166 related articles for article (PubMed ID: 25554733)
1. Structure-activity relationship studies of SETD8 inhibitors.
Ma A; Yu W; Xiong Y; Butler KV; Brown PJ; Jin J
Medchemcomm; 2014 Dec; 5(12):1892-1898. PubMed ID: 25554733
[TBL] [Abstract][Full Text] [Related]
2. Discovery of a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8.
Ma A; Yu W; Li F; Bleich RM; Herold JM; Butler KV; Norris JL; Korboukh V; Tripathy A; Janzen WP; Arrowsmith CH; Frye SV; Vedadi M; Brown PJ; Jin J
J Med Chem; 2014 Aug; 57(15):6822-33. PubMed ID: 25032507
[TBL] [Abstract][Full Text] [Related]
3. Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors.
Milite C; Feoli A; Viviano M; Rescigno D; Mai A; Castellano S; Sbardella G
ChemMedChem; 2016 Aug; 11(16):1680-5. PubMed ID: 27411844
[TBL] [Abstract][Full Text] [Related]
4. The emerging role of lysine methyltransferase SETD8 in human diseases.
Milite C; Feoli A; Viviano M; Rescigno D; Cianciulli A; Balzano AL; Mai A; Castellano S; Sbardella G
Clin Epigenetics; 2016; 8():102. PubMed ID: 27688818
[TBL] [Abstract][Full Text] [Related]
5. Epigenetic Modifier SETD8 as a Therapeutic Target for High-Grade Serous Ovarian Cancer.
Wada M; Kukita A; Sone K; Hamamoto R; Kaneko S; Komatsu M; Takahashi Y; Inoue F; Kojima M; Honjoh H; Taguchi A; Kashiyama T; Miyamoto Y; Tanikawa M; Tsuruga T; Mori-Uchino M; Wada-Hiraike O; Osuga Y; Fujii T
Biomolecules; 2020 Dec; 10(12):. PubMed ID: 33339442
[TBL] [Abstract][Full Text] [Related]
6. Roles for the methyltransferase SETD8 in DNA damage repair.
Xu L; Zhang L; Sun J; Hu X; Kalvakolanu DV; Ren H; Guo B
Clin Epigenetics; 2022 Mar; 14(1):34. PubMed ID: 35246238
[TBL] [Abstract][Full Text] [Related]
7. USP29 Deubiquitinates SETD8 and Regulates DNA Damage-Induced H4K20 Monomethylation and 53BP1 Focus Formation.
Hernández-Reyes Y; Paz-Cabrera MC; Freire R; Smits VAJ
Cells; 2022 Aug; 11(16):. PubMed ID: 36010569
[TBL] [Abstract][Full Text] [Related]
8. Small-molecule inhibitors of SETD8 with cellular activity.
Blum G; Ibáñez G; Rao X; Shum D; Radu C; Djaballah H; Rice JC; Luo M
ACS Chem Biol; 2014 Nov; 9(11):2471-8. PubMed ID: 25137013
[TBL] [Abstract][Full Text] [Related]
9. Histone lysine methyltransferase Pr-set7/SETD8 promotes neural stem cell reactivation.
Huang J; Gujar MR; Deng Q; Y Chia S; Li S; Tan P; Sung WK; Wang H
EMBO Rep; 2021 Apr; 22(4):e50994. PubMed ID: 33565211
[TBL] [Abstract][Full Text] [Related]
10. The Histone Methyltransferase SETD8 Regulates the Expression of Tumor Suppressor Genes via H4K20 Methylation and the p53 Signaling Pathway in Endometrial Cancer Cells.
Kukita A; Sone K; Kaneko S; Kawakami E; Oki S; Kojima M; Wada M; Toyohara Y; Takahashi Y; Inoue F; Tanimoto S; Taguchi A; Fukuda T; Miyamoto Y; Tanikawa M; Mori-Uchino M; Tsuruga T; Iriyama T; Matsumoto Y; Nagasaka K; Wada-Hiraike O; Oda K; Hamamoto R; Osuga Y
Cancers (Basel); 2022 Oct; 14(21):. PubMed ID: 36358786
[TBL] [Abstract][Full Text] [Related]
11. The Use of Nucleosome Substrates Improves Binding of SAM Analogs to SETD8.
Strelow JM; Xiao M; Cavitt RN; Fite NC; Margolis BJ; Park KJ
J Biomol Screen; 2016 Sep; 21(8):786-94. PubMed ID: 27369108
[TBL] [Abstract][Full Text] [Related]
12. The SETD8/PR-Set7 Methyltransferase Functions as a Barrier to Prevent Senescence-Associated Metabolic Remodeling.
Tanaka H; Takebayashi SI; Sakamoto A; Igata T; Nakatsu Y; Saitoh N; Hino S; Nakao M
Cell Rep; 2017 Feb; 18(9):2148-2161. PubMed ID: 28249161
[TBL] [Abstract][Full Text] [Related]
13. Targeting the methyltransferase SETD8 impairs tumor cell survival and overcomes drug resistance independently of p53 status in multiple myeloma.
Herviou L; Ovejero S; Izard F; Karmous-Gadacha O; Gourzones C; Bellanger C; De Smedt E; Ma A; Vincent L; Cartron G; Jin J; De Bruyne E; Grimaud C; Julien E; Moreaux J
Clin Epigenetics; 2021 Sep; 13(1):174. PubMed ID: 34530900
[TBL] [Abstract][Full Text] [Related]
14. Structural basis of nucleosomal H4K20 methylation by methyltransferase SET8.
Shi L; Huang L; Long H; Song A; Zhou Z
FASEB J; 2022 Jun; 36(6):e22338. PubMed ID: 35532550
[TBL] [Abstract][Full Text] [Related]
15. [The biological functions of lysine methyltransferase PR-SET7].
Liang XQ; Du YP; Wang DL; Yang Y
Yi Chuan; 2013 Mar; 35(3):241-54. PubMed ID: 23575530
[TBL] [Abstract][Full Text] [Related]
16. Inhibition of histone methyltransferase SETD8 represses DNA virus replication.
Chen L; Yang C; Tang SB; Long QY; Chen JD; Wu M; Li LY
Cell Insight; 2022 Jun; 1(3):100033. PubMed ID: 37193046
[TBL] [Abstract][Full Text] [Related]
17. The histone methyltransferase Setd8 acts in concert with c-Myc and is required to maintain skin.
Driskell I; Oda H; Blanco S; Nascimento E; Humphreys P; Frye M
EMBO J; 2012 Feb; 31(3):616-29. PubMed ID: 22117221
[TBL] [Abstract][Full Text] [Related]
18. Structure-Based Design of a Covalent Inhibitor of the SET Domain-Containing Protein 8 (SETD8) Lysine Methyltransferase.
Butler KV; Ma A; Yu W; Li F; Tempel W; Babault N; Pittella-Silva F; Shao J; Wang J; Luo M; Vedadi M; Brown PJ; Arrowsmith CH; Jin J
J Med Chem; 2016 Nov; 59(21):9881-9889. PubMed ID: 27804297
[TBL] [Abstract][Full Text] [Related]
19. The SET8 H4K20 protein lysine methyltransferase has a long recognition sequence covering seven amino acid residues.
Kudithipudi S; Dhayalan A; Kebede AF; Jeltsch A
Biochimie; 2012 Nov; 94(11):2212-8. PubMed ID: 22583696
[TBL] [Abstract][Full Text] [Related]
20. Histone lysine methyltransferase SETD8 promotes carcinogenesis by deregulating PCNA expression.
Takawa M; Cho HS; Hayami S; Toyokawa G; Kogure M; Yamane Y; Iwai Y; Maejima K; Ueda K; Masuda A; Dohmae N; Field HI; Tsunoda T; Kobayashi T; Akasu T; Sugiyama M; Ohnuma S; Atomi Y; Ponder BA; Nakamura Y; Hamamoto R
Cancer Res; 2012 Jul; 72(13):3217-27. PubMed ID: 22556262
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]