin-2-one derivatives with antagonist properties at alpha1-adrenoceptors.
    Sapa J; Kubacka M
    Eur J Pharmacol; 2011 Dec; 673(1-3):40-8. PubMed ID: 21605554
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Quinazoline based α
    Maestri V; Tarozzi A; Simoni E; Cilia A; Poggesi E; Naldi M; Nicolini B; Pruccoli L; Rosini M; Minarini A
    Eur J Med Chem; 2017 Aug; 136():259-269. PubMed ID: 28499171
    [TBL] [Abstract][Full Text] [Related]  

  • 25. Revelation on the potency of α(1) -blockers - parallel blockade of angiotensin II receptor: a new finding.
    Yadav MR; Gandhi HP; Naik PP; Giridhar R
    Pharm Biol; 2012 Apr; 50(4):439-42. PubMed ID: 22136253
    [TBL] [Abstract][Full Text] [Related]  

  • 26. Prazosin-related compounds. Effect of transforming the piperazinylquinazoline moiety into an aminomethyltetrahydroacridine system on the affinity for alpha1-adrenoreceptors.
    Rosini M; Antonello A; Cavalli A; Bolognesi ML; Minarini A; Marucci G; Poggesi E; Leonardi A; Melchiorre C
    J Med Chem; 2003 Nov; 46(23):4895-903. PubMed ID: 14584940
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Synthesis and SAR-study for novel arylpiperazine derivatives of 5-arylidenehydantoin with α₁-adrenoceptor antagonistic properties.
    Handzlik J; Szymańska E; Wójcik R; Dela A; Jastrzębska-Więsek M; Karolak-Wojciechowska J; Fruziński A; Siwek A; Filipek B; Kieć-Kononowicz K
    Bioorg Med Chem; 2012 Jul; 20(14):4245-57. PubMed ID: 22739084
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Design and synthesis of 6,7-dimethoxyquinazoline analogs as multi-targeted ligands for α1- and AII-receptors antagonism.
    Yadav MR; Naik PP; Gandhi HP; Chauhan BS; Giridhar R
    Bioorg Med Chem Lett; 2013 Jul; 23(13):3959-66. PubMed ID: 23683590
    [TBL] [Abstract][Full Text] [Related]  

  • 29. In vitro study on the effects of some selected agonists and antagonists of alpha(1)-adrenergic receptors on the contractility of the aneurysmally-changed aortic smooth muscle in humans.
    Gnus J; Czerski A; Ferenc S; Zawadzki W; Witkiewicz W; Hauzer W; Rusiecka A; Bujok J
    J Physiol Pharmacol; 2012 Feb; 63(1):29-34. PubMed ID: 22460458
    [TBL] [Abstract][Full Text] [Related]  

  • 30. 1-Aryl-4-(4-succinimidobutyl)piperazines and their conformationally constrained analogues: synthesis, binding to serotonin (5-HT1A, 5-HT2A, 5-HT7), alpha1-adrenergic, and dopaminergic D2 receptors, and in vivo 5-HT1A functional characteristics.
    Bojarski AJ; Paluchowska MH; Duszyńska B; Kłodzińska A; Tatarczyńska E; Chojnacka-Wójcik E
    Bioorg Med Chem; 2005 Mar; 13(6):2293-303. PubMed ID: 15727878
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Synthesis and blocking activities of a new class of α₁-adrenoceptor antagonists.
    Xi BM; Ni PZ; Jiang ZZ; Wu DQ; Zhang SH; Zhang HB; Wang T; Chen WH
    Chem Biol Drug Des; 2010 Dec; 76(6):505-10. PubMed ID: 20942837
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Comparative analysis of the impact of α1-and α2-adrenoreceptor blockade on cardiac function in rats during postnatal ontogeny.
    Zefirov TL; Ziatdinova NI; Khisamieva LI; Zefirov AL
    Bull Exp Biol Med; 2011 Oct; 151(6):664-6. PubMed ID: 22485202
    [TBL] [Abstract][Full Text] [Related]  

  • 33. Synthesis, Molecular Modeling of Novel Substituted Pyridazinones and their Vasorelaxant Activities.
    Ismail MMF; Soliman DHS; Elmoniem MHA; Jaleel GAA
    Med Chem; 2021; 17(2):171-186. PubMed ID: 32216740
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Drug metabolism-based design, synthesis, and bioactivities of 1-(2,6-dimethylphenoxy)-2-(3,4-dimethoxyphenylethylamino)propane hydrochloride (DDPH) analogs as α₁-adrenoceptors antagonists.
    Xi BM; Jiang ZZ; Zou JW; Ni PZ; Chen WH
    Bioorg Med Chem; 2011 Jan; 19(2):783-8. PubMed ID: 21215646
    [TBL] [Abstract][Full Text] [Related]  

  • 35. Dexmedetomidine induces both relaxations and contractions, via different {alpha}2-adrenoceptor subtypes, in the isolated mesenteric artery and aorta of the rat.
    Wong ES; Man RY; Vanhoutte PM; Ng KF
    J Pharmacol Exp Ther; 2010 Dec; 335(3):659-64. PubMed ID: 20837990
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Identification of 3,4-dihydro-2H-thiochromene 1,1-dioxide derivatives with a phenoxyethylamine group as highly potent and selective α
    Sakauchi N; Furukawa H; Shirai J; Sato A; Kuno H; Saikawa R; Yoshida M
    Eur J Med Chem; 2017 Oct; 139():114-127. PubMed ID: 28800452
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Functional characteristics of alpha adrenergic and endothelinergic receptors in pressurized rat mesenteric veins.
    Enouri S; Monteith G; Johnson R
    Can J Physiol Pharmacol; 2013 Jul; 91(7):538-46. PubMed ID: 23826642
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Design, synthesis, and biological evaluation of prazosin-related derivatives as multipotent compounds.
    Antonello A; Hrelia P; Leonardi A; Marucci G; Rosini M; Tarozzi A; Tumiatti V; Melchiorre C
    J Med Chem; 2005 Jan; 48(1):28-31. PubMed ID: 15633998
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Pharmacophore-based design, synthesis, biological evaluation, and 3D-QSAR studies of aryl-piperazines as alpha(1)-adrenoceptor antagonists.
    Li MY; Fang H; Xia L
    Bioorg Med Chem Lett; 2005 Jul; 15(13):3216-9. PubMed ID: 15935663
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Structure-activity relationships in 1,4-benzodioxan-related compounds. 6. Role of the dioxane unit on selectivity for alpha(1)-adrenoreceptor subtypes.
    Quaglia W; Pigini M; Piergentili A; Giannella M; Marucci G; Poggesi E; Leonardi A; Melchiorre C
    J Med Chem; 1999 Jul; 42(15):2961-8. PubMed ID: 10425105
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 5.