BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

211 related articles for article (PubMed ID: 26038181)

  • 1. N-Cinnamoylation of Antimalarial Classics: Effects of Using Acyl Groups Other than Cinnamoyl toward Dual-Stage Antimalarials.
    Gomes A; Machado M; Lobo L; Nogueira F; Prudêncio M; Teixeira C; Gomes P
    ChemMedChem; 2015 Aug; 10(8):1344-9. PubMed ID: 26038181
    [TBL] [Abstract][Full Text] [Related]  

  • 2. N-cinnamoylation of antimalarial classics: quinacrine analogues with decreased toxicity and dual-stage activity.
    Gomes A; Pérez B; Albuquerque I; Machado M; Prudêncio M; Nogueira F; Teixeira C; Gomes P
    ChemMedChem; 2014 Feb; 9(2):305-10. PubMed ID: 24474655
    [TBL] [Abstract][Full Text] [Related]  

  • 3. In vitro efficiency of 9-(N-cinnamoylbutyl)aminoacridines against blood- and liver-stage malaria parasites.
    Pérez B; Teixeira C; Gomes AS; Albuquerque IS; Gut J; Rosenthal PJ; Prudêncio M; Gomes P
    Bioorg Med Chem Lett; 2013 Feb; 23(3):610-3. PubMed ID: 23290049
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and antimalarial activity in vitro and in vivo of a new ferrocene-chloroquine analogue.
    Biot C; Glorian G; Maciejewski LA; Brocard JS
    J Med Chem; 1997 Nov; 40(23):3715-8. PubMed ID: 9371235
    [TBL] [Abstract][Full Text] [Related]  

  • 5. 3,5-bis(benzylidene)-4-piperidones and related N-acyl analogs: a novel cluster of antimalarials targeting the liver stage of Plasmodium falciparum.
    Das U; Singh RS; Alcorn J; Hickman MR; Sciotti RJ; Leed SE; Lee PJ; Roncal N; Dimmock JR
    Bioorg Med Chem; 2013 Dec; 21(23):7250-6. PubMed ID: 24139941
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Novel antimalarial chloroquine- and primaquine-quinoxaline 1,4-di-N-oxide hybrids: Design, synthesis, Plasmodium life cycle stage profile, and preliminary toxicity studies.
    Bonilla-Ramirez L; Rios A; Quiliano M; Ramirez-Calderon G; Beltrán-Hortelano I; Franetich JF; Corcuera L; Bordessoulles M; Vettorazzi A; López de Cerain A; Aldana I; Mazier D; Pabón A; Galiano S
    Eur J Med Chem; 2018 Oct; 158():68-81. PubMed ID: 30199706
    [TBL] [Abstract][Full Text] [Related]  

  • 7. N-cinnamoylated chloroquine analogues as dual-stage antimalarial leads.
    Pérez BC; Teixeira C; Albuquerque IS; Gut J; Rosenthal PJ; Gomes JR; Prudêncio M; Gomes P
    J Med Chem; 2013 Jan; 56(2):556-67. PubMed ID: 23273038
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Novel 4-aminoquinoline analogs highly active against the blood and sexual stages of Plasmodium in vivo and in vitro.
    Sáenz FE; Mutka T; Udenze K; Oduola AM; Kyle DE
    Antimicrob Agents Chemother; 2012 Sep; 56(9):4685-92. PubMed ID: 22710117
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Enantiopure Indolizinoindolones with in vitro Activity against Blood- and Liver-Stage Malaria Parasites.
    Pereira NA; Monteiro Â; Machado M; Gut J; Molins E; Perry MJ; Dourado J; Moreira R; Rosenthal PJ; Prudêncio M; Santos MM
    ChemMedChem; 2015 Dec; 10(12):2080-9. PubMed ID: 26525306
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Cinnamoylated chloroquine analogues: A new structural class of antimalarial agents.
    Gayam V; Ravi S
    Eur J Med Chem; 2017 Jul; 135():382-391. PubMed ID: 28460312
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Structure-activity relationship of new antimalarial 1-aryl-3-susbtituted propanol derivatives: Synthesis, preliminary toxicity profiling, parasite life cycle stage studies, target exploration, and targeted delivery.
    Quiliano M; Pabón A; Moles E; Bonilla-Ramirez L; Fabing I; Fong KY; Nieto-Aco DA; Wright DW; Pizarro JC; Vettorazzi A; López de Cerain A; Deharo E; Fernández-Busquets X; Garavito G; Aldana I; Galiano S
    Eur J Med Chem; 2018 May; 152():489-514. PubMed ID: 29754074
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Recycling antimalarial leads for cancer: Antiproliferative properties of N-cinnamoyl chloroquine analogues.
    Pérez BC; Fernandes I; Mateus N; Teixeira C; Gomes P
    Bioorg Med Chem Lett; 2013 Dec; 23(24):6769-72. PubMed ID: 24184076
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Antimalarial dual drugs based on potent inhibitors of glutathione reductase from Plasmodium falciparum.
    Friebolin W; Jannack B; Wenzel N; Furrer J; Oeser T; Sanchez CP; Lanzer M; Yardley V; Becker K; Davioud-Charvet E
    J Med Chem; 2008 Mar; 51(5):1260-77. PubMed ID: 18260613
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and antimalarial activity of new heterocyclic hybrids based on chloroquine and thiazolidinone scaffolds.
    Rojas Ruiz FA; García-Sánchez RN; Estupiñan SV; Gómez-Barrio A; Torres Amado DF; Pérez-Solórzano BM; Nogal-Ruiz JJ; Martínez-Fernández AR; Kouznetsov VV
    Bioorg Med Chem; 2011 Aug; 19(15):4562-73. PubMed ID: 21723734
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Probing the Azaaurone Scaffold against the Hepatic and Erythrocytic Stages of Malaria Parasites.
    Carrasco MP; Machado M; Gonçalves L; Sharma M; Gut J; Lukens AK; Wirth DF; André V; Duarte MT; Guedes RC; Dos Santos DJ; Rosenthal PJ; Mazitschek R; Prudêncio M; Moreira R
    ChemMedChem; 2016 Oct; 11(19):2194-2204. PubMed ID: 27538856
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Cinnamic acid/chloroquinoline conjugates as potent agents against chloroquine-resistant Plasmodium falciparum.
    Pérez B; Teixeira C; Gut J; Rosenthal PJ; Gomes JR; Gomes P
    ChemMedChem; 2012 Sep; 7(9):1537-40. PubMed ID: 22753234
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparum.
    Sashidhara KV; Avula SR; Palnati GR; Singh SV; Srivastava K; Puri SK; Saxena JK
    Bioorg Med Chem Lett; 2012 Sep; 22(17):5455-9. PubMed ID: 22850213
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Antimalarial activity of 4-(5-trifluoromethyl-1H-pyrazol-1-yl)-chloroquine analogues.
    Cunico W; Cechinel CA; Bonacorso HG; Martins MA; Zanatta N; de Souza MV; Freitas IO; Soares RP; Krettli AU
    Bioorg Med Chem Lett; 2006 Feb; 16(3):649-53. PubMed ID: 16257205
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Toward a novel metal-based chemotherapy against tropical diseases. 3. Synthesis and antimalarial activity in vitro and in vivo of the new gold-chloroquine complex [Au(PPh3)(CQ)]PF6.
    Navarro M; Pérez H; Sánchez-Delgado RA
    J Med Chem; 1997 Jun; 40(12):1937-9. PubMed ID: 9191972
    [No Abstract]   [Full Text] [Related]  

  • 20. A new class of phenazines with activity against a chloroquine resistant Plasmodium falciparum strain and antimicrobial activity.
    Hussain H; Specht S; Sarite SR; Saeftel M; Hoerauf A; Schulz B; Krohn K
    J Med Chem; 2011 Jul; 54(13):4913-7. PubMed ID: 21591758
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.