These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
155 related articles for article (PubMed ID: 24973695)
1. Positive allosteric modulation of the GHB high-affinity binding site by the GABAA receptor modulator monastrol and the flavonoid catechin. Eghorn LF; Hoestgaard-Jensen K; Kongstad KT; Bay T; Higgins D; Frølund B; Wellendorph P Eur J Pharmacol; 2014 Oct; 740():570-7. PubMed ID: 24973695 [TBL] [Abstract][Full Text] [Related]
2. Monastrol, a 3,4-dihydropyrimidin-2(1H)-thione, as structural scaffold for the development of modulators for GHB high-affinity binding sites and α Damgaard M; Al-Khawaja A; Nittegaard-Nielsen M; Petersen RF; Wellendorph P; Frølund B Eur J Med Chem; 2017 Sep; 138():300-312. PubMed ID: 28683403 [TBL] [Abstract][Full Text] [Related]
3. GHB receptor targets in the CNS: focus on high-affinity binding sites. Bay T; Eghorn LF; Klein AB; Wellendorph P Biochem Pharmacol; 2014 Jan; 87(2):220-8. PubMed ID: 24269284 [TBL] [Abstract][Full Text] [Related]
4. α4βδ GABA(A) receptors are high-affinity targets for γ-hydroxybutyric acid (GHB). Absalom N; Eghorn LF; Villumsen IS; Karim N; Bay T; Olsen JV; Knudsen GM; Bräuner-Osborne H; Frølund B; Clausen RP; Chebib M; Wellendorph P Proc Natl Acad Sci U S A; 2012 Aug; 109(33):13404-9. PubMed ID: 22753476 [TBL] [Abstract][Full Text] [Related]
6. Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site. Middendorp SJ; Maldifassi MC; Baur R; Sigel E Neuropharmacology; 2015 Aug; 95():459-67. PubMed ID: 25963418 [TBL] [Abstract][Full Text] [Related]
7. Autoradiographic imaging and quantification of the high-affinity GHB binding sites in rodent brain using Klein AB; Bay T; Villumsen IS; Falk-Petersen CB; Marek A; Frølund B; Clausen RP; Hansen HD; Knudsen GM; Wellendorph P Neurochem Int; 2016 Nov; 100():138-145. PubMed ID: 27615059 [TBL] [Abstract][Full Text] [Related]
8. Selective gamma-hydroxybutyric acid receptor ligands increase extracellular glutamate in the hippocampus, but fail to activate G protein and to produce the sedative/hypnotic effect of gamma-hydroxybutyric acid. Castelli MP; Ferraro L; Mocci I; Carta F; Carai MA; Antonelli T; Tanganelli S; Cignarella G; Gessa GL J Neurochem; 2003 Nov; 87(3):722-32. PubMed ID: 14535954 [TBL] [Abstract][Full Text] [Related]
9. Novel cyclic gamma-hydroxybutyrate (GHB) analogs with high affinity and stereoselectivity of binding to GHB sites in rat brain. Wellendorph P; Høg S; Greenwood JR; de Lichtenberg A; Nielsen B; Frølund B; Brehm L; Clausen RP; Bräuner-Osborne H J Pharmacol Exp Ther; 2005 Oct; 315(1):346-51. PubMed ID: 16014570 [TBL] [Abstract][Full Text] [Related]
10. Validation of high-affinity binding sites for succinic acid through distinguishable binding of gamma-hydroxybutyric acid receptor-specific NCS 382 antipodes. Molnár T; Visy J; Simon A; Moldvai I; Temesvári-Major E; Dörnyei G; Fekete EK; Kardos J Bioorg Med Chem Lett; 2008 Dec; 18(23):6290-2. PubMed ID: 18945616 [TBL] [Abstract][Full Text] [Related]
11. Pharmacology of the human gamma-aminobutyric acidA receptor alpha 4 subunit expressed in Xenopus laevis oocytes. Whittemore ER; Yang W; Drewe JA; Woodward RM Mol Pharmacol; 1996 Nov; 50(5):1364-75. PubMed ID: 8913369 [TBL] [Abstract][Full Text] [Related]
12. Novel high-affinity and selective biaromatic 4-substituted gamma-hydroxybutyric acid (GHB) analogues as GHB ligands: design, synthesis, and binding studies. Høg S; Wellendorph P; Nielsen B; Frydenvang K; Dahl IF; Bräuner-Osborne H; Brehm L; Frølund B; Clausen RP J Med Chem; 2008 Dec; 51(24):8088-95. PubMed ID: 19053823 [TBL] [Abstract][Full Text] [Related]
13. Phenylacetic acids and the structurally related non-steroidal anti-inflammatory drug diclofenac bind to specific gamma-hydroxybutyric acid sites in rat brain. Wellendorph P; Høg S; Skonberg C; Bräuner-Osborne H Fundam Clin Pharmacol; 2009 Apr; 23(2):207-13. PubMed ID: 19645815 [TBL] [Abstract][Full Text] [Related]
14. A review of pharmacology of NCS-382, a putative antagonist of gamma-hydroxybutyric acid (GHB) receptor. Castelli MP; Pibiri F; Carboni G; Piras AP CNS Drug Rev; 2004; 10(3):243-60. PubMed ID: 15492774 [TBL] [Abstract][Full Text] [Related]
15. Dihydropyrimidinone positive modulation of delta-subunit-containing gamma-aminobutyric acid type A receptors, including an epilepsy-linked mutant variant. Lewis RW; Mabry J; Polisar JG; Eagen KP; Ganem B; Hess GP Biochemistry; 2010 Jun; 49(23):4841-51. PubMed ID: 20450160 [TBL] [Abstract][Full Text] [Related]
16. Endogenous gamma-aminobutyric acid (GABA)(A) receptor active neurosteroids and the sedative/hypnotic action of gamma-hydroxybutyric acid (GHB): a study in GHB-S (sensitive) and GHB-R (resistant) rat lines. Barbaccia ML; Carai MA; Colombo G; Lobina C; Purdy RH; Gessa GL Neuropharmacology; 2005 Jul; 49(1):48-58. PubMed ID: 15992580 [TBL] [Abstract][Full Text] [Related]
17. The interaction of general anaesthetics with recombinant GABAA and glycine receptors expressed in Xenopus laevis oocytes: a comparative study. Pistis M; Belelli D; Peters JA; Lambert JJ Br J Pharmacol; 1997 Dec; 122(8):1707-19. PubMed ID: 9422818 [TBL] [Abstract][Full Text] [Related]
18. Characterization and pharmacology of the GHB receptor. Ticku MK; Mehta AK Ann N Y Acad Sci; 2008 Oct; 1139():374-85. PubMed ID: 18991884 [TBL] [Abstract][Full Text] [Related]
19. The γ-hydroxybutyric acid (GHB) analogue NCS-382 is a substrate for both monocarboxylate transporters subtypes 1 and 4. Thiesen L; Belew ZM; Griem-Krey N; Pedersen SF; Crocoll C; Nour-Eldin HH; Wellendorph P Eur J Pharm Sci; 2020 Feb; 143():105203. PubMed ID: 31866563 [TBL] [Abstract][Full Text] [Related]
20. Gamma-hydroxybutyric acid (GHB) and the mesoaccumbens reward circuit: evidence for GABA(B) receptor-mediated effects. Pistis M; Muntoni AL; Pillolla G; Perra S; Cignarella G; Melis M; Gessa GL Neuroscience; 2005; 131(2):465-74. PubMed ID: 15708487 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]