BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

307 related articles for article (PubMed ID: 24890564)

  • 21. The molecular biology of moenomycins: towards novel antibiotics based on inhibition of bacterial peptidoglycan glycosyltransferases.
    Ostash B; Doud E; Fedorenko V
    Biol Chem; 2010 May; 391(5):499-504. PubMed ID: 20302515
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Design and synthesis of marine natural product-based 1H-indole-2,3-dione scaffold as a new antifouling/antibacterial agent against fouling bacteria.
    Majik MS; Rodrigues C; Mascarenhas S; D'Souza L
    Bioorg Chem; 2014 Jun; 54():89-95. PubMed ID: 24875126
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Design, synthesis, antibacterial evaluation and docking study of novel 2-hydroxy-3-(nitroimidazolyl)-propyl-derived quinolone.
    Li Q; Xing J; Cheng H; Wang H; Wang J; Wang S; Zhou J; Zhang H
    Chem Biol Drug Des; 2015 Jan; 85(1):79-90. PubMed ID: 25048811
    [TBL] [Abstract][Full Text] [Related]  

  • 24. 4-alkoxy-3-arylfuran-2(5H)-ones as inhibitors of tyrosyl-tRNA synthetase: synthesis, molecular docking and antibacterial evaluation.
    Xiao ZP; Ouyang H; Wang XD; Lv PC; Huang ZJ; Yu SR; Yi TF; Yang YL; Zhu HL
    Bioorg Med Chem; 2011 Jul; 19(13):3884-91. PubMed ID: 21669535
    [TBL] [Abstract][Full Text] [Related]  

  • 25. Synthesis, antibacterial activities and molecular docking studies of Schiff bases derived from N-(2/4-benzaldehyde-amino) phenyl-N'-phenyl-thiourea.
    Zhang HJ; Qin X; Liu K; Zhu DD; Wang XM; Zhu HL
    Bioorg Med Chem; 2011 Sep; 19(18):5708-15. PubMed ID: 21872479
    [TBL] [Abstract][Full Text] [Related]  

  • 26. Discovery of (phenylureido)piperidinyl benzamides as prospective inhibitors of bacterial autolysin E from Staphylococcus aureus.
    Borišek J; Pintar S; Ogrizek M; Grdadolnik SG; Hodnik V; Turk D; Perdih A; Novič M
    J Enzyme Inhib Med Chem; 2018 Dec; 33(1):1239-1247. PubMed ID: 30141354
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Design, synthesis and antimicrobial activities of nitroimidazole derivatives containing 1,3,4-oxadiazole scaffold as FabH inhibitors.
    Li Y; Luo Y; Hu Y; Zhu DD; Zhang S; Liu ZJ; Gong HB; Zhu HL
    Bioorg Med Chem; 2012 Jul; 20(14):4316-22. PubMed ID: 22710102
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Discovery of 4-Pyridone derivatives as specific inhibitors of enoyl-acyl carrier protein reductase (FabI) with antibacterial activity against Staphylococcus aureus.
    Takahata S; Iida M; Yoshida T; Kumura K; Kitagawa H; Hoshiko S
    J Antibiot (Tokyo); 2007 Feb; 60(2):123-8. PubMed ID: 17420562
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Positive cooperativity between acceptor and donor sites of the peptidoglycan glycosyltransferase.
    Bury D; Dahmane I; Derouaux A; Dumbre S; Herdewijn P; Matagne A; Breukink E; Mueller-Seitz E; Petz M; Terrak M
    Biochem Pharmacol; 2015 Jan; 93(2):141-50. PubMed ID: 25462814
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Scaffold hopping-guided design of some isatin based rigid analogs as fatty acid amide hydrolase inhibitors: Synthesis and evaluation.
    Jaiswal S; Tripathi RKP; Ayyannan SR
    Biomed Pharmacother; 2018 Nov; 107():1611-1623. PubMed ID: 30257379
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Design, synthesis and molecular docking of salicylic acid derivatives containing metronidazole as a new class of antimicrobial agents.
    Guo ZH; Yin Y; Wang C; Wang PF; Zhang XT; Wang ZC; Zhu HL
    Bioorg Med Chem; 2015 Sep; 23(18):6148-56. PubMed ID: 26304108
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Design, synthesis and antibacterial activities of 5-(pyrazin-2-yl)-4H-1,2,4-triazole-3-thiol derivatives containing Schiff base formation as FabH inhibitory.
    Zhang F; Wen Q; Wang SF; Shahla Karim B; Yang YS; Liu JJ; Zhang WM; Zhu HL
    Bioorg Med Chem Lett; 2014 Jan; 24(1):90-5. PubMed ID: 24332628
    [TBL] [Abstract][Full Text] [Related]  

  • 33. A new efficient route to 7-aryl-6-fluoro-8-nitroquinolones as potent antibacterial agents.
    Al-Trawneh SA; El-Abadelah MM; Al-Abadleh MM; Zani F; Incerti M; Vicini P
    Eur J Med Chem; 2014 Oct; 86():364-7. PubMed ID: 25180924
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Discovery of diethyl 2,5-diaminothiophene-3,4-dicarboxylate derivatives as potent anticancer and antimicrobial agents and screening of anti-diabetic activity: synthesis and in vitro biological evaluation. Part 1.
    Bozorov K; Ma HR; Zhao JY; Zhao HQ; Chen H; Bobakulov K; Xin XL; Elmuradov B; Shakhidoyatov K; Aisa HA
    Eur J Med Chem; 2014 Sep; 84():739-45. PubMed ID: 25064350
    [TBL] [Abstract][Full Text] [Related]  

  • 35. Identification of a new class of FtsZ inhibitors by structure-based design and in vitro screening.
    Chan FY; Sun N; Neves MA; Lam PC; Chung WH; Wong LK; Chow HY; Ma DL; Chan PH; Leung YC; Chan TH; Abagyan R; Wong KY
    J Chem Inf Model; 2013 Aug; 53(8):2131-40. PubMed ID: 23848971
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Discovery of novel bacterial FabH inhibitors (Pyrazol-Benzimidazole amide derivatives): Design, synthesis, bioassay, molecular docking and crystal structure determination.
    Wang YT; Shi TQ; Fu J; Zhu HL
    Eur J Med Chem; 2019 Jun; 171():209-220. PubMed ID: 30925337
    [TBL] [Abstract][Full Text] [Related]  

  • 37. A combine approach of chemical synthesis, biological evaluation and structural dynamics studies revealed thiazole substituted arylamine derivatives as potent FabH enzyme inhibitors.
    Ahmad H; Ahmad F; Parveen S; Ahmad S; Azam SS; Hassan A
    Bioorg Chem; 2020 Dec; 105():104426. PubMed ID: 33161255
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Synthesis and antimicrobial activity of N-Mannich bases of 3-[N'-sulphadoximino] isatin and its methyl derivative.
    Surendra ; Pandeya N; Yogeeswari P; Ram DS; Nath G
    Boll Chim Farm; 1998 Sep; 137(8):321-4. PubMed ID: 9835147
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Synthesis and biological evaluation of N-acylhydrazones as inhibitors of MurC and MurD ligases.
    Sink R; Kovac A; Tomasić T; Rupnik V; Boniface A; Bostock J; Chopra I; Blanot D; Masic LP; Gobec S; Zega A
    ChemMedChem; 2008 Sep; 3(9):1362-70. PubMed ID: 18651694
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Structural analysis of the contacts anchoring moenomycin to peptidoglycan glycosyltransferases and implications for antibiotic design.
    Yuan Y; Fuse S; Ostash B; Sliz P; Kahne D; Walker S
    ACS Chem Biol; 2008 Jul; 3(7):429-36. PubMed ID: 18642800
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 16.