BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

238 related articles for article (PubMed ID: 26083464)

  • 1. Highly Selective, Reversible Inhibitor Identified by Comparative Chemoproteomics Modulates Diacylglycerol Lipase Activity in Neurons.
    Baggelaar MP; Chameau PJ; Kantae V; Hummel J; Hsu KL; Janssen F; van der Wel T; Soethoudt M; Deng H; den Dulk H; Allarà M; Florea BI; Di Marzo V; Wadman WJ; Kruse CG; Overkleeft HS; Hankemeier T; Werkman TR; Cravatt BF; van der Stelt M
    J Am Chem Soc; 2015 Jul; 137(27):8851-7. PubMed ID: 26083464
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Diacylglycerol Lipase-Alpha Regulates Hippocampal-Dependent Learning and Memory Processes in Mice.
    Schurman LD; Carper MC; Moncayo LV; Ogasawara D; Richardson K; Yu L; Liu X; Poklis JL; Liu QS; Cravatt BF; Lichtman AH
    J Neurosci; 2019 Jul; 39(30):5949-5965. PubMed ID: 31127001
    [TBL] [Abstract][Full Text] [Related]  

  • 3. A novel fluorophosphonate inhibitor of the biosynthesis of the endocannabinoid 2-arachidonoylglycerol with potential anti-obesity effects.
    Bisogno T; Mahadevan A; Coccurello R; Chang JW; Allarà M; Chen Y; Giacovazzo G; Lichtman A; Cravatt B; Moles A; Di Marzo V
    Br J Pharmacol; 2013 Jun; 169(4):784-93. PubMed ID: 23072382
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Diacylglycerol lipase is not involved in depolarization-induced suppression of inhibition at unitary inhibitory connections in mouse hippocampus.
    Min R; Testa-Silva G; Heistek TS; Canto CB; Lodder JC; Bisogno T; Di Marzo V; Brussaard AB; Burnashev N; Mansvelder HD
    J Neurosci; 2010 Feb; 30(7):2710-5. PubMed ID: 20164355
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Competitive ABPP of Serine Hydrolases: A Case Study on DAGL-Alpha.
    Baggelaar MP; Van der Stelt M
    Methods Mol Biol; 2017; 1491():161-169. PubMed ID: 27778288
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition.
    Ogasawara D; Deng H; Viader A; Baggelaar MP; Breman A; den Dulk H; van den Nieuwendijk AM; Soethoudt M; van der Wel T; Zhou J; Overkleeft HS; Sanchez-Alavez M; Mori S; Nguyen W; Conti B; Liu X; Chen Y; Liu QS; Cravatt BF; van der Stelt M
    Proc Natl Acad Sci U S A; 2016 Jan; 113(1):26-33. PubMed ID: 26668358
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Development and optimization of piperidyl-1,2,3-triazole ureas as selective chemical probes of endocannabinoid biosynthesis.
    Hsu KL; Tsuboi K; Whitby LR; Speers AE; Pugh H; Inloes J; Cravatt BF
    J Med Chem; 2013 Nov; 56(21):8257-69. PubMed ID: 24152245
    [TBL] [Abstract][Full Text] [Related]  

  • 8. A natural substrate-based fluorescence assay for inhibitor screening on diacylglycerol lipase α.
    van der Wel T; Janssen FJ; Baggelaar MP; Deng H; den Dulk H; Overkleeft HS; van der Stelt M
    J Lipid Res; 2015 Apr; 56(4):927-35. PubMed ID: 25684760
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Identification of small molecules that selectively inhibit diacylglycerol lipase-α activity.
    Appiah KK; Blat Y; Robertson BJ; Pearce BC; Pedicord DL; Gentles RG; Yu XC; Mseeh F; Nguyen N; Swaffield JC; Harden DG; Westphal RS; Banks MN; O'Connell JC
    J Biomol Screen; 2014 Apr; 19(4):595-605. PubMed ID: 24241710
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Postsynaptic diacylglycerol lipase mediates retrograde endocannabinoid suppression of inhibition in mouse prefrontal cortex.
    Yoshino H; Miyamae T; Hansen G; Zambrowicz B; Flynn M; Pedicord D; Blat Y; Westphal RS; Zaczek R; Lewis DA; Gonzalez-Burgos G
    J Physiol; 2011 Oct; 589(Pt 20):4857-84. PubMed ID: 21807615
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Brain regional cannabinoid CB(1) receptor signalling and alternative enzymatic pathways for 2-arachidonoylglycerol generation in brain sections of diacylglycerol lipase deficient mice.
    Aaltonen N; Riera Ribas C; Lehtonen M; Savinainen JR; Laitinen JT
    Eur J Pharm Sci; 2014 Jan; 51():87-95. PubMed ID: 24012970
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Inhibition of diacylglycerol lipase β modulates lipid and endocannabinoid levels in the
    Berger N; van der Wel T; Hirschmugl B; Baernthaler T; Gindlhuber J; Fawzy N; Eichmann T; Birner-Gruenberger R; Zimmermann R; van der Stelt M; Wadsack C
    Front Endocrinol (Lausanne); 2023; 14():1092024. PubMed ID: 36864832
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Multiple Forms of Endocannabinoid and Endovanilloid Signaling Regulate the Tonic Control of GABA Release.
    Lee SH; Ledri M; Tóth B; Marchionni I; Henstridge CM; Dudok B; Kenesei K; Barna L; Szabó SI; Renkecz T; Oberoi M; Watanabe M; Limoli CL; Horvai G; Soltesz I; Katona I
    J Neurosci; 2015 Jul; 35(27):10039-57. PubMed ID: 26157003
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Discovery of glycine sulfonamides as dual inhibitors of sn-1-diacylglycerol lipase α and α/β-hydrolase domain 6.
    Janssen FJ; Deng H; Baggelaar MP; Allarà M; van der Wel T; den Dulk H; Ligresti A; van Esbroeck AC; McGuire R; Di Marzo V; Overkleeft HS; van der Stelt M
    J Med Chem; 2014 Aug; 57(15):6610-22. PubMed ID: 24988361
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Cannabinoid receptor subtype influence on neuritogenesis in human SH-SY5Y cells.
    Lyons EL; Leone-Kabler S; Kovach AL; Thomas BF; Howlett AC
    Mol Cell Neurosci; 2020 Dec; 109():103566. PubMed ID: 33049367
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Simplified assays of lipolysis enzymes for drug discovery and specificity assessment of known inhibitors.
    Iglesias J; Lamontagne J; Erb H; Gezzar S; Zhao S; Joly E; Truong VL; Skorey K; Crane S; Madiraju SR; Prentki M
    J Lipid Res; 2016 Jan; 57(1):131-41. PubMed ID: 26423520
    [TBL] [Abstract][Full Text] [Related]  

  • 17. DAG lipase involvement in depolarization-induced suppression of inhibition: does endocannabinoid biosynthesis always meet the demand?
    Min R; Di Marzo V; Mansvelder HD
    Neuroscientist; 2010 Dec; 16(6):608-13. PubMed ID: 20837870
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Chemical tools to modulate 2-arachidonoylglycerol biosynthesis.
    Deng H; van der Stelt M
    Biotechnol Appl Biochem; 2018 Jan; 65(1):9-15. PubMed ID: 28589628
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Investigation of Diacylglycerol Lipase Alpha Inhibition in the Mouse Lipopolysaccharide Inflammatory Pain Model.
    Wilkerson JL; Donvito G; Grim TW; Abdullah RA; Ogasawara D; Cravatt BF; Lichtman AH
    J Pharmacol Exp Ther; 2017 Dec; 363(3):394-401. PubMed ID: 28970359
    [TBL] [Abstract][Full Text] [Related]  

  • 20.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

    [Next]    [New Search]
    of 12.