298 related articles for article (PubMed ID: 25771108)
1. Synthesis, crystal structure and biological evaluation of substituted quinazolinone benzoates as novel antituberculosis agents targeting acetohydroxyacid synthase.
Lu W; Baig IA; Sun HJ; Cui CJ; Guo R; Jung IP; Wang D; Dong M; Yoon MY; Wang JG
Eur J Med Chem; 2015 Apr; 94():298-305. PubMed ID: 25771108
[TBL] [Abstract][Full Text] [Related]
2. Discovery of novel acetohydroxyacid synthase inhibitors as active agents against Mycobacterium tuberculosis by virtual screening and bioassay.
Wang D; Zhu X; Cui C; Dong M; Jiang H; Li Z; Liu Z; Zhu W; Wang JG
J Chem Inf Model; 2013 Feb; 53(2):343-53. PubMed ID: 23316686
[TBL] [Abstract][Full Text] [Related]
3. Development of potent chemical antituberculosis agents targeting Mycobacterium tuberculosis acetohydroxyacid synthase.
Jung IP; Ha NR; Lee SC; Ryoo SW; Yoon MY
Int J Antimicrob Agents; 2016 Sep; 48(3):247-58. PubMed ID: 27451857
[TBL] [Abstract][Full Text] [Related]
4. Development of ssDNA aptamers as potent inhibitors of Mycobacterium tuberculosis acetohydroxyacid synthase.
Baig IA; Moon JY; Lee SC; Ryoo SW; Yoon MY
Biochim Biophys Acta; 2015 Oct; 1854(10 Pt A):1338-50. PubMed ID: 25988243
[TBL] [Abstract][Full Text] [Related]
5. In vitro and ex vivo activity of new derivatives of acetohydroxyacid synthase inhibitors against Mycobacterium tuberculosis and non-tuberculous mycobacteria.
Sohn H; Lee KS; Ko YK; Ryu JW; Woo JC; Koo DW; Shin SJ; Ahn SJ; Shin AR; Song CH; Jo EK; Park JK; Kim HJ
Int J Antimicrob Agents; 2008 Jun; 31(6):567-71. PubMed ID: 18337064
[TBL] [Abstract][Full Text] [Related]
6. Characterization of acetohydroxyacid synthase from Mycobacterium tuberculosis and the identification of its new inhibitor from the screening of a chemical library.
Choi KJ; Yu YG; Hahn HG; Choi JD; Yoon MY
FEBS Lett; 2005 Aug; 579(21):4903-10. PubMed ID: 16111681
[TBL] [Abstract][Full Text] [Related]
7. Rational design based on bioactive conformation analysis of pyrimidinylbenzoates as acetohydroxyacid synthase inhibitors by integrating molecular docking, CoMFA, CoMSIA, and DFT calculations.
He YZ; Li YX; Zhu XL; Xi Z; Niu C; Wan J; Zhang L; Yang GF
J Chem Inf Model; 2007; 47(6):2335-44. PubMed ID: 17887745
[TBL] [Abstract][Full Text] [Related]
8. Evaluation of the in vitro and intracellular efficacy of new monosubstituted sulfonylureas against extensively drug-resistant tuberculosis.
Wang D; Pan L; Cao G; Lei H; Meng X; He J; Dong M; Li Z; Liu Z
Int J Antimicrob Agents; 2012 Nov; 40(5):463-6. PubMed ID: 22867883
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and biological evaluation of phaitanthrin congeners as anti-mycobacterial agents.
Kamal A; Reddy BV; Sridevi B; Ravikumar A; Venkateswarlu A; Sravanthi G; Sridevi JP; Yogeeswari P; Sriram D
Bioorg Med Chem Lett; 2015 Sep; 25(18):3867-72. PubMed ID: 26253635
[TBL] [Abstract][Full Text] [Related]
10. Sulfonylureas have antifungal activity and are potent inhibitors of Candida albicans acetohydroxyacid synthase.
Lee YT; Cui CJ; Chow EW; Pue N; Lonhienne T; Wang JG; Fraser JA; Guddat LW
J Med Chem; 2013 Jan; 56(1):210-9. PubMed ID: 23237384
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and biological evaluation of nonsymmetrical aromatic disulfides as novel inhibitors of acetohydroxyacid synthase.
Li ZS; Wang WM; Lu W; Niu CW; Li YH; Li ZM; Wang JG
Bioorg Med Chem Lett; 2013 Jul; 23(13):3723-7. PubMed ID: 23726033
[TBL] [Abstract][Full Text] [Related]
12. Identification of some novel AHAS inhibitors via molecular docking and virtual screening approach.
Wang JG; Xiao YJ; Li YH; Ma Y; Li ZM
Bioorg Med Chem; 2007 Jan; 15(1):374-80. PubMed ID: 17049866
[TBL] [Abstract][Full Text] [Related]
13. Identification of inhibitors targeting polyketide synthase 13 of Mycobacterium tuberculosis as antituberculosis drug leads.
Wang X; Zhao W; Wang B; Ding W; Guo H; Zhao H; Meng J; Liu S; Lu Y; Liu Y; Zhang D
Bioorg Chem; 2021 Sep; 114():105110. PubMed ID: 34175719
[TBL] [Abstract][Full Text] [Related]
14. Chemical synthesis, in vitro acetohydroxyacid synthase (AHAS) inhibition, herbicidal activity, and computational studies of isatin derivatives.
Wang J; Tan H; Li Y; Ma Y; Li Z; Guddat LW
J Agric Food Chem; 2011 Sep; 59(18):9892-900. PubMed ID: 21838297
[TBL] [Abstract][Full Text] [Related]
15. Novel amide and sulphonamide derivatives of 6-(piperazin-1-yl)phenanthridine as potent Mycobacterium tuberculosis H37Rv inhibitors.
Naidu KM; Nagesh HN; Singh M; Sriram D; Yogeeswari P; Gowri Chandra Sekhar KV
Eur J Med Chem; 2015 Mar; 92():415-26. PubMed ID: 25590862
[TBL] [Abstract][Full Text] [Related]
16. In vitro efficacy of acetohydroxyacid synthase inhibitors against clinical strains of Mycobacterium tuberculosis isolated from a hospital in Beijing, China.
Dong M; Wang D; Jiang Y; Zhao L; Yang C; Wu C
Saudi Med J; 2011 Nov; 32(11):1122-6. PubMed ID: 22057598
[TBL] [Abstract][Full Text] [Related]
17. Design, synthesis and molecular docking study of novel triazole-quinazolinone hybrids as antimalarial and antitubercular agents.
Mhetre UV; Haval NB; Bondle GM; Rathod SS; Choudhari PB; Kumari J; Sriram D; Haval KP
Bioorg Med Chem Lett; 2024 Aug; 108():129800. PubMed ID: 38763480
[TBL] [Abstract][Full Text] [Related]
18. Design and synthesis of 11α-substituted bile acid derivatives as potential anti-tuberculosis agents.
Pore VS; Divse JM; Charolkar CR; Nawale LU; Khedkar VM; Sarkar D
Bioorg Med Chem Lett; 2015 Oct; 25(19):4185-90. PubMed ID: 26299346
[TBL] [Abstract][Full Text] [Related]
19. Development of novel tetrahydrothieno[2,3-c]pyridine-3-carboxamide based Mycobacterium tuberculosis pantothenate synthetase inhibitors: molecular hybridization from known antimycobacterial leads.
Samala G; Devi PB; Nallangi R; Sridevi JP; Saxena S; Yogeeswari P; Sriram D
Bioorg Med Chem; 2014 Mar; 22(6):1938-47. PubMed ID: 24565972
[TBL] [Abstract][Full Text] [Related]
20. Discovery and development of novel salicylate synthase (MbtI) furanic inhibitors as antitubercular agents.
Chiarelli LR; Mori M; Barlocco D; Beretta G; Gelain A; Pini E; Porcino M; Mori G; Stelitano G; Costantino L; Lapillo M; Bonanni D; Poli G; Tuccinardi T; Villa S; Meneghetti F
Eur J Med Chem; 2018 Jul; 155():754-763. PubMed ID: 29940465
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]