234 related articles for article (PubMed ID: 25872983)
1. Design and synthesis of novel 1,2-dithiolan-4-yl benzoate derivatives as PTP1B inhibitors.
Chen J; Gao LX; Gong JX; Jiang CS; Yao LG; Li JY; Li J; Xiao W; Guo YW
Bioorg Med Chem Lett; 2015; 25(10):2211-6. PubMed ID: 25872983
[TBL] [Abstract][Full Text] [Related]
2. Design, synthesis and molecular modelling studies of novel 3-acetamido-4-methyl benzoic acid derivatives as inhibitors of protein tyrosine phosphatase 1B.
Rakse M; Karthikeyan C; Deora GS; Moorthy NS; Rathore V; Rawat AK; Srivastava AK; Trivedi P
Eur J Med Chem; 2013; 70():469-76. PubMed ID: 24185377
[TBL] [Abstract][Full Text] [Related]
3. [Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].
Du X; Zhang SE; Liu JZ; Nie FL; Ye F; Tian JY; Xiao ZY
Yao Xue Xue Bao; 2012 Mar; 47(3):367-73. PubMed ID: 22645761
[TBL] [Abstract][Full Text] [Related]
4. Design, synthesis, and biological evaluation of bromophenol derivatives as protein tyrosine phosphatase 1B inhibitors.
Jiang B; Shi D; Cui Y; Guo S
Arch Pharm (Weinheim); 2012 Jun; 345(6):444-53. PubMed ID: 22307562
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors.
Wang WL; Huang C; Gao LX; Tang CL; Wang JQ; Wu MC; Sheng L; Chen HJ; Nan FJ; Li JY; Li J; Feng B
Bioorg Med Chem Lett; 2014 Apr; 24(8):1889-94. PubMed ID: 24684845
[TBL] [Abstract][Full Text] [Related]
6. Design, synthesis and insulin-sensitising effects of novel PTP1B inhibitors.
Tang YB; Lu D; Chen Z; Hu C; Yang Y; Tian JY; Ye F; Wu L; Zhang ZY; Xiao Z
Bioorg Med Chem Lett; 2013 Apr; 23(8):2313-8. PubMed ID: 23499238
[TBL] [Abstract][Full Text] [Related]
7. Design, synthesis, and biological evaluation of 2-substituted ethenesulfonic acid ester derivatives as selective PTP1B inhibitors.
Liu J; Deng X; Jin Y; Xu B; Liu W; Jiang F; Fu L
Pharmazie; 2015 Jul; 70(7):446-51. PubMed ID: 26373204
[TBL] [Abstract][Full Text] [Related]
8. The first synthesis of natural disulfide bruguiesulfurol and biological evaluation of its derivatives as a novel scaffold for PTP1B inhibitors.
Chen J; Jiang CS; Ma WQ; Gao LX; Gong JX; Li JY; Li J; Guo YW
Bioorg Med Chem Lett; 2013 Sep; 23(18):5061-5. PubMed ID: 23942421
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and biological evaluation of (±)-3-(2-(2-fluorobenzyloxy) naphthalen-6-yl)-2-aminopropanoic acid derivatives as novel PTP1B inhibitors.
Sun LP; Shen Q; Piao HH; Ma WP; Gao LX; Zhang W; Nan FJ; Li J; Piao HR
Eur J Med Chem; 2011 Sep; 46(9):3630-8. PubMed ID: 21680062
[TBL] [Abstract][Full Text] [Related]
10. Design, synthesis and docking study of 5-(substituted benzylidene)thiazolidine-2,4-dione derivatives as inhibitors of protein tyrosine phosphatase 1B.
Wang Z; Liu Z; Lee W; Kim SN; Yoon G; Cheon SH
Bioorg Med Chem Lett; 2014 Aug; 24(15):3337-40. PubMed ID: 24953600
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and biological evaluation of heterocyclic ring-substituted maslinic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.
Qiu WW; Shen Q; Yang F; Wang B; Zou H; Li JY; Li J; Tang J
Bioorg Med Chem Lett; 2009 Dec; 19(23):6618-22. PubMed ID: 19846303
[TBL] [Abstract][Full Text] [Related]
12. Design, synthesis and in vitro activity of phidianidine B derivatives as novel PTP1B inhibitors with specific selectivity.
Zhang L; Jiang CS; Gao LX; Gong JX; Wang ZH; Li JY; Li J; Li XW; Guo YW
Bioorg Med Chem Lett; 2016 Feb; 26(3):778-781. PubMed ID: 26774579
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and biological evaluation of novel thiadiazole amides as potent Cdc25B and PTP1B inhibitors.
Li Y; Yu Y; Jin K; Gao L; Luo T; Sheng L; Shao X; Li J
Bioorg Med Chem Lett; 2014 Sep; 24(17):4125-8. PubMed ID: 25124112
[TBL] [Abstract][Full Text] [Related]
14. Identification of 2-substituted ethenesulfonic acid ester derivatives as novel, potent and selective inhibitors of protein tyrosine phosphatase 1B.
Deng X; Liu J; Jin Y; Zhang Y; He W; Bao J; Liu W; Jiang F; Fu L
Pharmazie; 2015 Dec; 70(12):777-83. PubMed ID: 26817274
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis, and biological evaluation of novel 2-ethyl-5-phenylthiazole-4-carboxamide derivatives as protein tyrosine phosphatase 1B inhibitors with improved cellular efficacy.
Chen YT; Tang CL; Ma WP; Gao LX; Wei Y; Zhang W; Li JY; Li J; Nan FJ
Eur J Med Chem; 2013 Nov; 69():399-412. PubMed ID: 24090912
[TBL] [Abstract][Full Text] [Related]
16. The discovery of a novel and selective inhibitor of PTP1B over TCPTP: 3D QSAR pharmacophore modeling, virtual screening, synthesis, and biological evaluation.
Ma Y; Jin YY; Wang YL; Wang RL; Lu XH; Kong DX; Xu WR
Chem Biol Drug Des; 2014 Jun; 83(6):697-709. PubMed ID: 24418013
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and characterization of 5,7-dihydroxyflavanone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
Sun LP; Ma WP; Gao LX; Yang LL; Quan YC; Li J; Piao HR
J Enzyme Inhib Med Chem; 2013 Dec; 28(6):1199-204. PubMed ID: 23009604
[TBL] [Abstract][Full Text] [Related]
18. Design, synthesis, and evaluation of bromo-retrochalcone derivatives as protein tyrosine phosphatase 1B inhibitors.
Liu Z; Lee W; Kim SN; Yoon G; Cheon SH
Bioorg Med Chem Lett; 2011 Jun; 21(12):3755-8. PubMed ID: 21555221
[TBL] [Abstract][Full Text] [Related]
19. Design, Synthesis and Biological Evaluation of Stilbene Derivatives as Novel Inhibitors of Protein Tyrosine Phosphatase 1B.
He H; Ge Y; Dai H; Cui S; Ye F; Jin J; Shi Y
Molecules; 2016 Dec; 21(12):. PubMed ID: 27999292
[TBL] [Abstract][Full Text] [Related]
20. Isothiazolidinone inhibitors of PTP1B containing imidazoles and imidazolines.
Douty B; Wayland B; Ala PJ; Bower MJ; Pruitt J; Bostrom L; Wei M; Klabe R; Gonneville L; Wynn R; Burn TC; Liu PC; Combs AP; Yue EW
Bioorg Med Chem Lett; 2008 Jan; 18(1):66-71. PubMed ID: 18037290
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]