119 related articles for article (PubMed ID: 25537913)
1. [Design, synthesis and biological activity assessment of phenoxybutyric acid derivatives as nonsteroidal 5α-reductase inhibitors].
Chen K; Jiang Z; Chen W; Xi B
Nan Fang Yi Ke Da Xue Xue Bao; 2014 Dec; 34(12):1830-3. PubMed ID: 25537913
[TBL] [Abstract][Full Text] [Related]
2. Synthesis of tricyclic compounds as steroid 5alpha-reductase inhibitors.
Takami H; Nonaka H; Kishibayashi N; Ishii A; Kase H; Kumazawa T
Chem Pharm Bull (Tokyo); 2000 Apr; 48(4):552-5. PubMed ID: 10783077
[TBL] [Abstract][Full Text] [Related]
3. Design, synthesis and biological evaluation of novel 3-oxo-4-oxa-5α-androst-17β-amide derivatives as dual 5α-reductase inhibitors and androgen receptor antagonists.
Lao K; Sun J; Wang C; Wang Y; You Q; Xiao H; Xiang H
Bioorg Med Chem Lett; 2017 Sep; 27(17):4212-4217. PubMed ID: 28757062
[TBL] [Abstract][Full Text] [Related]
4. Design, synthesis and biological evaluation of novel androst-3,5-diene-3-carboxylic acid derivatives as inhibitors of 5α-reductase type 1 and 2.
Lao K; Sun J; Wang C; Lyu W; Zhou B; Zhao R; Xu Q; You Q; Xiang H
Steroids; 2017 Aug; 124():29-34. PubMed ID: 28549802
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and activity of novel 16-dehydropregnenolone acetate derivatives as inhibitors of type 1 5α-reductase and on cancer cell line SK-LU-1.
Silva-Ortiz AV; Bratoeff E; Ramírez-Apan T; Heuze Y; Sánchez A; Soriano J; Cabeza M
Bioorg Med Chem; 2015 Dec; 23(24):7535-42. PubMed ID: 26631442
[TBL] [Abstract][Full Text] [Related]
6. Design, synthesis, and biological evaluation of novel androst-17β-amide structurally related compounds as dual 5α-reductase inhibitors and androgen receptor antagonists.
Lao K; Xun G; Gou X; Xiang H
J Enzyme Inhib Med Chem; 2019 Dec; 34(1):1597-1606. PubMed ID: 31469015
[TBL] [Abstract][Full Text] [Related]
7. Activity of steroid 4 and derivatives 4a-4f as inhibitors of the enzyme 5α-reductase 1.
Arellano Y; Bratoeff E; Heuze Y; Bravo M; Soriano J; Cabeza M
Bioorg Med Chem; 2018 Aug; 26(14):4058-4064. PubMed ID: 30007568
[TBL] [Abstract][Full Text] [Related]
8. Synthesis, Biological Evaluation and Molecular Docking of Avicequinone C Analogues as Potential Steroid 5α-Reductase Inhibitors.
Karnsomwan W; Netcharoensirisuk P; Rungrotmongkol T; De-Eknamkul W; Chamni S
Chem Pharm Bull (Tokyo); 2017; 65(3):253-260. PubMed ID: 28250347
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and characterization of 3β-substituted amides of 17a-aza-D-homo- 4-androsten-17-one as potent 5α-reductase inhibitors and antimicrobial agents.
Malhotra M; Sharma R; Rawal RK; Heer H; Bhardwaj TR
Curr Top Med Chem; 2013 Aug; 13(16):2047-61. PubMed ID: 23895091
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and biological evaluation of novel unsaturated carboxysteroids as human 5α-reductase inhibitors: a legitimate approach.
Aggarwal S; Thareja S; Bhardwaj TR; Haupenthal J; Hartmann RW; Kumar M
Eur J Med Chem; 2012 Aug; 54():728-39. PubMed ID: 22776417
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and 5α-reductase inhibitory activity of C₂₁ steroids having 1,4-diene or 4,6-diene 20-ones and 4-azasteroid 20-oximes.
Kim S; Kim YU; Ma E
Molecules; 2011 Dec; 17(1):355-68. PubMed ID: 22210173
[TBL] [Abstract][Full Text] [Related]
12. In vivo and in vitro effect of androstene derivatives as 5α-reductase type 1 enzyme inhibitors.
Bratoeff E; Sánchez A; Arellano Y; Heuze Y; Soriano J; Cabeza M
J Enzyme Inhib Med Chem; 2013 Dec; 28(6):1247-54. PubMed ID: 23051174
[TBL] [Abstract][Full Text] [Related]
13. Steroidal pyrazolines and pyrazoles as potential 5α-reductase inhibitors: synthesis and biological evaluation.
Banday AH; Shameem SA; Jeelani S
Steroids; 2014 Dec; 92():13-9. PubMed ID: 25278254
[TBL] [Abstract][Full Text] [Related]
14. Hydrazonoyl halides as precursors for new fused heterocycles of 5α-reductase inhibitors.
Farghaly TA; Gomha SM; Abbas EM; Abdalla MM
Arch Pharm (Weinheim); 2012 Feb; 345(2):117-22. PubMed ID: 21997851
[TBL] [Abstract][Full Text] [Related]
15. New Potent 5α- Reductase and Aromatase Inhibitors Derived from 1,2,3-Triazole Derivative.
El-Naggar M; El-All ASA; El-Naem SIA; Abdalla MM; Rashdan HRM
Molecules; 2020 Feb; 25(3):. PubMed ID: 32033281
[TBL] [Abstract][Full Text] [Related]
16. 5α-reductase inhibitors, antiviral and anti-tumor activities of some steroidal cyanopyridinone derivatives.
Al-Mohizea AM; Al-Omar MA; Abdalla MM; Amr AG
Int J Biol Macromol; 2012 Jan; 50(1):171-9. PubMed ID: 22057085
[TBL] [Abstract][Full Text] [Related]
17. Steroid 5alpha-reductase inhibitors.
Flores E; Bratoeff E; Cabeza M; Ramirez E; Quiroz A; Heuze I
Mini Rev Med Chem; 2003 May; 3(3):225-37. PubMed ID: 12570838
[TBL] [Abstract][Full Text] [Related]
18. Synthesis of new derivatives of 21-imidazolyl-16-dehydropregnenolone as inhibitors of 5α-reductase 2 and with cytotoxic activity in cancer cells.
Silva-Ortiz AV; Bratoeff E; Ramírez-Apan T; Heuze Y; Soriano J; Moreno I; Bravo M; Bautista L; Cabeza M
Bioorg Med Chem; 2017 Mar; 25(5):1600-1607. PubMed ID: 28174065
[TBL] [Abstract][Full Text] [Related]
19. Synthesis of bioactive polyheterocyclic ring systems as 5α-reductase inhibitors.
Abdel Hafez NA; Farghaly TA; Al-Omar MA; Abdalla MM
Eur J Med Chem; 2010 Nov; 45(11):4838-44. PubMed ID: 20739104
[TBL] [Abstract][Full Text] [Related]
20. 4-(Benzoylindolizinyl)butyric acids; novel nonsteroidal inhibitors of steroid 5alpha-reductase. III.
Sawada K; Okada S; Kuroda A; Watanabe S; Sawada Y; Tanaka H
Chem Pharm Bull (Tokyo); 2001 Jul; 49(7):799-813. PubMed ID: 11456083
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
