331 related articles for article (PubMed ID: 25575161)
21. 3D structure and allosteric modulation of the transmembrane domain of pentameric ligand-gated ion channels.
Baenziger JE; Corringer PJ
Neuropharmacology; 2011 Jan; 60(1):116-25. PubMed ID: 20713066
[TBL] [Abstract][Full Text] [Related]
22. 2-Guanidine-4-methylquinazoline acts as a novel competitive antagonist of A type γ-aminobutyric acid receptors.
Xiao X; Zhu MX; Xu TL
Neuropharmacology; 2013 Dec; 75():126-37. PubMed ID: 23916476
[TBL] [Abstract][Full Text] [Related]
23. Neurosteroids allosterically modulate binding of the anesthetic etomidate to gamma-aminobutyric acid type A receptors.
Li GD; Chiara DC; Cohen JB; Olsen RW
J Biol Chem; 2009 May; 284(18):11771-5. PubMed ID: 19282280
[TBL] [Abstract][Full Text] [Related]
24. Photoaffinity labeling the propofol binding site in GLIC.
Chiara DC; Gill JF; Chen Q; Tillman T; Dailey WP; Eckenhoff RG; Xu Y; Tang P; Cohen JB
Biochemistry; 2014 Jan; 53(1):135-42. PubMed ID: 24341978
[TBL] [Abstract][Full Text] [Related]
25. A residue in loop 9 of the beta2-subunit stabilizes the closed state of the GABAA receptor.
Williams CA; Bell SV; Jenkins A
J Biol Chem; 2010 Mar; 285(10):7281-7. PubMed ID: 20007704
[TBL] [Abstract][Full Text] [Related]
26. Functional asymmetry of the conserved cystine loops in alphabetagamma GABA A receptors revealed by the response to GABA activation and drug potentiation.
Tierney ML; Luu T; Gage PW
Int J Biochem Cell Biol; 2008; 40(5):968-79. PubMed ID: 18083058
[TBL] [Abstract][Full Text] [Related]
27. The interaction of general anaesthetics with recombinant GABAA and glycine receptors expressed in Xenopus laevis oocytes: a comparative study.
Pistis M; Belelli D; Peters JA; Lambert JJ
Br J Pharmacol; 1997 Dec; 122(8):1707-19. PubMed ID: 9422818
[TBL] [Abstract][Full Text] [Related]
28. Modeling the closed and open state conformations of the GABA(A) ion channel--plausible structural insights for channel gating.
Vijayan RS; Trivedi N; Roy SN; Bera I; Manoharan P; Payghan PV; Bhattacharyya D; Ghoshal N
J Chem Inf Model; 2012 Nov; 52(11):2958-69. PubMed ID: 23116339
[TBL] [Abstract][Full Text] [Related]
29. Functional characterization of neurotransmitter activation and modulation in a nematode model ligand-gated ion channel.
Heusser SA; Yoluk Ö; Klement G; Riederer EA; Lindahl E; Howard RJ
J Neurochem; 2016 Jul; 138(2):243-53. PubMed ID: 27102368
[TBL] [Abstract][Full Text] [Related]
30. Propofol Is an Allosteric Agonist with Multiple Binding Sites on Concatemeric Ternary GABA
Shin DJ; Germann AL; Johnson AD; Forman SA; Steinbach JH; Akk G
Mol Pharmacol; 2018 Feb; 93(2):178-189. PubMed ID: 29192122
[TBL] [Abstract][Full Text] [Related]
31. A conserved tyrosine in the beta2 subunit M4 segment is a determinant of gamma-aminobutyric acid type A receptor sensitivity to propofol.
Richardson JE; Garcia PS; O'Toole KK; Derry JM; Bell SV; Jenkins A
Anesthesiology; 2007 Sep; 107(3):412-8. PubMed ID: 17721243
[TBL] [Abstract][Full Text] [Related]
32. Functional validation of virtual screening for novel agents with general anesthetic action at ligand-gated ion channels.
Heusser SA; Howard RJ; Borghese CM; Cullins MA; Broemstrup T; Lee US; Lindahl E; Carlsson J; Harris RA
Mol Pharmacol; 2013 Nov; 84(5):670-8. PubMed ID: 23950219
[TBL] [Abstract][Full Text] [Related]
33. Homomeric beta 1 gamma-aminobutyric acid A receptor-ion channels: evaluation of pharmacological and physiological properties.
Krishek BJ; Moss SJ; Smart TG
Mol Pharmacol; 1996 Mar; 49(3):494-504. PubMed ID: 8643089
[TBL] [Abstract][Full Text] [Related]
34. A unitary anesthetic binding site at high resolution.
Vedula LS; Brannigan G; Economou NJ; Xi J; Hall MA; Liu R; Rossi MJ; Dailey WP; Grasty KC; Klein ML; Eckenhoff RG; Loll PJ
J Biol Chem; 2009 Sep; 284(36):24176-84. PubMed ID: 19605349
[TBL] [Abstract][Full Text] [Related]
35. Evaluation of a proposed mechanism of ligand-gated ion channel activation in the GABAA and glycine receptors.
Kash TL; Kim T; Trudell JR; Harrison NL
Neurosci Lett; 2004 Nov; 371(2-3):230-4. PubMed ID: 15519763
[TBL] [Abstract][Full Text] [Related]
36. The Cys-loop superfamily of ligand-gated ion channels: the impact of receptor structure on function.
Connolly CN; Wafford KA
Biochem Soc Trans; 2004 Jun; 32(Pt3):529-34. PubMed ID: 15157178
[TBL] [Abstract][Full Text] [Related]
37. Binding modes of noncompetitive GABA-channel blockers revisited using engineered affinity-labeling reactions combined with new docking studies.
Charon S; Taly A; Rodrigo J; Perret P; Goeldner M
J Agric Food Chem; 2011 Apr; 59(7):2803-7. PubMed ID: 20839772
[TBL] [Abstract][Full Text] [Related]
38. Inverse effects on gating and modulation caused by a mutation in the M2-M3 Linker of the GABA(A) receptor gamma subunit.
O'Shea SM; Williams CA; Jenkins A
Mol Pharmacol; 2009 Sep; 76(3):641-51. PubMed ID: 19553237
[TBL] [Abstract][Full Text] [Related]
39. Halothane and propofol modulation of gamma-aminobutyric acidA receptor single-channel currents.
Kitamura A; Sato R; Marszalec W; Yeh JZ; Ogawa R; Narahashi T
Anesth Analg; 2004 Aug; 99(2):409-15, table of contents. PubMed ID: 15271715
[TBL] [Abstract][Full Text] [Related]
40. A potent photoreactive general anesthetic with novel binding site selectivity for GABA
Shalabi AR; Yu Z; Zhou X; Jounaidi Y; Chen H; Dai J; Kent DE; Feng HJ; Forman SA; Cohen JB; Bruzik KS; Miller KW
Eur J Med Chem; 2020 May; 194():112261. PubMed ID: 32247113
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
