106 related articles for article (PubMed ID: 2544725)
1. Hexestrol-linked cytotoxic agents: synthesis and binding affinity for estrogen receptors.
Köhle H; Krohn K; Leclercq G
J Med Chem; 1989 Jul; 32(7):1538-47. PubMed ID: 2544725
[TBL] [Abstract][Full Text] [Related]
2. Estrogenic affinity labels: synthesis, irreversible receptor binding, and bioactivity of aziridine-substituted hexestrol derivatives.
Zablocki JA; Katzenellenbogen JA; Carlson KE; Norman MJ; Katzenellenbogen BS
J Med Chem; 1987 May; 30(5):829-38. PubMed ID: 3033242
[TBL] [Abstract][Full Text] [Related]
3. Influence of alkyl chain ramification on estradiol receptor binding affinity and intrinsic activity of 1,2-dialkylated 1,2-bis(4- or 3-hydroxyphenyl)ethane estrogens and antiestrogens.
Hartmann RW
J Med Chem; 1986 Sep; 29(9):1668-74. PubMed ID: 3018243
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, receptor binding, and target-tissue uptake of carbon-11 labeled carbamate derivatives of estradiol and hexestrol.
Ouellet R; Rousseau J; Brasseur N; van Lier JE; Diksic M; Westera G
J Med Chem; 1984 Apr; 27(4):509-13. PubMed ID: 6323712
[TBL] [Abstract][Full Text] [Related]
5. Preparation, receptor binding, and fluorescence properties of hexestrol-fluorophore conjugates: evaluation of site of attachment, fluorophore structure, and fluorophore-ligand spacing.
Fevig TL; Lloyd JE; Zablocki JA; Katzenellenbogen JA
J Med Chem; 1987 Jan; 30(1):156-65. PubMed ID: 3027331
[TBL] [Abstract][Full Text] [Related]
6. Nonsteroidal estrogens: synthesis and estrogen receptor binding affinity of derivatives of (3R*,4S*)-3,4-bis(4-hydroxyphenyl)hexane (hexestrol) and (2R*,3S*)-2,3-bis(4-hydroxyphenyl)pentane (norhexestrol) functionalized on the side chain.
Landvatter SW; Katzenellenbogen JA
J Med Chem; 1982 Nov; 25(11):1300-7. PubMed ID: 6292423
[TBL] [Abstract][Full Text] [Related]
7. [Synthesis of 3,3'disubstituted hexestrol derivatives and their binding affinity to cytoplasmatic estrogen receptors (author's transl)].
Hamacher H
Arch Pharm (Weinheim); 1981 Jul; 314(7):631-44. PubMed ID: 6271092
[No Abstract] [Full Text] [Related]
8. Estrogen photoaffinity labels. 2. Reversible binding and covalent attachment of photosensitive hexestrol derivatives to the uterine estrogen receptor.
Katzenellenbogen JA; Carlson KE; Johnson HJ; Myers HN
Biochemistry; 1977 May; 16(9):1970-6. PubMed ID: 870034
[TBL] [Abstract][Full Text] [Related]
9. Ring-substituted 1,2-dialkylated 1,2-bis(hydroxyphenyl)ethanes. 1. Synthesis and estrogen receptor binding affinity of 2,2'- and 3,3'-disubstituted hexestrols.
Hartmann RW; Schwarz W; Schönenberger H
J Med Chem; 1983 Aug; 26(8):1137-44. PubMed ID: 6308256
[TBL] [Abstract][Full Text] [Related]
10. Chemically reactive estrogens: synthesis and estrogen receptor interactions of hexestrol ether derivatives and 4-substituted deoxyhexestrol derivatives bearing alkylating functions.
Katzenellenbogen JA; McGorrin RJ; Tatee T; Kempton RJ; Carlson KE; Kinder DH
J Med Chem; 1981 Apr; 24(4):435-50. PubMed ID: 6267281
[TBL] [Abstract][Full Text] [Related]
11. (2R*, 3S*)-1-[18F]fluoro-2,3-bis(4-hydroxyphenyl)pentane [( 18F]fluoronor-hexestrol), a positron-emitting estrogen that shows highly-selective, receptor-mediated uptake by target tissues in vivo.
Landvatter SW; Kiesewetter DO; Kilbourn MR; Katzenellenbogen JA; Welch MJ
Life Sci; 1983 Nov; 33(19):1933-8. PubMed ID: 6316052
[TBL] [Abstract][Full Text] [Related]
12. [Potential antineoplastics, 6. Synthesis of hexestrol derivatives with alkylating side chains].
Hamacher H; Mangold C
Arch Pharm (Weinheim); 1983; 316(3):271-81. PubMed ID: 6305306
[No Abstract] [Full Text] [Related]
13. Diethylstilbestrol-linked cytotoxic agents: synthesis and binding affinity for estrogen receptors.
Krohn K; Kulikowski K; Leclercq G
J Med Chem; 1989 Jul; 32(7):1532-8. PubMed ID: 2738889
[TBL] [Abstract][Full Text] [Related]
14. Estrogen receptor based imaging agents. 2. Synthesis and receptor binding affinity of side-chain halogenated hexestrol derivatives.
Goswami R; Harsy SG; Heiman DF; Katzenellenbogen JA
J Med Chem; 1980 Sep; 23(9):1002-8. PubMed ID: 6251218
[TBL] [Abstract][Full Text] [Related]
15. Synthesis, receptor binding and target-tissue uptake of carbon-11-labeled carbamate derivatives of estradiol and hexestrol.
Ali H; Rousseau J; Diksic M; van Lier JE
Int J Rad Appl Instrum B; 1992 Feb; 19(2):175-82. PubMed ID: 1318291
[TBL] [Abstract][Full Text] [Related]
16. 3,4-bis(3'-hydroxyphenyl)hexane--a new mammary tumor-inhibiting compound.
Kranzfelder G; Hartmann RW; von Angerer E; Schönenberger H; Bogden AE
J Cancer Res Clin Oncol; 1982; 103(2):165-80. PubMed ID: 6284766
[TBL] [Abstract][Full Text] [Related]
17. Coumestrol, NBD-norhexestrol, and dansyl-norhexestrol, fluorescent probes of estrogen-binding protiens.
Lee YJ; Notides AC; Tsay YG; Kende AS
Biochemistry; 1977 Jun; 16(13):2896-901. PubMed ID: 880286
[No Abstract] [Full Text] [Related]
18. Ring-substituted 1,1,2,2-tetraalkylated 1,2-bis(hydroxyphenyl)ethanes. 4. Synthesis, estrogen receptor binding affinity, and evaluation of antiestrogenic and mammary tumor inhibiting activity of symmetrically disubstituted 1,1,2,2-tetramethyl-1,2-bis(hydroxyphenyl)ethanes.
Hartmann RW; Schwarz W; Heindl A; Schönenberger H
J Med Chem; 1985 Sep; 28(9):1295-301. PubMed ID: 2993619
[TBL] [Abstract][Full Text] [Related]
19. Ring-substituted 1,2-dialkylated 1,2-bis(hydroxyphenyl)ethanes. 3. Synthesis, estrogen receptor binding affinity, and evaluation of antiestrogenic and mammary tumor inhibiting activity of 2,2'-disubstituted butestrols and 6,6'-disubstituted metabutestrols.
Hartmann RW; Heindl A; Schwarz W; Schönenberger H
J Med Chem; 1984 Jul; 27(7):819-24. PubMed ID: 6330356
[TBL] [Abstract][Full Text] [Related]
20. Synthesis of novel hexestrol and diethylstilbestrol derivatives as potential anticancer and estrogenic agents.
Ibrahim ES; Omar AM; Khalil MA; Makar MA; Soliman MT; Daabees TT
Pharmazie; 1980 Feb; 35(2):80-4. PubMed ID: 6247720
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]