362 related articles for article (PubMed ID: 25124112)
1. Synthesis and biological evaluation of novel thiadiazole amides as potent Cdc25B and PTP1B inhibitors.
Li Y; Yu Y; Jin K; Gao L; Luo T; Sheng L; Shao X; Li J
Bioorg Med Chem Lett; 2014 Sep; 24(17):4125-8. PubMed ID: 25124112
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors.
Wang WL; Huang C; Gao LX; Tang CL; Wang JQ; Wu MC; Sheng L; Chen HJ; Nan FJ; Li JY; Li J; Feng B
Bioorg Med Chem Lett; 2014 Apr; 24(8):1889-94. PubMed ID: 24684845
[TBL] [Abstract][Full Text] [Related]
3. Design and synthesis of new potent PTP1B inhibitors with the skeleton of 2-substituted imino-3-substituted-5-heteroarylidene-1,3-thiazolidine-4-one: Part I.
Meng G; Zheng M; Wang M; Tong J; Ge W; Zhang J; Zheng A; Li J; Gao L; Li J
Eur J Med Chem; 2016 Oct; 122():756-769. PubMed ID: 27526040
[TBL] [Abstract][Full Text] [Related]
4. [Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].
Du X; Zhang SE; Liu JZ; Nie FL; Ye F; Tian JY; Xiao ZY
Yao Xue Xue Bao; 2012 Mar; 47(3):367-73. PubMed ID: 22645761
[TBL] [Abstract][Full Text] [Related]
5. Benzo[c][1,2,5]thiadiazole derivatives: A new class of potent Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors.
Wang WL; Chen XY; Gao Y; Gao LX; Sheng L; Zhu J; Xu L; Ding ZZ; Zhang C; Li JY; Li J; Zhou YB
Bioorg Med Chem Lett; 2017 Dec; 27(23):5154-5157. PubMed ID: 29100798
[TBL] [Abstract][Full Text] [Related]
6. 2,4-Dihydroxychalcone derivatives as novel potent cell division cycle 25B phosphatase inhibitors and protein tyrosine phosphatase 1B inhibitors.
Xie C; Sun Y; Pan CY; Tang LM; Guan LP
Pharmazie; 2014 Apr; 69(4):257-62. PubMed ID: 24791588
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and evaluation of several oleanolic acid glycoconjugates as protein tyrosine phosphatase 1B inhibitors.
Liu Q; Guo T; Li D; Li F; Li W
Eur J Med Chem; 2014 May; 79():34-46. PubMed ID: 24721313
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and biological evaluation of novel N-aryl-ω-(benzoazol-2-yl)-sulfanylalkanamides as dual inhibitors of α-glucosidase and protein tyrosine phosphatase 1B.
Wang MY; Cheng XC; Chen XB; Li Y; Zang LL; Duan YQ; Chen MZ; Yu P; Sun H; Wang RL
Chem Biol Drug Des; 2018 Sep; 92(3):1647-1656. PubMed ID: 29745030
[TBL] [Abstract][Full Text] [Related]
9. Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B.
Li XQ; Xu Q; Luo J; Wang LJ; Jiang B; Zhang RS; Shi DY
Eur J Med Chem; 2017 Aug; 136():348-359. PubMed ID: 28511130
[TBL] [Abstract][Full Text] [Related]
10. Peptidomimetics as potent and selective PTP1B inhibitors.
Patel D; Jain M; Shah SR; Bahekar R; Jadav P; Shah K; Joharapurkar A; Shaikh M; Sairam KV
Med Chem; 2013 Aug; 9(5):660-71. PubMed ID: 23030658
[TBL] [Abstract][Full Text] [Related]
11. Facile fabrication of promising protein tyrosine phosphatase (PTP) inhibitor entities based on 'clicked' serine/threonine-monosaccharide hybrids.
He XP; Deng Q; Gao LX; Li C; Zhang W; Zhou YB; Tang Y; Shi XX; Xie J; Li J; Chen GR; Chen K
Bioorg Med Chem; 2011 Jul; 19(13):3892-900. PubMed ID: 21665482
[TBL] [Abstract][Full Text] [Related]
12. Synthesis and biological evaluation of oleanolic acid derivatives as PTP1B inhibitors.
Liu QC; Guo TT; Zhang L; Yu Y; Wang P; Yang JF; Li YX
Eur J Med Chem; 2013 May; 63():511-22. PubMed ID: 23531458
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and characterization of 5,7-dihydroxyflavanone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
Sun LP; Ma WP; Gao LX; Yang LL; Quan YC; Li J; Piao HR
J Enzyme Inhib Med Chem; 2013 Dec; 28(6):1199-204. PubMed ID: 23009604
[TBL] [Abstract][Full Text] [Related]
14. Synthesis, characterization and biological evaluation of thiadiazole amide derivatives as nucleoside triphosphate diphosphohydrolases (NTPDases) inhibitors.
Abbas S; Afzal S; Nadeem H; Hussain D; Langer P; Sévigny J; Ashraf Z; Iqbal J
Bioorg Chem; 2022 Jan; 118():105456. PubMed ID: 34800887
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis and docking study of 5-(substituted benzylidene)thiazolidine-2,4-dione derivatives as inhibitors of protein tyrosine phosphatase 1B.
Wang Z; Liu Z; Lee W; Kim SN; Yoon G; Cheon SH
Bioorg Med Chem Lett; 2014 Aug; 24(15):3337-40. PubMed ID: 24953600
[TBL] [Abstract][Full Text] [Related]
16. Synthesis of miltirone analogues as inhibitors of Cdc25 phosphatases.
Huang W; Li J; Zhang W; Zhou Y; Xie C; Luo Y; Li Y; Wang J; Li J; Lu W
Bioorg Med Chem Lett; 2006 Apr; 16(7):1905-8. PubMed ID: 16434190
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and biological evaluation of tryptophan-derived rhodanine derivatives as PTP1B inhibitors and anti-bacterial agents.
Liu H; Sun D; Du H; Zheng C; Li J; Piao H; Li J; Sun L
Eur J Med Chem; 2019 Jun; 172():163-173. PubMed ID: 30978561
[TBL] [Abstract][Full Text] [Related]
18. Design and synthesis of novel 1,2-dithiolan-4-yl benzoate derivatives as PTP1B inhibitors.
Chen J; Gao LX; Gong JX; Jiang CS; Yao LG; Li JY; Li J; Xiao W; Guo YW
Bioorg Med Chem Lett; 2015; 25(10):2211-6. PubMed ID: 25872983
[TBL] [Abstract][Full Text] [Related]
19. Design and synthesis of novel bis-thiazolone derivatives as micromolar CDC25 phosphatase inhibitors: effect of dimerisation on phosphatase inhibition.
Sarkis M; Tran DN; Kolb S; Miteva MA; Villoutreix BO; Garbay C; Braud E
Bioorg Med Chem Lett; 2012 Dec; 22(24):7345-50. PubMed ID: 23141909
[TBL] [Abstract][Full Text] [Related]
20. Toward a treatment of diabesity: Rational design, synthesis and biological evaluation of benzene-sulfonamide derivatives as a new class of PTP-1B inhibitors.
Ghareb N; El-Sayed NM; Abdelhameed R; Yamada K; Elgawish MS
Bioorg Chem; 2019 May; 86():322-338. PubMed ID: 30743173
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]