315 related articles for article (PubMed ID: 24986232)
1. Synthesis and structure-activity relationship of thiobarbituric acid derivatives as potent inhibitors of urease.
Khan KM; Rahim F; Khan A; Shabeer M; Hussain S; Rehman W; Taha M; Khan M; Perveen S; Choudhary MI
Bioorg Med Chem; 2014 Aug; 22(15):4119-23. PubMed ID: 24986232
[TBL] [Abstract][Full Text] [Related]
2. Design and synthesis of new barbituric- and thiobarbituric acid derivatives as potent urease inhibitors: Structure activity relationship and molecular modeling studies.
Rauf A; Shahzad S; Bajda M; Yar M; Ahmed F; Hussain N; Akhtar MN; Khan A; Jończyk J
Bioorg Med Chem; 2015 Sep; 23(17):6049-58. PubMed ID: 26081763
[TBL] [Abstract][Full Text] [Related]
3. Synthesis of 4-thiazolidinone analogs as potent in vitro anti-urease agents.
Rahim F; Zaman K; Ullah H; Taha M; Wadood A; Javed MT; Rehman W; Ashraf M; Uddin R; Uddin I; Asghar H; Khan AA; Khan KM
Bioorg Chem; 2015 Dec; 63():123-31. PubMed ID: 26520885
[TBL] [Abstract][Full Text] [Related]
4. Novel thiobarbiturates as potent urease inhibitors with potential antibacterial activity: Design, synthesis, radiolabeling and biodistribution study.
Abdulwahab HG; Harras MF; El Menofy NG; Hegab AM; Essa BM; Selim AA; Sakr TM; El-Zahabi HSA
Bioorg Med Chem; 2020 Dec; 28(23):115759. PubMed ID: 32992246
[TBL] [Abstract][Full Text] [Related]
5. Synthesis, in vitro urease inhibitory activity, and molecular docking studies of thiourea and urea derivatives.
Bano B; Kanwal ; Khan KM; Lodhi A; Salar U; Begum F; Ali M; Taha M; Perveen S
Bioorg Chem; 2018 Oct; 80():129-144. PubMed ID: 29913313
[TBL] [Abstract][Full Text] [Related]
6. Hybrid benzothiazole analogs as antiurease agent: Synthesis and molecular docking studies.
Taha M; Ismail NH; Imran S; Wadood A; Rahim F; Khan KM; Riaz M
Bioorg Chem; 2016 Jun; 66():80-7. PubMed ID: 27038849
[TBL] [Abstract][Full Text] [Related]
7. Synthesis of 2-acylated and sulfonated 4-hydroxycoumarins: In vitro urease inhibition and molecular docking studies.
Rashid U; Rahim F; Taha M; Arshad M; Ullah H; Mahmood T; Ali M
Bioorg Chem; 2016 Jun; 66():111-6. PubMed ID: 27140727
[TBL] [Abstract][Full Text] [Related]
8. Synthesis of potent urease inhibitors based on disulfide scaffold and their molecular docking studies.
Taha M; Ismail NH; Imran S; Wadood A; Rahim F; Riaz M
Bioorg Med Chem; 2015 Nov; 23(22):7211-8. PubMed ID: 26507431
[TBL] [Abstract][Full Text] [Related]
9. 1-[(4'-Chlorophenyl) carbonyl-4-(aryl) thiosemicarbazide derivatives as potent urease inhibitors: Synthesis, in vitro and in silico studies.
Ali B; Khan KM; Salar U; Kanwal ; Hussain S; Ashraf M; Riaz M; Wadood A; Taha M; Perveen S
Bioorg Chem; 2018 Sep; 79():363-371. PubMed ID: 29859384
[TBL] [Abstract][Full Text] [Related]
10. Syntheses of 4,6-dihydroxypyrimidine diones, their urease inhibition, in vitro, in silico, and kinetic studies.
Muhammad MT; Khan KM; Arshia ; Khan A; Arshad F; Fatima B; Choudhary MI; Syed N; Moin ST
Bioorg Chem; 2017 Dec; 75():317-331. PubMed ID: 29080496
[TBL] [Abstract][Full Text] [Related]
11. New barbiturates and thiobarbiturates as potential enzyme inhibitors.
Qureshi AM; Mumtaz S; Rauf A; Ashraf M; Nasar R; Chohan ZH
J Enzyme Inhib Med Chem; 2015 Feb; 30(1):119-25. PubMed ID: 24666295
[TBL] [Abstract][Full Text] [Related]
12. Synthesis, biological evaluation and molecular docking of N-phenyl thiosemicarbazones as urease inhibitors.
Hameed A; Khan KM; Zehra ST; Ahmed R; Shafiq Z; Bakht SM; Yaqub M; Hussain M; de la Vega de León A; Furtmann N; Bajorath J; Shad HA; Tahir MN; Iqbal J
Bioorg Chem; 2015 Aug; 61():51-7. PubMed ID: 26119990
[TBL] [Abstract][Full Text] [Related]
13. Bisindolylmethane thiosemicarbazides as potential inhibitors of urease: Synthesis and molecular modeling studies.
Taha M; Ullah H; Al Muqarrabun LMR; Khan MN; Rahim F; Ahmat N; Javid MT; Ali M; Khan KM
Bioorg Med Chem; 2018 Jan; 26(1):152-160. PubMed ID: 29183662
[TBL] [Abstract][Full Text] [Related]
14. New 1,2,3-triazole-(thio)barbituric acid hybrids as urease inhibitors: Design, synthesis, in vitro urease inhibition, docking study, and molecular dynamic simulation.
Asgari MS; Azizian H; Nazari Montazer M; Mohammadi-Khanaposhtani M; Asadi M; Sepehri S; Ranjbar PR; Rahimi R; Biglar M; Larijani B; Amanlou M; Mahdavi M
Arch Pharm (Weinheim); 2020 Sep; 353(9):e2000023. PubMed ID: 32596826
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis, molecular docking studies and in vitro screening of ethyl 4-(3-benzoylthioureido) benzoates as urease inhibitors.
Saeed A; Khan MS; Rafique H; Shahid M; Iqbal J
Bioorg Chem; 2014 Feb; 52():1-7. PubMed ID: 24269986
[TBL] [Abstract][Full Text] [Related]
16. Syntheses, in vitro urease inhibitory activities of urea and thiourea derivatives of tryptamine, their molecular docking and cytotoxic studies.
Kanwal ; Khan M; Arshia ; Khan KM; Parveen S; Shaikh M; Fatima N; Choudhary MI
Bioorg Chem; 2019 Mar; 83():595-610. PubMed ID: 30513472
[TBL] [Abstract][Full Text] [Related]
17. Benzylidine indane-1,3-diones: As novel urease inhibitors; synthesis, in vitro, and in silico studies.
Bano B; Kanwal ; Khan KM; Begum F; Lodhi MA; Salar U; Khalil R; Ul-Haq Z; Perveen S
Bioorg Chem; 2018 Dec; 81():658-671. PubMed ID: 30253339
[TBL] [Abstract][Full Text] [Related]
18. Synthesis, biological assay in vitro and molecular docking studies of new Schiff base derivatives as potential urease inhibitors.
Aslam MA; Mahmood SU; Shahid M; Saeed A; Iqbal J
Eur J Med Chem; 2011 Nov; 46(11):5473-9. PubMed ID: 21981981
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and in vitro urease inhibitory activity of N,N'-disubstituted thioureas.
Khan KM; Naz F; Taha M; Khan A; Perveen S; Choudhary MI; Voelter W
Eur J Med Chem; 2014 Mar; 74():314-23. PubMed ID: 24486414
[TBL] [Abstract][Full Text] [Related]
20. A facile one-pot synthesis of 2-arylamino-5-aryloxylalkyl-1,3,4-oxadiazoles and their urease inhibition studies.
Akhtar T; Khan MA; Iqbal J; Jones PG; Hameed S
Chem Biol Drug Des; 2014 Jul; 84(1):92-8. PubMed ID: 24495281
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]