148 related articles for article (PubMed ID: 25455485)
1. Synthesis of novel triazole-linked mefloquine derivatives: biological evaluation against Plasmodium falciparum.
Hamann AR; de Kock C; Smith PJ; van Otterlo WA; Blackie MA
Bioorg Med Chem Lett; 2014 Dec; 24(23):5466-9. PubMed ID: 25455485
[TBL] [Abstract][Full Text] [Related]
2. New compounds hybrids 1h-1,2,3-triazole-quinoline against Plasmodium falciparum.
Boechat N; Ferreira Mde L; Pinheiro LC; Jesus AM; Leite MM; Júnior CC; Aguiar AC; de Andrade IM; Krettli AU
Chem Biol Drug Des; 2014 Sep; 84(3):325-32. PubMed ID: 24803084
[TBL] [Abstract][Full Text] [Related]
3. 1H-1,2,3-triazole tethered mono- and bis-ferrocenylchalcone-β-lactam conjugates: synthesis and antimalarial evaluation.
Kumar K; Pradines B; Madamet M; Amalvict R; Kumar V
Eur J Med Chem; 2014 Oct; 86():113-21. PubMed ID: 25147153
[TBL] [Abstract][Full Text] [Related]
4. In vitro antiplasmodial activity of triazole-linked chloroquinoline derivatives synthesized from 7-chloro-N-(prop-2-yn-1-yl)quinolin-4-amine.
Taleli L; de Kock C; Smith PJ; Pelly SC; Blackie MAL; van Otterlo WAL
Bioorg Med Chem; 2015 Aug; 23(15):4163-4171. PubMed ID: 26174655
[TBL] [Abstract][Full Text] [Related]
5. In vitro antimalarial activity of novel trifluoromethyl- and bis(trifluoromethyl)quinoline derivatives.
Kgokong JL; Matsabisa GM; Breytenbach JC
Arzneimittelforschung; 2001 Feb; 51(2):163-8. PubMed ID: 11258047
[TBL] [Abstract][Full Text] [Related]
6. In vitro antimalarial activity, β-haematin inhibition and structure-activity relationships in a series of quinoline triazoles.
Joshi MC; Wicht KJ; Taylor D; Hunter R; Smith PJ; Egan TJ
Eur J Med Chem; 2013 Nov; 69():338-47. PubMed ID: 24077524
[TBL] [Abstract][Full Text] [Related]
7. Diversification of quinoline-triazole scaffolds with CORMs: Synthesis, in vitro and in silico biological evaluation against Plasmodium falciparum.
Ishmail FZ; Melis DR; Mbaba M; Smith GS
J Inorg Biochem; 2021 Feb; 215():111328. PubMed ID: 33340802
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and Antiplasmodial Activity of 1,2,3-Triazole-Naphthoquinone Conjugates.
Oramas-Royo S; López-Rojas P; Amesty Á; Gutiérrez D; Flores N; Martín-Rodríguez P; Fernández-Pérez L; Estévez-Braun A
Molecules; 2019 Oct; 24(21):. PubMed ID: 31671684
[TBL] [Abstract][Full Text] [Related]
9. New hybrid trifluoromethylquinolines as antiplasmodium agents.
da Silva RMRJ; Gandi MO; Mendonça JS; Carvalho AS; Coutinho JP; Aguiar ACC; Krettli AU; Boechat N
Bioorg Med Chem; 2019 Mar; 27(6):1002-1008. PubMed ID: 30737133
[TBL] [Abstract][Full Text] [Related]
10. Enhanced activity of mefloquine and artesunic acid against Plasmodium falciparum in vitro and P. berghei in mice by combination with ciprofloxacin.
Andrade AA; de Pilla Varotti F; de Freitas IO; de Souza MV; Vasconcelos TR; Boechat N; Krettli AU
Eur J Pharmacol; 2007 Mar; 558(1-3):194-8. PubMed ID: 17214980
[TBL] [Abstract][Full Text] [Related]
11. Susceptibility of Plasmodium falciparum to the drugs used to treat severe malaria (quinine) and to prevent malaria (mefloquine, cycloguanil) in Comoros Union and Madagascar.
Randrianarivelojosia M; Randrianasolo L; Randremanana RV; Randriamanantena A; Ratsimbasoa A; Rakotoson JD
S Afr Med J; 2004 Jan; 94(1):47-51. PubMed ID: 14971233
[TBL] [Abstract][Full Text] [Related]
12. [Mefloquine resistance in Plasmodium falciparum malaria].
Garavelli PL
Recenti Prog Med; 2003; 94(7-8):343. PubMed ID: 12868243
[No Abstract] [Full Text] [Related]
13. 7-Chloroquinolinotriazoles: synthesis by the azide-alkyne cycloaddition click chemistry, antimalarial activity, cytotoxicity and SAR studies.
Pereira GR; Brandão GC; Arantes LM; de Oliveira HA; de Paula RC; do Nascimento MF; dos Santos FM; da Rocha RK; Lopes JC; de Oliveira AB
Eur J Med Chem; 2014 Feb; 73():295-309. PubMed ID: 24469080
[TBL] [Abstract][Full Text] [Related]
14. In-vitro sensitivity of Plasmodium falciparum to chloroquine, halofantrine, mefloquine and quinine in Madagascar.
Randrianarivelojosia M; Ratsimbasoa A; Randrianasolo L; Randrianarijaona A; Jambou R
East Afr Med J; 2002 May; 79(5):237-41. PubMed ID: 12638806
[TBL] [Abstract][Full Text] [Related]
15. In vitro antiplasmodial efficacy of synthetic coumarin-triazole analogs.
Yadav N; Agarwal D; Kumar S; Dixit AK; Gupta RD; Awasthi SK
Eur J Med Chem; 2018 Feb; 145():735-745. PubMed ID: 29366931
[TBL] [Abstract][Full Text] [Related]
16. 3,5-bis(benzylidene)-4-piperidones and related N-acyl analogs: a novel cluster of antimalarials targeting the liver stage of Plasmodium falciparum.
Das U; Singh RS; Alcorn J; Hickman MR; Sciotti RJ; Leed SE; Lee PJ; Roncal N; Dimmock JR
Bioorg Med Chem; 2013 Dec; 21(23):7250-6. PubMed ID: 24139941
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and antiplasmodial activity of novel indoleamide derivatives bearing sulfonamide and triazole pharmacophores.
Devender N; Gunjan S; Tripathi R; Tripathi RP
Eur J Med Chem; 2017 May; 131():171-184. PubMed ID: 28319782
[TBL] [Abstract][Full Text] [Related]
18. Targeting Asexual and Sexual Blood Stages of the Human Malaria Parasite P. falciparum with 7-Chloroquinoline-Based 1,2,3-Triazoles.
Wadi I; Prasad D; Batra N; Srivastava K; Anvikar AR; Valecha N; Nath M
ChemMedChem; 2019 Feb; 14(4):484-493. PubMed ID: 30609264
[TBL] [Abstract][Full Text] [Related]
19. [Evaluation of the Plasmodium falciparum response to chloroquine, quinine and mefloquine].
Di Santi SM; Camargo Neves VL; Boulos M; Dutra AP; Ramos AM; Santos M; Barata LC
Rev Inst Med Trop Sao Paulo; 1988; 30(3):147-52. PubMed ID: 3065907
[No Abstract] [Full Text] [Related]
20. In vitro susceptibility of chloroquine resistant Plasmodium falciparum to mefloquine in Delhi.
Gajanana A; Sinha S; Vasisth S
Indian J Malariol; 1986 Dec; 23(2):91-4. PubMed ID: 3552761
[No Abstract] [Full Text] [Related]
[Next] [New Search]