88 related articles for article (PubMed ID: 25333655)
1. Identification of structural features of 2-alkylidene-1,3-dicarbonyl derivatives that induce inhibition and/or activation of histone acetyltransferases KAT3B/p300 and KAT2B/PCAF.
Castellano S; Milite C; Feoli A; Viviano M; Mai A; Novellino E; Tosco A; Sbardella G
ChemMedChem; 2015 Jan; 10(1):144-57. PubMed ID: 25333655
[TBL] [Abstract][Full Text] [Related]
2. Histone acetylation and histone acetyltransferases show significant alterations in human abdominal aortic aneurysm.
Han Y; Tanios F; Reeps C; Zhang J; Schwamborn K; Eckstein HH; Zernecke A; Pelisek J
Clin Epigenetics; 2016; 8():3. PubMed ID: 26767057
[TBL] [Abstract][Full Text] [Related]
3. Inhibition of lysine acetyltransferase KAT3B/p300 activity by a naturally occurring hydroxynaphthoquinone, plumbagin.
Ravindra KC; Selvi BR; Arif M; Reddy BA; Thanuja GR; Agrawal S; Pradhan SK; Nagashayana N; Dasgupta D; Kundu TK
J Biol Chem; 2009 Sep; 284(36):24453-64. PubMed ID: 19570987
[TBL] [Abstract][Full Text] [Related]
4. Dissociable roles for histone acetyltransferases p300 and PCAF in hippocampus and perirhinal cortex-mediated object memory.
Mitchnick KA; Creighton SD; Cloke JM; Wolter M; Zaika O; Christen B; Van Tiggelen M; Kalisch BE; Winters BD
Genes Brain Behav; 2016 Jul; 15(6):542-57. PubMed ID: 27251651
[TBL] [Abstract][Full Text] [Related]
5. Probing p300/CBP associated factor (PCAF)-dependent pathways with a small molecule inhibitor.
Modak R; Basha J; Bharathy N; Maity K; Mizar P; Bhat AV; Vasudevan M; Rao VK; Kok WK; Natesh N; Taneja R; Kundu TK
ACS Chem Biol; 2013; 8(6):1311-23. PubMed ID: 23570531
[TBL] [Abstract][Full Text] [Related]
6. Identification and characterization of small-molecule inhibitors of lysine acetyltransferases.
Liao D
Methods Mol Biol; 2015; 1238():539-48. PubMed ID: 25421679
[TBL] [Abstract][Full Text] [Related]
7. Inhibition of acetyltransferase alters different histone modifications: probed by small molecule inhibitor plumbagin.
Dalvoy Vasudevarao M; Dhanasekaran K; Selvi RB; Kundu TK
J Biochem; 2012 Nov; 152(5):453-62. PubMed ID: 22923743
[TBL] [Abstract][Full Text] [Related]
8. Identification of long chain alkylidenemalonates as novel small molecule modulators of histone acetyltransferases.
Sbardella G; Castellano S; Vicidomini C; Rotili D; Nebbioso A; Miceli M; Altucci L; Mai A
Bioorg Med Chem Lett; 2008 May; 18(9):2788-92. PubMed ID: 18434144
[TBL] [Abstract][Full Text] [Related]
9. Histone acetyl transferases as emerging drug targets.
Dekker FJ; Haisma HJ
Drug Discov Today; 2009 Oct; 14(19-20):942-8. PubMed ID: 19577000
[TBL] [Abstract][Full Text] [Related]
10. A novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach.
Milite C; Feoli A; Sasaki K; La Pietra V; Balzano AL; Marinelli L; Mai A; Novellino E; Castellano S; Tosco A; Sbardella G
J Med Chem; 2015 Mar; 58(6):2779-98. PubMed ID: 25730130
[TBL] [Abstract][Full Text] [Related]
11. Targeted degradation of the enhancer lysine acetyltransferases CBP and p300.
Vannam R; Sayilgan J; Ojeda S; Karakyriakou B; Hu E; Kreuzer J; Morris R; Herrera Lopez XI; Rai S; Haas W; Lawrence M; Ott CJ
Cell Chem Biol; 2021 Apr; 28(4):503-514.e12. PubMed ID: 33400925
[TBL] [Abstract][Full Text] [Related]
12. The identification of a novel natural activator of p300 histone acetyltranferase provides new insights into the modulation mechanism of this enzyme.
Dal Piaz F; Tosco A; Eletto D; Piccinelli AL; Moltedo O; Franceschelli S; Sbardella G; Remondelli P; Rastrelli L; Vesci L; Pisano C; De Tommasi N
Chembiochem; 2010 Apr; 11(6):818-27. PubMed ID: 20373302
[TBL] [Abstract][Full Text] [Related]
13. Deciphering the binding mode and mechanistic insights of pentadecylidenemalonate (1b) as activator of histone acetyltransferase PCAF.
Suryanarayanan V; Singh SK
J Biomol Struct Dyn; 2019 Jun; 37(9):2296-2309. PubMed ID: 30044210
[TBL] [Abstract][Full Text] [Related]
14. Profiling Cellular Substrates of Lysine Acetyltransferases GCN5 and p300 with Orthogonal Labeling and Click Chemistry.
Han Z; Chou CW; Yang X; Bartlett MG; Zheng YG
ACS Chem Biol; 2017 Jun; 12(6):1547-1555. PubMed ID: 28426192
[TBL] [Abstract][Full Text] [Related]
15. Discovery of spirohydantoins as selective, orally bioavailable inhibitors of p300/CBP histone acetyltransferases.
Ji Z; Clark RF; Bhat V; Matthew Hansen T; Lasko LM; Bromberg KD; Manaves V; Algire M; Martin R; Qiu W; Torrent M; Jakob CG; Liu H; Cole PA; Marmorstein R; Kesicki EA; Lai A; Michaelides MR
Bioorg Med Chem Lett; 2021 May; 39():127854. PubMed ID: 33631370
[TBL] [Abstract][Full Text] [Related]
16. Histone acetyltransferases interact with and acetylate p70 ribosomal S6 kinases in vitro and in vivo.
Fenton TR; Gwalter J; Ericsson J; Gout IT
Int J Biochem Cell Biol; 2010 Feb; 42(2):359-66. PubMed ID: 19961954
[TBL] [Abstract][Full Text] [Related]
17. Modulation of the activity of histone acetyltransferases by long chain alkylidenemalonates (LoCAMs).
Milite C; Castellano S; Benedetti R; Tosco A; Ciliberti C; Vicidomini C; Boully L; Franci G; Altucci L; Mai A; Sbardella G
Bioorg Med Chem; 2011 Jun; 19(12):3690-701. PubMed ID: 21292492
[TBL] [Abstract][Full Text] [Related]
18. Regulation of histone acetyltransferase activity of p300 and PCAF by proto-oncogene protein DEK.
Ko SI; Lee IS; Kim JY; Kim SM; Kim DW; Lee KS; Woo KM; Baek JH; Choo JK; Seo SB
FEBS Lett; 2006 May; 580(13):3217-22. PubMed ID: 16696975
[TBL] [Abstract][Full Text] [Related]
19. Bisubstrate analogue structure-activity relationships for p300 histone acetyltransferase inhibitors.
Sagar V; Zheng W; Thompson PR; Cole PA
Bioorg Med Chem; 2004 Jun; 12(12):3383-90. PubMed ID: 15158807
[TBL] [Abstract][Full Text] [Related]
20. Structure-Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase.
Madia VN; Benedetti R; Barreca ML; Ngo L; Pescatori L; Messore A; Pupo G; Saccoliti F; Valente S; Mai A; Scipione L; Zheng YG; Tintori C; Botta M; Cecchetti V; Altucci L; Di Santo R; Costi R
ChemMedChem; 2017 Aug; 12(16):1359-1368. PubMed ID: 28346821
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]