224 related articles for article (PubMed ID: 25792505)
1. Biological evaluation and molecular modelling study of thiosemicarbazide derivatives as bacterial type IIA topoisomerases inhibitors.
Paneth A; Stączek P; Plech T; Strzelczyk A; Dzitko K; Wujec M; Kuśmierz E; Kosikowska U; Grzegorczyk A; Paneth P
J Enzyme Inhib Med Chem; 2016; 31(1):14-22. PubMed ID: 25792505
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and structure-activity relationship studies of 4-arylthiosemicarbazides as topoisomerase IV inhibitors with Gram-positive antibacterial activity. Search for molecular basis of antibacterial activity of thiosemicarbazides.
Siwek A; Stączek P; Stefańska J
Eur J Med Chem; 2011 Nov; 46(11):5717-26. PubMed ID: 21978836
[TBL] [Abstract][Full Text] [Related]
3. Synthesis, and antibacterial activity of novel 4,5-dihydro-1H-pyrazole derivatives as DNA gyrase inhibitors.
Liu JJ; Sun J; Fang YB; Yang YA; Jiao RH; Zhu HL
Org Biomol Chem; 2014 Feb; 12(6):998-1008. PubMed ID: 24382549
[TBL] [Abstract][Full Text] [Related]
4. Thiosemicarbazide Derivatives Decrease the ATPase Activity of
Kowalczyk A; Paneth A; Trojanowski D; Paneth P; Zakrzewska-Czerwińska J; Stączek P
Int J Mol Sci; 2021 Apr; 22(8):. PubMed ID: 33918623
[TBL] [Abstract][Full Text] [Related]
5. New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity.
Durcik M; Lovison D; Skok Ž; Durante Cruz C; Tammela P; Tomašič T; Benedetto Tiz D; Draskovits G; Nyerges Á; Pál C; Ilaš J; Peterlin Mašič L; Kikelj D; Zidar N
Eur J Med Chem; 2018 Jun; 154():117-132. PubMed ID: 29778894
[TBL] [Abstract][Full Text] [Related]
6. Novel 3-fluoro-6-methoxyquinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV.
Mitton-Fry MJ; Brickner SJ; Hamel JC; Barham R; Brennan L; Casavant JM; Ding X; Finegan S; Hardink J; Hoang T; Huband MD; Maloney M; Marfat A; McCurdy SP; McLeod D; Subramanyam C; Plotkin M; Reilly U; Schafer J; Stone GG; Uccello DP; Wisialowski T; Yoon K; Zaniewski R; Zook C
Bioorg Med Chem Lett; 2017 Aug; 27(15):3353-3358. PubMed ID: 28610977
[TBL] [Abstract][Full Text] [Related]
7. Synergistic Effects of Thiosemicarbazides with Clinical Drugs against
Chudzik-Rząd B; Malm A; Trotsko N; Wujec M; Plech T; Paneth A
Molecules; 2020 May; 25(10):. PubMed ID: 32422899
[TBL] [Abstract][Full Text] [Related]
8. Design, synthesis and biological evaluation of α-substituted isonipecotic acid benzothiazole analogues as potent bacterial type II topoisomerase inhibitors.
Axford LC; Agarwal PK; Anderson KH; Andrau LN; Atherall J; Barker S; Bennett JM; Blair M; Collins I; Czaplewski LG; Davies DT; Gannon CT; Kumar D; Lancett P; Logan A; Lunniss CJ; Mitchell DR; Offermann DA; Palmer JT; Palmer N; Pitt GR; Pommier S; Price D; Narasinga Rao B; Saxena R; Shukla T; Singh AK; Singh M; Srivastava A; Steele C; Stokes NR; Thomaides-Brears HB; Tyndall EM; Watson D; Haydon DJ
Bioorg Med Chem Lett; 2013 Dec; 23(24):6598-603. PubMed ID: 24239017
[TBL] [Abstract][Full Text] [Related]
9. Design, Synthesis, and Evaluation of Novel Tyrosine-Based DNA Gyrase B Inhibitors.
Cotman AE; Trampuž M; Brvar M; Kikelj D; Ilaš J; Peterlin-Mašič L; Montalvão S; Tammela P; Frlan R
Arch Pharm (Weinheim); 2017 Aug; 350(8):. PubMed ID: 28621824
[TBL] [Abstract][Full Text] [Related]
10. N-thiadiazole-4-hydroxy-2-quinolone-3-carboxamides bearing heteroaromatic rings as novel antibacterial agents: Design, synthesis, biological evaluation and target identification.
Xue W; Li X; Ma G; Zhang H; Chen Y; Kirchmair J; Xia J; Wu S
Eur J Med Chem; 2020 Feb; 188():112022. PubMed ID: 31901744
[TBL] [Abstract][Full Text] [Related]
11. Design, synthesis and biological evaluation of 4-benzoyl-1-dichlorobenzoylthiosemicarbazides as potent Gram-positive antibacterial agents.
Paneth A; Plech T; Kaproń B; Hagel D; Kosikowska U; Kuśmierz E; Dzitko K; Paneth P
J Enzyme Inhib Med Chem; 2016; 31(3):434-40. PubMed ID: 25897586
[TBL] [Abstract][Full Text] [Related]
12. Dual inhibition of Staphylococcus aureus DNA gyrase and topoisomerase IV activity by phenylalanine-derived (Z)-5-arylmethylidene rhodanines.
Werner MM; Patel BA; Talele TT; Ashby CR; Li Z; Zauhar RJ
Bioorg Med Chem; 2015 Sep; 23(18):6125-37. PubMed ID: 26320664
[TBL] [Abstract][Full Text] [Related]
13. Novel quinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV.
Mitton-Fry MJ; Brickner SJ; Hamel JC; Brennan L; Casavant JM; Chen M; Chen T; Ding X; Driscoll J; Hardink J; Hoang T; Hua E; Huband MD; Maloney M; Marfat A; McCurdy SP; McLeod D; Plotkin M; Reilly U; Robinson S; Schafer J; Shepard RM; Smith JF; Stone GG; Subramanyam C; Yoon K; Yuan W; Zaniewski RP; Zook C
Bioorg Med Chem Lett; 2013 May; 23(10):2955-61. PubMed ID: 23566517
[TBL] [Abstract][Full Text] [Related]
14. Dual Antibacterial and Anticancer Activity of 4-Benzoyl-1-dichlorobenzoylthiosemicarbazide Derivatives.
Kapron B; Czarnomysy R; Paneth A; Wujec M; Bielawski K; Bielawska A; Swiatek L; Rajtar B; Polz-Dacewicz M; Plech T
Anticancer Agents Med Chem; 2018; 18(4):529-540. PubMed ID: 29065843
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis, and biological evaluation of 1-ethyl-3-(thiazol-2-yl)urea derivatives as Escherichia coli DNA gyrase inhibitors.
Tomašič T; Barančoková M; Zidar N; Ilaš J; Tammela P; Kikelj D
Arch Pharm (Weinheim); 2018 Jan; 351(1):. PubMed ID: 29239018
[TBL] [Abstract][Full Text] [Related]
16. Molecular docking, discovery, synthesis, and pharmacological properties of new 6-substituted-2-(3-phenoxyphenyl)-4-phenyl quinoline derivatives; an approach to developing potent DNA gyrase inhibitors/antibacterial agents.
Alagumuthu M; Arumugam S
Bioorg Med Chem; 2017 Feb; 25(4):1448-1455. PubMed ID: 28094220
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and Evaluation of N-Phenylpyrrolamides as DNA Gyrase B Inhibitors.
Durcik M; Tammela P; Barančoková M; Tomašič T; Ilaš J; Kikelj D; Zidar N
ChemMedChem; 2018 Jan; 13(2):186-198. PubMed ID: 29206345
[TBL] [Abstract][Full Text] [Related]
18. Design, synthesis and molecular modeling studies of new series of s-triazine derivatives as antimicrobial agents against multi-drug resistant clinical isolates.
Haiba NS; Khalil HH; Moniem MA; El-Wakil MH; Bekhit AA; Khattab SN
Bioorg Chem; 2019 Aug; 89():103013. PubMed ID: 31174040
[TBL] [Abstract][Full Text] [Related]
19. Probing linker design in citric acid-ciprofloxacin conjugates.
Milner SJ; Snelling AM; Kerr KG; Abd-El-Aziz A; Thomas GH; Hubbard RE; Routledge A; Duhme-Klair AK
Bioorg Med Chem; 2014 Aug; 22(16):4499-505. PubMed ID: 24794750
[TBL] [Abstract][Full Text] [Related]
20. Design, green one-pot synthesis and molecular docking study of novel N,N-bis(cyanoacetyl)hydrazines and bis-coumarins as effective inhibitors of DNA gyrase and topoisomerase IV.
Metwally NH; Abdallah SO; Mohsen MMA
Bioorg Chem; 2020 Apr; 97():103672. PubMed ID: 32145481
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]