These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

164 related articles for article (PubMed ID: 25375781)

  • 41. Synthesis and biological evaluation of analogues of 7-chloro-4,5-dihydro-4- oxo-8-(1,2,4-triazol-4-yl)-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylic acid (TQX-173) as novel selective AMPA receptor antagonists.
    Catarzi D; Colotta V; Varano F; Calabri FR; Filacchioni G; Galli A; Costagli C; Carlà V
    J Med Chem; 2004 Jan; 47(1):262-72. PubMed ID: 14695840
    [TBL] [Abstract][Full Text] [Related]  

  • 42. Simultaneous determination of enantiomerization and hydrolysis kinetic parameters of chiral N-alkylbenzothiadiazine derivatives.
    Carrozzo MM; Cannazza G; Battisti U; Braghiroli D; Parenti C
    Chirality; 2010 May; 22(4):389-97. PubMed ID: 19575466
    [TBL] [Abstract][Full Text] [Related]  

  • 43. Heteroaryl analogues of AMPA. 2. Synthesis, absolute stereochemistry, photochemistry, and structure-activity relationships.
    Falch E; Brehm L; Mikkelsen I; Johansen TN; Skjaerbaek N; Nielsen B; Stensbøl TB; Ebert B; Krogsgaard-Larsen P
    J Med Chem; 1998 Jul; 41(14):2513-23. PubMed ID: 9651156
    [TBL] [Abstract][Full Text] [Related]  

  • 44. Structural analysis of the positive AMPA receptor modulators CX516 and Me-CX516 in complex with the GluA2 ligand-binding domain.
    Krintel C; Harpsøe K; Zachariassen LG; Peters D; Frydenvang K; Pickering DS; Gajhede M; Kastrup JS
    Acta Crystallogr D Biol Crystallogr; 2013 Sep; 69(Pt 9):1645-52. PubMed ID: 23999288
    [TBL] [Abstract][Full Text] [Related]  

  • 45. Synthesis and biological evaluation of new 3-aralkylamino-2-aryl-2H-1, 2,4-pyridothiadiazine 1,1-dioxides as potential CCK-receptor ligands.
    De Tullio P; Pirotte B; Neven P; Masereel B; Dewalque D; Diouf O; Podona T; Caignard D; Renard P; Delarge J
    J Pharm Pharmacol; 1997 May; 49(5):463-71. PubMed ID: 9178178
    [TBL] [Abstract][Full Text] [Related]  

  • 46. [3-Amino-2H-1,2,4-benzothiadiazine-1,1-dioxides with antihypertensive and possibly diabetogenic activity (author's transl)].
    Wollweber H; Horstmann H; Stoepel K; Garthoff B; Puls W; Krause HP; Thomas G
    Arzneimittelforschung; 1981; 31(2):279-88. PubMed ID: 7013769
    [TBL] [Abstract][Full Text] [Related]  

  • 47. Positive allosteric modulators of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor.
    Grove SJ; Jamieson C; Maclean JK; Morrow JA; Rankovic Z
    J Med Chem; 2010 Oct; 53(20):7271-9. PubMed ID: 20839777
    [No Abstract]   [Full Text] [Related]  

  • 48. [Synthesis of several benzothiadiazine derivatives. 3-substituted 7-chloro-2H-1,2,4-benzothiadizine 1, 1-dioxide and 3-substituted 7-chloro-3, 4-dihydro-2H-1, 2,4-benzothiadiazine 1, 1-dioxide].
    SUZUE S; HAYASHI S
    Yakugaku Zasshi; 1962 Aug; 82():1192-4. PubMed ID: 13979452
    [No Abstract]   [Full Text] [Related]  

  • 49. Pharmacological characterization of cGMP regulation by the biarylpropylsulfonamide class of positive, allosteric modulators of alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptors.
    Ryder JW; Falcone JF; Manro JR; Svensson KA; Merchant KM
    J Pharmacol Exp Ther; 2006 Oct; 319(1):293-8. PubMed ID: 16803862
    [TBL] [Abstract][Full Text] [Related]  

  • 50. Triphenylphosphonium salts of 1,2,4-benzothiadiazine 1,1-dioxides related to diazoxide targeting mitochondrial ATP-sensitive potassium channels.
    Constant-Urban C; Charif M; Goffin E; Van Heugen JC; Elmoualij B; Chiap P; Mouithys-Mickalad A; Serteyn D; Lebrun P; Pirotte B; De Tullio P
    Bioorg Med Chem Lett; 2013 Nov; 23(21):5878-81. PubMed ID: 24055044
    [TBL] [Abstract][Full Text] [Related]  

  • 51. Novel arylpyrazino[2,3-c][1,2,6]thiadiazine 2,2-dioxides as inhibitors of platelet aggregation. 1. Synthesis and pharmacological evaluation.
    Campillo N; García C; Goya P; Páez JA; Carrasco E; Grau M
    J Med Chem; 1999 May; 42(10):1698-704. PubMed ID: 10346922
    [TBL] [Abstract][Full Text] [Related]  

  • 52. The diazoxide derivative IDRA 21 enhances ischemic hippocampal neuron injury.
    Yamada KA; Covey DF; Hsu CY; Hu R; Hu Y; He YY
    Ann Neurol; 1998 May; 43(5):664-9. PubMed ID: 9585363
    [TBL] [Abstract][Full Text] [Related]  

  • 53. Positive modulation of alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid (AMPA) receptors in prefrontal cortical pyramidal neurons by a novel allosteric potentiator.
    Baumbarger PJ; Muhlhauser M; Zhai J; Yang CR; Nisenbaum ES
    J Pharmacol Exp Ther; 2001 Jul; 298(1):86-102. PubMed ID: 11408529
    [TBL] [Abstract][Full Text] [Related]  

  • 54. Synthesis, theoretical and structural analyses, and enantiopharmacology of 3-carboxy homologs of AMPA.
    Brehm L; Greenwood JR; Sløk FA; Holm MM; Nielsen B; Geneser U; Stensbøl TB; Bräuner-Osborne H; Begtrup M; Egebjerg J; Krogsgaard-Larsen P
    Chirality; 2004 Aug; 16(7):452-66. PubMed ID: 15236343
    [TBL] [Abstract][Full Text] [Related]  

  • 55. Alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor channels lacking the N-terminal domain.
    Pasternack A; Coleman SK; Jouppila A; Mottershead DG; Lindfors M; Pasternack M; Keinänen K
    J Biol Chem; 2002 Dec; 277(51):49662-7. PubMed ID: 12393905
    [TBL] [Abstract][Full Text] [Related]  

  • 56. Comparison of single vs. multiple administrations of the AMPA receptors modulator S 18986 in the object recognition task in rats.
    Bertaina-Anglade V; la Rochelle CD; Muñoz C; Morain P; Bernard K
    Fundam Clin Pharmacol; 2007 Aug; 21(4):349-54. PubMed ID: 17635172
    [TBL] [Abstract][Full Text] [Related]  

  • 57. Probing the allosteric modulator binding site of GluR2 with thiazide derivatives.
    Ptak CP; Ahmed AH; Oswald RE
    Biochemistry; 2009 Sep; 48(36):8594-602. PubMed ID: 19673491
    [TBL] [Abstract][Full Text] [Related]  

  • 58. The structure of a mixed GluR2 ligand-binding core dimer in complex with (S)-glutamate and the antagonist (S)-NS1209.
    Kasper C; Pickering DS; Mirza O; Olsen L; Kristensen AS; Greenwood JR; Liljefors T; Schousboe A; Wätjen F; Gajhede M; Sigurskjold BW; Kastrup JS
    J Mol Biol; 2006 Apr; 357(4):1184-201. PubMed ID: 16483599
    [TBL] [Abstract][Full Text] [Related]  

  • 59. DRUG FOCUS: S 18986: A positive allosteric modulator of AMPA-type glutamate receptors pharmacological profile of a novel cognitive enhancer.
    Bernard K; Danober L; Thomas JY; Lebrun C; Muñoz C; Cordi A; Desos P; Lestage P; Morain P
    CNS Neurosci Ther; 2010 Oct; 16(5):e193-212. PubMed ID: 21050420
    [TBL] [Abstract][Full Text] [Related]  

  • 60. Enantiomeric resolution with a new chiral stationary phase of 7-chloro-3-methyl-3,4-dihydro-2H-1,2,4-benzothiadiazine S,S-dioxide, a cognition-enhancing benzothiadiazine derivative.
    Uzunov DP; Zivkovich I; Pirkle WH; Costa E; Guidotti A
    J Pharm Sci; 1995 Aug; 84(8):937-42. PubMed ID: 7500277
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 9.