These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
514 related articles for article (PubMed ID: 25856009)
1. Discovery of I-BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition. Theodoulou NH; Bamborough P; Bannister AJ; Becher I; Bit RA; Che KH; Chung CW; Dittmann A; Drewes G; Drewry DH; Gordon L; Grandi P; Leveridge M; Lindon M; Michon AM; Molnar J; Robson SC; Tomkinson NC; Kouzarides T; Prinjha RK; Humphreys PG J Med Chem; 2016 Feb; 59(4):1425-39. PubMed ID: 25856009 [TBL] [Abstract][Full Text] [Related]
2. Research progress of selective small molecule bromodomain-containing protein 9 inhibitors. Hui M; Jian Z; Peiyuan Z; Zhenwei W; Huibin Z Future Med Chem; 2018 Apr; 10(8):895-906. PubMed ID: 29620420 [TBL] [Abstract][Full Text] [Related]
3. Inhibition of bromodomain-containing protein 9 for the prevention of epigenetically-defined drug resistance. Crawford TD; Vartanian S; Côté A; Bellon S; Duplessis M; Flynn EM; Hewitt M; Huang HR; Kiefer JR; Murray J; Nasveschuk CG; Pardo E; Romero FA; Sandy P; Tang Y; Taylor AM; Tsui V; Wang J; Wang S; Zawadzke L; Albrecht BK; Magnuson SR; Cochran AG; Stokoe D Bioorg Med Chem Lett; 2017 Aug; 27(15):3534-3541. PubMed ID: 28606761 [TBL] [Abstract][Full Text] [Related]
4. Application of Atypical Acetyl-lysine Methyl Mimetics in the Development of Selective Inhibitors of the Bromodomain-Containing Protein 7 (BRD7)/Bromodomain-Containing Protein 9 (BRD9) Bromodomains. Clegg MA; Bamborough P; Chung CW; Craggs PD; Gordon L; Grandi P; Leveridge M; Lindon M; Liwicki GM; Michon AM; Molnar J; Rioja I; Soden PE; Theodoulou NH; Werner T; Tomkinson NCO; Prinjha RK; Humphreys PG J Med Chem; 2020 Jun; 63(11):5816-5840. PubMed ID: 32410449 [TBL] [Abstract][Full Text] [Related]
5. Molecular mechanism study of several inhibitors binding to BRD9 bromodomain based on molecular simulations. Song LT; Tu J; Liu RR; Zhu M; Meng YJ; Zhai HL J Biomol Struct Dyn; 2019 Jul; 37(11):2970-2979. PubMed ID: 30058436 [TBL] [Abstract][Full Text] [Related]
6. Structural Basis of Inhibitor Selectivity in the BRD7/9 Subfamily of Bromodomains. Karim RM; Chan A; Zhu JY; Schönbrunn E J Med Chem; 2020 Mar; 63(6):3227-3237. PubMed ID: 32091206 [TBL] [Abstract][Full Text] [Related]
7. An Advanced Tool To Interrogate BRD9. Karim RM; Schönbrunn E J Med Chem; 2016 May; 59(10):4459-61. PubMed ID: 27120693 [TBL] [Abstract][Full Text] [Related]
8. Covalent-Fragment Screening of BRD4 Identifies a Ligandable Site Orthogonal to the Acetyl-Lysine Binding Sites. Olp MD; Sprague DJ; Goetz CJ; Kathman SG; Wynia-Smith SL; Shishodia S; Summers SB; Xu Z; Statsyuk AV; Smith BC ACS Chem Biol; 2020 Apr; 15(4):1036-1049. PubMed ID: 32149490 [TBL] [Abstract][Full Text] [Related]
9. Disrupting Acetyl-Lysine Recognition: Progress in the Development of Bromodomain Inhibitors. Romero FA; Taylor AM; Crawford TD; Tsui V; Côté A; Magnuson S J Med Chem; 2016 Feb; 59(4):1271-98. PubMed ID: 26572217 [TBL] [Abstract][Full Text] [Related]
10. Discovery of Benzo[ Jiang F; Hu Q; Zhang Z; Li H; Li H; Zhang D; Li H; Ma Y; Xu J; Chen H; Cui Y; Zhi Y; Zhang Y; Xu J; Zhu J; Lu T; Chen Y J Med Chem; 2019 Dec; 62(24):11080-11107. PubMed ID: 31789032 [TBL] [Abstract][Full Text] [Related]
11. Discovery of Tetrahydroquinoxalines as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the Second Bromodomain. Law RP; Atkinson SJ; Bamborough P; Chung CW; Demont EH; Gordon LJ; Lindon M; Prinjha RK; Watson AJB; Hirst DJ J Med Chem; 2018 May; 61(10):4317-4334. PubMed ID: 29656650 [TBL] [Abstract][Full Text] [Related]
12. NMR Fragment Screening Hit Induces Plasticity of BRD7/9 Bromodomains. Wang N; Li F; Bao H; Li J; Wu J; Ruan K Chembiochem; 2016 Aug; 17(15):1456-63. PubMed ID: 27194508 [TBL] [Abstract][Full Text] [Related]
13. LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor. Clark PG; Vieira LC; Tallant C; Fedorov O; Singleton DC; Rogers CM; Monteiro OP; Bennett JM; Baronio R; Müller S; Daniels DL; Méndez J; Knapp S; Brennan PE; Dixon DJ Angew Chem Int Ed Engl; 2015 May; 54(21):6217-21. PubMed ID: 25864491 [TBL] [Abstract][Full Text] [Related]
14. Design, synthesis and biological evaluation of imidazo[1,5-a]pyrazin-8(7H)-one derivatives as BRD9 inhibitors. Zheng P; Zhang J; Ma H; Yuan X; Chen P; Zhou J; Zhang H Bioorg Med Chem; 2019 Apr; 27(7):1391-1404. PubMed ID: 30824168 [TBL] [Abstract][Full Text] [Related]
15. Potent and selective bivalent inhibitors of BET bromodomains. Waring MJ; Chen H; Rabow AA; Walker G; Bobby R; Boiko S; Bradbury RH; Callis R; Clark E; Dale I; Daniels DL; Dulak A; Flavell L; Holdgate G; Jowitt TA; Kikhney A; McAlister M; Méndez J; Ogg D; Patel J; Petteruti P; Robb GR; Robers MB; Saif S; Stratton N; Svergun DI; Wang W; Whittaker D; Wilson DM; Yao Y Nat Chem Biol; 2016 Dec; 12(12):1097-1104. PubMed ID: 27775716 [TBL] [Abstract][Full Text] [Related]
16. Insight into selective mechanism of class of I-BRD9 inhibitors toward BRD9 based on molecular dynamics simulations. Su J; Liu X; Zhang S; Yan F; Zhang Q; Chen J Chem Biol Drug Des; 2019 Feb; 93(2):163-176. PubMed ID: 30225973 [TBL] [Abstract][Full Text] [Related]
17. Epigenetic modulation by targeting bromodomain containing protein 9 (BRD9): Its therapeutic potential and selective inhibition. Ali MM; Naz S; Ashraf S; Knapp S; Ul-Haq Z Int J Biol Macromol; 2023 Mar; 230():123428. PubMed ID: 36709803 [TBL] [Abstract][Full Text] [Related]
18. Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor. Martin LJ; Koegl M; Bader G; Cockcroft XL; Fedorov O; Fiegen D; Gerstberger T; Hofmann MH; Hohmann AF; Kessler D; Knapp S; Knesl P; Kornigg S; Müller S; Nar H; Rogers C; Rumpel K; Schaaf O; Steurer S; Tallant C; Vakoc CR; Zeeb M; Zoephel A; Pearson M; Boehmelt G; McConnell D J Med Chem; 2016 May; 59(10):4462-75. PubMed ID: 26914985 [TBL] [Abstract][Full Text] [Related]
19. 9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain. Picaud S; Strocchia M; Terracciano S; Lauro G; Mendez J; Daniels DL; Riccio R; Bifulco G; Bruno I; Filippakopoulos P J Med Chem; 2015 Mar; 58(6):2718-36. PubMed ID: 25703523 [TBL] [Abstract][Full Text] [Related]
20. Identification of Selective BRD9 Inhibitor via Integrated Computational Approach. Ali MM; Ashraf S; Nure-E-Alam M; Qureshi U; Khan KM; Ul-Haq Z Int J Mol Sci; 2022 Nov; 23(21):. PubMed ID: 36362300 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]