BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

137 related articles for article (PubMed ID: 25059502)

  • 1. Cyclic acyl guanidines bearing carbamate moieties allow potent and dirigible cholinesterase inhibition of either acetyl- or butyrylcholinesterase.
    Darras FH; Kling B; Sawatzky E; Heilmann J; Decker M
    Bioorg Med Chem; 2014 Sep; 22(17):5020-34. PubMed ID: 25059502
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation.
    Belluti F; Rampa A; Piazzi L; Bisi A; Gobbi S; Bartolini M; Andrisano V; Cavalli A; Recanatini M; Valenti P
    J Med Chem; 2005 Jun; 48(13):4444-56. PubMed ID: 15974596
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Acetylcholinesterase inhibitors: synthesis and structure-activity relationships of omega-[N-methyl-N-(3-alkylcarbamoyloxyphenyl)- methyl]aminoalkoxyheteroaryl derivatives.
    Rampa A; Bisi A; Valenti P; Recanatini M; Cavalli A; Andrisano V; Cavrini V; Fin L; Buriani A; Giusti P
    J Med Chem; 1998 Oct; 41(21):3976-86. PubMed ID: 9767635
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis of novel phenserine-based-selective inhibitors of butyrylcholinesterase for Alzheimer's disease.
    Yu Q; Holloway HW; Utsuki T; Brossi A; Greig NH
    J Med Chem; 1999 May; 42(10):1855-61. PubMed ID: 10346939
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Methyl analogues of the experimental Alzheimer drug phenserine: synthesis and structure/activity relationships for acetyl- and butyrylcholinesterase inhibitory action.
    Yu Q; Holloway HW; Flippen-Anderson JL; Hoffman B; Brossi A; Greig NH
    J Med Chem; 2001 Nov; 44(24):4062-71. PubMed ID: 11708910
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Novel anticholinesterases based on the molecular skeletons of furobenzofuran and methanobenzodioxepine.
    Luo W; Yu QS; Zhan M; Parrish D; Deschamps JR; Kulkarni SS; Holloway HW; Alley GM; Lahiri DK; Brossi A; Greig NH
    J Med Chem; 2005 Feb; 48(4):986-94. PubMed ID: 15715468
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design and synthesis of N-benzylpiperidine-purine derivatives as new dual inhibitors of acetyl- and butyrylcholinesterase.
    Rodríguez-Franco MI; Fernández-Bachiller MI; Pérez C; Castro A; Martínez A
    Bioorg Med Chem; 2005 Dec; 13(24):6795-802. PubMed ID: 16183292
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues.
    Bolognesi ML; Bartolini M; Cavalli A; Andrisano V; Rosini M; Minarini A; Melchiorre C
    J Med Chem; 2004 Nov; 47(24):5945-52. PubMed ID: 15537349
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Carbamate analogues of (-)-physostigmine: in vitro inhibition of acetyl- and butyrylcholinesterase.
    Yu QS; Atack JR; Rapoport SI; Brossi A
    FEBS Lett; 1988 Jul; 234(1):127-30. PubMed ID: 3391264
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Ortho effects for inhibition mechanisms of butyrylcholinesterase by o-substituted phenyl N-butyl carbamates and comparison with acetylcholinesterase, cholesterol esterase, and lipase.
    Lin G; Lee YR; Liu YC; Wu YG
    Chem Res Toxicol; 2005 Jul; 18(7):1124-31. PubMed ID: 16022504
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Syntheses and anticholinesterase activities of (3aS)-N1, N8-bisnorphenserine, (3aS)-N1,N8-bisnorphysostigmine, their antipodal isomers, and other potential metabolites of phenserine.
    Yu Q; Greig NH; Holloway HW; Brossi A
    J Med Chem; 1998 Jun; 41(13):2371-9. PubMed ID: 9632370
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Cholinesterase inhibition by derivatives of 2-amino-4,6-dimethylpyridine.
    Debord J; N'Diaye P; Bollinger JC; Fikri K; Penicaut B; Robert JM; Robert-Piessard S; Le Baut G
    J Enzyme Inhib; 1997 Apr; 12(1):13-26. PubMed ID: 9204379
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Cholinesterase inhibitors proposed for treating dementia in Alzheimer's disease: selectivity toward human brain acetylcholinesterase compared with butyrylcholinesterase.
    Pacheco G; Palacios-Esquivel R; Moss DE
    J Pharmacol Exp Ther; 1995 Aug; 274(2):767-70. PubMed ID: 7636741
    [TBL] [Abstract][Full Text] [Related]  

  • 14. N-methylated diazabicyclo[3.2.2]nonane substituted triterpenoic acids are excellent, hyperbolic and selective inhibitors for butyrylcholinesterase.
    Heise N; Friedrich S; Temml V; Schuster D; Siewert B; Csuk R
    Eur J Med Chem; 2022 Jan; 227():113947. PubMed ID: 34731766
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Cage amines as the stopper inhibitors of cholinesterases.
    Lin G; Tsai HJ; Tsai YH
    Bioorg Med Chem Lett; 2003 Sep; 13(17):2887-90. PubMed ID: 14611850
    [TBL] [Abstract][Full Text] [Related]  

  • 16. SAR-mediated Similarity Assessment of the Property Profile for New, Silicon-Based AChE/BChE Inhibitors.
    Bak A; Pizova H; Kozik V; Vorcakova K; Kos J; Treml J; Odehnalova K; Oravec M; Imramovsky A; Bobal P; Smolinski A; Trávníček Z; Jampilek J
    Int J Mol Sci; 2019 Oct; 20(21):. PubMed ID: 31671776
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Acetylcholinesterase inhibitors: SAR and kinetic studies on omega-[N-methyl-N-(3-alkylcarbamoyloxyphenyl)methyl]aminoalkoxyaryl derivatives.
    Rampa A; Piazzi L; Belluti F; Gobbi S; Bisi A; Bartolini M; Andrisano V; Cavrini V; Cavalli A; Recanatini M; Valenti P
    J Med Chem; 2001 Nov; 44(23):3810-20. PubMed ID: 11689067
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Molecular recognition by acetylcholinesterase at the peripheral anionic site: structure-activity relationships for inhibitions by aryl carbamates.
    Lin G; Lai CY; Liao WC
    Bioorg Med Chem; 1999 Dec; 7(12):2683-9. PubMed ID: 10658572
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Amino acid residues involved in the interaction of acetylcholinesterase and butyrylcholinesterase with the carbamates Ro 02-0683 and bambuterol, and with terbutaline.
    Kovarik Z; Radić Z; Grgas B; Skrinjarić-Spoljar M; Reiner E; Simeon-Rudolf V
    Biochim Biophys Acta; 1999 Aug; 1433(1-2):261-71. PubMed ID: 10446376
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Acetyl- and butyryl-cholinesterase inhibitory activities of the edible brown alga Eisenia bicyclis.
    Choi JS; Haulader S; Karki S; Jung HJ; Kim HR; Jung HA
    Arch Pharm Res; 2015 Aug; 38(8):1477-87. PubMed ID: 25370610
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.