BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

150 related articles for article (PubMed ID: 25937210)

  • 1. Direct visualisation of internalization of the adenosine A3 receptor and localization with arrestin3 using a fluorescent agonist.
    Stoddart LA; Vernall AJ; Briddon SJ; Kellam B; Hill SJ
    Neuropharmacology; 2015 Nov; 98():68-77. PubMed ID: 25937210
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Agonist-occupied A3 adenosine receptors exist within heterogeneous complexes in membrane microdomains of individual living cells.
    Cordeaux Y; Briddon SJ; Alexander SP; Kellam B; Hill SJ
    FASEB J; 2008 Mar; 22(3):850-60. PubMed ID: 17959910
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Efficient G protein coupling is not required for agonist-mediated internalization and membrane reorganization of the adenosine A
    Stoddart LA; Kilpatrick LE; Corriden R; Kellam B; Briddon SJ; Hill SJ
    FASEB J; 2021 Apr; 35(4):e21211. PubMed ID: 33710641
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Effect of a toggle switch mutation in TM6 of the human adenosine A₃ receptor on Gi protein-dependent signalling and Gi-independent receptor internalization.
    Stoddart LA; Kellam B; Briddon SJ; Hill SJ
    Br J Pharmacol; 2014 Aug; 171(16):3827-44. PubMed ID: 24750014
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Subtype-specific regulation of receptor internalization and recycling by the carboxyl-terminal domains of the human A1 and rat A3 adenosine receptors: consequences for agonist-stimulated translocation of arrestin3.
    Ferguson G; Watterson KR; Palmer TM
    Biochemistry; 2002 Dec; 41(50):14748-61. PubMed ID: 12475223
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Allosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics.
    May LT; Bridge LJ; Stoddart LA; Briddon SJ; Hill SJ
    FASEB J; 2011 Oct; 25(10):3465-76. PubMed ID: 21715680
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and evaluation of adenosine derivatives as A
    Bednarska-Szczepaniak K; Mieczkowski A; Kierozalska A; Pavlović Saftić D; Głąbała K; Przygodzki T; Stańczyk L; Karolczak K; Watała C; Rao H; Gao ZG; Jacobson KA; Leśnikowski ZJ
    Eur J Med Chem; 2021 Nov; 223():113607. PubMed ID: 34171656
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Flexible modulation of agonist efficacy at the human A3 adenosine receptor by the imidazoquinoline allosteric enhancer LUF6000.
    Gao ZG; Ye K; Göblyös A; Ijzerman AP; Jacobson KA
    BMC Pharmacol; 2008 Dec; 8():20. PubMed ID: 19077268
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Arrestin specificity for G protein-coupled receptors in human airway smooth muscle.
    Penn RB; Pascual RM; Kim YM; Mundell SJ; Krymskaya VP; Panettieri RA; Benovic JL
    J Biol Chem; 2001 Aug; 276(35):32648-56. PubMed ID: 11418617
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Different efficacy of adenosine and NECA derivatives at the human A3 adenosine receptor: insight into the receptor activation switch.
    Dal Ben D; Buccioni M; Lambertucci C; Kachler S; Falgner N; Marucci G; Thomas A; Cristalli G; Volpini R; Klotz KN
    Biochem Pharmacol; 2014 Jan; 87(2):321-31. PubMed ID: 24161786
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Effects of synthetic A3 adenosine receptor agonists on cell proliferation and viability are receptor independent at micromolar concentrations.
    Mlejnek P; Dolezel P; Frydrych I
    J Physiol Biochem; 2013 Sep; 69(3):405-17. PubMed ID: 23184730
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Functionally biased modulation of A(3) adenosine receptor agonist efficacy and potency by imidazoquinolinamine allosteric enhancers.
    Gao ZG; Verzijl D; Zweemer A; Ye K; Göblyös A; Ijzerman AP; Jacobson KA
    Biochem Pharmacol; 2011 Sep; 82(6):658-68. PubMed ID: 21718691
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Adenosine A(2A) receptor dynamics studied with the novel fluorescent agonist Alexa488-APEC.
    Brand F; Klutz AM; Jacobson KA; Fredholm BB; Schulte G
    Eur J Pharmacol; 2008 Aug; 590(1-3):36-42. PubMed ID: 18603240
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Influence of fluorophore and linker composition on the pharmacology of fluorescent adenosine A1 receptor ligands.
    Baker JG; Middleton R; Adams L; May LT; Briddon SJ; Kellam B; Hill SJ
    Br J Pharmacol; 2010 Feb; 159(4):772-86. PubMed ID: 20105183
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Antagonist selective modulation of adenosine A1 and A3 receptor pharmacology by the food dye Brilliant Black BN: evidence for allosteric interactions.
    May LT; Briddon SJ; Hill SJ
    Mol Pharmacol; 2010 Apr; 77(4):678-86. PubMed ID: 20086038
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.
    Klotz KN; Hessling J; Hegler J; Owman C; Kull B; Fredholm BB; Lohse MJ
    Naunyn Schmiedebergs Arch Pharmacol; 1998 Jan; 357(1):1-9. PubMed ID: 9459566
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Structure-Activity Analysis of Biased Agonism at the Human Adenosine A3 Receptor.
    Baltos JA; Paoletta S; Nguyen AT; Gregory KJ; Tosh DK; Christopoulos A; Jacobson KA; May LT
    Mol Pharmacol; 2016 Jul; 90(1):12-22. PubMed ID: 27136943
    [TBL] [Abstract][Full Text] [Related]  

  • 18. 7-Nitrobenzofurazan (NBD) derivatives of 5'-N-ethylcarboxamidoadenosine (NECA) as new fluorescent probes for human A(3) adenosine receptors.
    Macchia M; Salvetti F; Bertini S; Di Bussolo V; Gattuso L; Gesi M; Hamdan M; Klotz KN; Laragione T; Lucacchini A; Minutolo F; Nencetti S; Papi C; Tuscano D; Martini C
    Bioorg Med Chem Lett; 2001 Dec; 11(23):3023-6. PubMed ID: 11714602
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Regulation of p42/p44 mitogen-activated protein kinase by the human adenosine A3 receptor in transfected CHO cells.
    Graham S; Combes P; Crumiere M; Klotz KN; Dickenson JM
    Eur J Pharmacol; 2001 May; 420(1):19-26. PubMed ID: 11412835
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Cloning of a chick A3 adenosine receptor: characterization of ligand binding and receptor-effector coupling of chick A1 and A3 adenosine receptors.
    Durand IH; Green RD
    Naunyn Schmiedebergs Arch Pharmacol; 2001 Jan; 363(1):81-6. PubMed ID: 11191840
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.