These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

365 related articles for article (PubMed ID: 25124112)

  • 1. Synthesis and biological evaluation of novel thiadiazole amides as potent Cdc25B and PTP1B inhibitors.
    Li Y; Yu Y; Jin K; Gao L; Luo T; Sheng L; Shao X; Li J
    Bioorg Med Chem Lett; 2014 Sep; 24(17):4125-8. PubMed ID: 25124112
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors.
    Wang WL; Huang C; Gao LX; Tang CL; Wang JQ; Wu MC; Sheng L; Chen HJ; Nan FJ; Li JY; Li J; Feng B
    Bioorg Med Chem Lett; 2014 Apr; 24(8):1889-94. PubMed ID: 24684845
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Design and synthesis of new potent PTP1B inhibitors with the skeleton of 2-substituted imino-3-substituted-5-heteroarylidene-1,3-thiazolidine-4-one: Part I.
    Meng G; Zheng M; Wang M; Tong J; Ge W; Zhang J; Zheng A; Li J; Gao L; Li J
    Eur J Med Chem; 2016 Oct; 122():756-769. PubMed ID: 27526040
    [TBL] [Abstract][Full Text] [Related]  

  • 4. [Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].
    Du X; Zhang SE; Liu JZ; Nie FL; Ye F; Tian JY; Xiao ZY
    Yao Xue Xue Bao; 2012 Mar; 47(3):367-73. PubMed ID: 22645761
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Benzo[c][1,2,5]thiadiazole derivatives: A new class of potent Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors.
    Wang WL; Chen XY; Gao Y; Gao LX; Sheng L; Zhu J; Xu L; Ding ZZ; Zhang C; Li JY; Li J; Zhou YB
    Bioorg Med Chem Lett; 2017 Dec; 27(23):5154-5157. PubMed ID: 29100798
    [TBL] [Abstract][Full Text] [Related]  

  • 6. 2,4-Dihydroxychalcone derivatives as novel potent cell division cycle 25B phosphatase inhibitors and protein tyrosine phosphatase 1B inhibitors.
    Xie C; Sun Y; Pan CY; Tang LM; Guan LP
    Pharmazie; 2014 Apr; 69(4):257-62. PubMed ID: 24791588
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and evaluation of several oleanolic acid glycoconjugates as protein tyrosine phosphatase 1B inhibitors.
    Liu Q; Guo T; Li D; Li F; Li W
    Eur J Med Chem; 2014 May; 79():34-46. PubMed ID: 24721313
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and biological evaluation of novel N-aryl-ω-(benzoazol-2-yl)-sulfanylalkanamides as dual inhibitors of α-glucosidase and protein tyrosine phosphatase 1B.
    Wang MY; Cheng XC; Chen XB; Li Y; Zang LL; Duan YQ; Chen MZ; Yu P; Sun H; Wang RL
    Chem Biol Drug Des; 2018 Sep; 92(3):1647-1656. PubMed ID: 29745030
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B.
    Li XQ; Xu Q; Luo J; Wang LJ; Jiang B; Zhang RS; Shi DY
    Eur J Med Chem; 2017 Aug; 136():348-359. PubMed ID: 28511130
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Peptidomimetics as potent and selective PTP1B inhibitors.
    Patel D; Jain M; Shah SR; Bahekar R; Jadav P; Shah K; Joharapurkar A; Shaikh M; Sairam KV
    Med Chem; 2013 Aug; 9(5):660-71. PubMed ID: 23030658
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Facile fabrication of promising protein tyrosine phosphatase (PTP) inhibitor entities based on 'clicked' serine/threonine-monosaccharide hybrids.
    He XP; Deng Q; Gao LX; Li C; Zhang W; Zhou YB; Tang Y; Shi XX; Xie J; Li J; Chen GR; Chen K
    Bioorg Med Chem; 2011 Jul; 19(13):3892-900. PubMed ID: 21665482
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and biological evaluation of oleanolic acid derivatives as PTP1B inhibitors.
    Liu QC; Guo TT; Zhang L; Yu Y; Wang P; Yang JF; Li YX
    Eur J Med Chem; 2013 May; 63():511-22. PubMed ID: 23531458
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and characterization of 5,7-dihydroxyflavanone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
    Sun LP; Ma WP; Gao LX; Yang LL; Quan YC; Li J; Piao HR
    J Enzyme Inhib Med Chem; 2013 Dec; 28(6):1199-204. PubMed ID: 23009604
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis, characterization and biological evaluation of thiadiazole amide derivatives as nucleoside triphosphate diphosphohydrolases (NTPDases) inhibitors.
    Abbas S; Afzal S; Nadeem H; Hussain D; Langer P; Sévigny J; Ashraf Z; Iqbal J
    Bioorg Chem; 2022 Jan; 118():105456. PubMed ID: 34800887
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Design, synthesis and docking study of 5-(substituted benzylidene)thiazolidine-2,4-dione derivatives as inhibitors of protein tyrosine phosphatase 1B.
    Wang Z; Liu Z; Lee W; Kim SN; Yoon G; Cheon SH
    Bioorg Med Chem Lett; 2014 Aug; 24(15):3337-40. PubMed ID: 24953600
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of miltirone analogues as inhibitors of Cdc25 phosphatases.
    Huang W; Li J; Zhang W; Zhou Y; Xie C; Luo Y; Li Y; Wang J; Li J; Lu W
    Bioorg Med Chem Lett; 2006 Apr; 16(7):1905-8. PubMed ID: 16434190
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and biological evaluation of tryptophan-derived rhodanine derivatives as PTP1B inhibitors and anti-bacterial agents.
    Liu H; Sun D; Du H; Zheng C; Li J; Piao H; Li J; Sun L
    Eur J Med Chem; 2019 Jun; 172():163-173. PubMed ID: 30978561
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design and synthesis of novel 1,2-dithiolan-4-yl benzoate derivatives as PTP1B inhibitors.
    Chen J; Gao LX; Gong JX; Jiang CS; Yao LG; Li JY; Li J; Xiao W; Guo YW
    Bioorg Med Chem Lett; 2015; 25(10):2211-6. PubMed ID: 25872983
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Design and synthesis of novel bis-thiazolone derivatives as micromolar CDC25 phosphatase inhibitors: effect of dimerisation on phosphatase inhibition.
    Sarkis M; Tran DN; Kolb S; Miteva MA; Villoutreix BO; Garbay C; Braud E
    Bioorg Med Chem Lett; 2012 Dec; 22(24):7345-50. PubMed ID: 23141909
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Toward a treatment of diabesity: Rational design, synthesis and biological evaluation of benzene-sulfonamide derivatives as a new class of PTP-1B inhibitors.
    Ghareb N; El-Sayed NM; Abdelhameed R; Yamada K; Elgawish MS
    Bioorg Chem; 2019 May; 86():322-338. PubMed ID: 30743173
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 19.