460 related articles for article (PubMed ID: 24859458)
1. Targeting histone lysine demethylases - progress, challenges, and the future.
Thinnes CC; England KS; Kawamura A; Chowdhury R; Schofield CJ; Hopkinson RJ
Biochim Biophys Acta; 2014 Dec; 1839(12):1416-32. PubMed ID: 24859458
[TBL] [Abstract][Full Text] [Related]
2. Assessing histone demethylase inhibitors in cells: lessons learned.
Hatch SB; Yapp C; Montenegro RC; Savitsky P; Gamble V; Tumber A; Ruda GF; Bavetsias V; Fedorov O; Atrash B; Raynaud F; Lanigan R; Carmichael L; Tomlin K; Burke R; Westaway SM; Brown JA; Prinjha RK; Martinez ED; Oppermann U; Schofield CJ; Bountra C; Kawamura A; Blagg J; Brennan PE; Rossanese O; Müller S
Epigenetics Chromatin; 2017; 10():9. PubMed ID: 28265301
[TBL] [Abstract][Full Text] [Related]
3. The catalytic domains of all human KDM5 JmjC demethylases catalyse N-methyl arginine demethylation.
Bonnici J; Oueini R; Salah E; Johansson C; Schofield CJ; Kawamura A
FEBS Lett; 2023 Apr; 597(7):933-946. PubMed ID: 36700827
[TBL] [Abstract][Full Text] [Related]
4. Recent Progress in Histone Demethylase Inhibitors.
McAllister TE; England KS; Hopkinson RJ; Brennan PE; Kawamura A; Schofield CJ
J Med Chem; 2016 Feb; 59(4):1308-29. PubMed ID: 26710088
[TBL] [Abstract][Full Text] [Related]
5. Studies on the catalytic domains of multiple JmjC oxygenases using peptide substrates.
Williams ST; Walport LJ; Hopkinson RJ; Madden SK; Chowdhury R; Schofield CJ; Kawamura A
Epigenetics; 2014 Dec; 9(12):1596-603. PubMed ID: 25625844
[TBL] [Abstract][Full Text] [Related]
6. KDM1 class flavin-dependent protein lysine demethylases.
Burg JM; Link JE; Morgan BS; Heller FJ; Hargrove AE; McCafferty DG
Biopolymers; 2015 Jul; 104(4):213-46. PubMed ID: 25787087
[TBL] [Abstract][Full Text] [Related]
7. Lysine Demethylation in Pathogenesis.
Cao J; Yan Q
Adv Exp Med Biol; 2023; 1433():1-14. PubMed ID: 37751133
[TBL] [Abstract][Full Text] [Related]
8. A scintillation proximity assay for histone demethylases.
Yu W; Eram MS; Hajian T; Szykowska A; Burgess-Brown N; Vedadi M; Brown PJ
Anal Biochem; 2014 Oct; 463():54-60. PubMed ID: 25010373
[TBL] [Abstract][Full Text] [Related]
9. Structural insights into histone lysine demethylation.
Hou H; Yu H
Curr Opin Struct Biol; 2010 Dec; 20(6):739-48. PubMed ID: 20970991
[TBL] [Abstract][Full Text] [Related]
10. Emerging of lysine demethylases (KDMs): From pathophysiological insights to novel therapeutic opportunities.
Arifuzzaman S; Khatun MR; Khatun R
Biomed Pharmacother; 2020 Sep; 129():110392. PubMed ID: 32574968
[TBL] [Abstract][Full Text] [Related]
11. Lysine-241 Has a Role in Coupling 2OG Turnover with Substrate Oxidation During KDM4-Catalysed Histone Demethylation.
Hancock RL; Abboud MI; Smart TJ; Flashman E; Kawamura A; Schofield CJ; Hopkinson RJ
Chembiochem; 2018 May; 19(9):917-921. PubMed ID: 29443450
[TBL] [Abstract][Full Text] [Related]
12. Deferiprone: Pan-selective Histone Lysine Demethylase Inhibition Activity and Structure Activity Relationship Study.
Khodaverdian V; Tapadar S; MacDonald IA; Xu Y; Ho PY; Bridges A; Rajpurohit P; Sanghani BA; Fan Y; Thangaraju M; Hathaway NA; Oyelere AK
Sci Rep; 2019 Mar; 9(1):4802. PubMed ID: 30886160
[TBL] [Abstract][Full Text] [Related]
13. Recent developments in catalysis and inhibition of the Jumonji histone demethylases.
Sarah L; Fujimori DG
Curr Opin Struct Biol; 2023 Dec; 83():102707. PubMed ID: 37832177
[TBL] [Abstract][Full Text] [Related]
14. The emerging role of histone lysine demethylases in prostate cancer.
Crea F; Sun L; Mai A; Chiang YT; Farrar WL; Danesi R; Helgason CD
Mol Cancer; 2012 Aug; 11():52. PubMed ID: 22867098
[TBL] [Abstract][Full Text] [Related]
15. Arginine demethylation is catalysed by a subset of JmjC histone lysine demethylases.
Walport LJ; Hopkinson RJ; Chowdhury R; Schiller R; Ge W; Kawamura A; Schofield CJ
Nat Commun; 2016 Jun; 7():11974. PubMed ID: 27337104
[TBL] [Abstract][Full Text] [Related]
16. Targeting the LSD1/KDM1 Family of Lysine Demethylases in Cancer and Other Human Diseases.
Mao F; Shi YG
Adv Exp Med Biol; 2023; 1433():15-49. PubMed ID: 37751134
[TBL] [Abstract][Full Text] [Related]
17. Inhibitors of both the
Bonnici J; Tumber A; Kawamura A; Schofield CJ
Philos Trans R Soc Lond B Biol Sci; 2018 Jun; 373(1748):. PubMed ID: 29685975
[TBL] [Abstract][Full Text] [Related]
18. Reaction Mechanism of Histone Demethylation in αKG-dependent Non-Heme Iron Enzymes.
Singh W; Quinn D; Moody TS; Huang M
J Phys Chem B; 2019 Sep; 123(37):7801-7811. PubMed ID: 31469562
[TBL] [Abstract][Full Text] [Related]
19. Structural insight into inhibitors of flavin adenine dinucleotide-dependent lysine demethylases.
Niwa H; Umehara T
Epigenetics; 2017 May; 12(5):340-352. PubMed ID: 28277979
[TBL] [Abstract][Full Text] [Related]
20. The emerging therapeutic potential of histone methyltransferase and demethylase inhibitors.
Spannhoff A; Hauser AT; Heinke R; Sippl W; Jung M
ChemMedChem; 2009 Oct; 4(10):1568-82. PubMed ID: 19739196
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
