These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
3. ISRIB Blunts the Integrated Stress Response by Allosterically Antagonising the Inhibitory Effect of Phosphorylated eIF2 on eIF2B. Zyryanova AF; Kashiwagi K; Rato C; Harding HP; Crespillo-Casado A; Perera LA; Sakamoto A; Nishimoto M; Yonemochi M; Shirouzu M; Ito T; Ron D Mol Cell; 2021 Jan; 81(1):88-103.e6. PubMed ID: 33220178 [TBL] [Abstract][Full Text] [Related]
4. Structure of the nucleotide exchange factor eIF2B reveals mechanism of memory-enhancing molecule. Tsai JC; Miller-Vedam LE; Anand AA; Jaishankar P; Nguyen HC; Renslo AR; Frost A; Walter P Science; 2018 Mar; 359(6383):. PubMed ID: 29599213 [TBL] [Abstract][Full Text] [Related]
5. Structural insights into ISRIB, a memory-enhancing inhibitor of the integrated stress response. Anand AA; Walter P FEBS J; 2020 Jan; 287(2):239-245. PubMed ID: 31550413 [TBL] [Abstract][Full Text] [Related]
6. Pharmacological dimerization and activation of the exchange factor eIF2B antagonizes the integrated stress response. Sidrauski C; Tsai JC; Kampmann M; Hearn BR; Vedantham P; Jaishankar P; Sokabe M; Mendez AS; Newton BW; Tang EL; Verschueren E; Johnson JR; Krogan NJ; Fraser CS; Weissman JS; Renslo AR; Walter P Elife; 2015 Apr; 4():e07314. PubMed ID: 25875391 [TBL] [Abstract][Full Text] [Related]
7. Binding of ISRIB reveals a regulatory site in the nucleotide exchange factor eIF2B. Zyryanova AF; Weis F; Faille A; Alard AA; Crespillo-Casado A; Sekine Y; Harding HP; Allen F; Parts L; Fromont C; Fischer PM; Warren AJ; Ron D Science; 2018 Mar; 359(6383):1533-1536. PubMed ID: 29599245 [TBL] [Abstract][Full Text] [Related]
8. Small molecule ISRIB suppresses the integrated stress response within a defined window of activation. Rabouw HH; Langereis MA; Anand AA; Visser LJ; de Groot RJ; Walter P; van Kuppeveld FJM Proc Natl Acad Sci U S A; 2019 Feb; 116(6):2097-2102. PubMed ID: 30674674 [TBL] [Abstract][Full Text] [Related]
9. Vanishing white matter: deregulated integrated stress response as therapy target. Abbink TEM; Wisse LE; Jaku E; Thiecke MJ; Voltolini-González D; Fritsen H; Bobeldijk S; Ter Braak TJ; Polder E; Postma NL; Bugiani M; Struijs EA; Verheijen M; Straat N; van der Sluis S; Thomas AAM; Molenaar D; van der Knaap MS Ann Clin Transl Neurol; 2019 Aug; 6(8):1407-1422. PubMed ID: 31402619 [TBL] [Abstract][Full Text] [Related]
10. The small molecule ISRIB reverses the effects of eIF2α phosphorylation on translation and stress granule assembly. Sidrauski C; McGeachy AM; Ingolia NT; Walter P Elife; 2015 Feb; 4():. PubMed ID: 25719440 [TBL] [Abstract][Full Text] [Related]
11. Paradoxical Sensitivity to an Integrated Stress Response Blocking Mutation in Vanishing White Matter Cells. Sekine Y; Zyryanova A; Crespillo-Casado A; Amin-Wetzel N; Harding HP; Ron D PLoS One; 2016; 11(11):e0166278. PubMed ID: 27812215 [TBL] [Abstract][Full Text] [Related]
12. The small molecule ISRIB rescues the stability and activity of Vanishing White Matter Disease eIF2B mutant complexes. Wong YL; LeBon L; Edalji R; Lim HB; Sun C; Sidrauski C Elife; 2018 Feb; 7():. PubMed ID: 29489452 [TBL] [Abstract][Full Text] [Related]
13. The beta/Gcd7 subunit of eukaryotic translation initiation factor 2B (eIF2B), a guanine nucleotide exchange factor, is crucial for binding eIF2 in vivo. Dev K; Qiu H; Dong J; Zhang F; Barthlme D; Hinnebusch AG Mol Cell Biol; 2010 Nov; 30(21):5218-33. PubMed ID: 20805354 [TBL] [Abstract][Full Text] [Related]
14. Identification of domains and residues within the epsilon subunit of eukaryotic translation initiation factor 2B (eIF2Bepsilon) required for guanine nucleotide exchange reveals a novel activation function promoted by eIF2B complex formation. Gomez E; Pavitt GD Mol Cell Biol; 2000 Jun; 20(11):3965-76. PubMed ID: 10805739 [TBL] [Abstract][Full Text] [Related]
15. Suppression of MEHMO Syndrome Mutation in eIF2 by Small Molecule ISRIB. Young-Baird SK; Lourenço MB; Elder MK; Klann E; Liebau S; Dever TE Mol Cell; 2020 Feb; 77(4):875-886.e7. PubMed ID: 31836389 [TBL] [Abstract][Full Text] [Related]
16. A point mutation in the nucleotide exchange factor eIF2B constitutively activates the integrated stress response by allosteric modulation. Boone M; Wang L; Lawrence RE; Frost A; Walter P; Schoof M Elife; 2022 Apr; 11():. PubMed ID: 35416150 [TBL] [Abstract][Full Text] [Related]
17. Cellular eIF2B subunit localization: implications for the integrated stress response and its control by small molecule drugs. Hodgson RE; Varanda BA; Ashe MP; Allen KE; Campbell SG Mol Biol Cell; 2019 Apr; 30(8):942-958. PubMed ID: 30726166 [TBL] [Abstract][Full Text] [Related]
18. Small molecule cognitive enhancer reverses age-related memory decline in mice. Krukowski K; Nolan A; Frias ES; Boone M; Ureta G; Grue K; Paladini MS; Elizarraras E; Delgado L; Bernales S; Walter P; Rosi S Elife; 2020 Dec; 9():. PubMed ID: 33258451 [TBL] [Abstract][Full Text] [Related]
19. Small-Molecule Integrated Stress Response Inhibitor Reduces Susceptibility to Postinfarct Atrial Fibrillation in Rats via the Inhibition of Integrated Stress Responses. Zhang T; Wu Y; Hu Z; Xing W; Kun LV; Wang D; Hu N J Pharmacol Exp Ther; 2021 Sep; 378(3):197-206. PubMed ID: 34215702 [TBL] [Abstract][Full Text] [Related]
20. Novel mechanisms of eIF2B action and regulation by eIF2α phosphorylation. Bogorad AM; Lin KY; Marintchev A Nucleic Acids Res; 2017 Nov; 45(20):11962-11979. PubMed ID: 29036434 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]