BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

273 related articles for article (PubMed ID: 26114811)

  • 1. Synthesis, antiplasmodial activity and mechanistic studies of pyrimidine-5-carbonitrile and quinoline hybrids.
    Kaur H; Balzarini J; de Kock C; Smith PJ; Chibale K; Singh K
    Eur J Med Chem; 2015 Aug; 101():52-62. PubMed ID: 26114811
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Quinoline-pyrimidine hybrids: synthesis, antiplasmodial activity, SAR, and mode of action studies.
    Singh K; Kaur H; Smith P; de Kock C; Chibale K; Balzarini J
    J Med Chem; 2014 Jan; 57(2):435-48. PubMed ID: 24354322
    [TBL] [Abstract][Full Text] [Related]  

  • 3. N-Piperonyl substitution on aminoquinoline-pyrimidine hybrids: Effect on the antiplasmodial potency.
    Kholiya R; Khan SI; Bahuguna A; Tripathi M; Rawat DS
    Eur J Med Chem; 2017 May; 131():126-140. PubMed ID: 28315598
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and in vitro antiplasmodial activity of ferrocenyl aminoquinoline derivatives.
    Mwande Maguene G; Lekana-Douki JB; Mouray E; Bousquet T; Grellier P; Pellegrini S; Toure Ndouo FS; Lebibi J; Pélinski L
    Eur J Med Chem; 2015 Jan; 90():519-25. PubMed ID: 25486423
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Design and synthesis of quinoline-pyrimidine inspired hybrids as potential plasmodial inhibitors.
    Kayamba F; Malimabe T; Ademola IK; Pooe OJ; Kushwaha ND; Mahlalela M; van Zyl RL; Gordon M; Mudau PT; Zininga T; Shonhai A; Nyamori VO; Karpoormath R
    Eur J Med Chem; 2021 May; 217():113330. PubMed ID: 33744688
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis, characterization and antimalarial activity of quinoline-pyrimidine hybrids.
    Pretorius SI; Breytenbach WJ; de Kock C; Smith PJ; N'Da DD
    Bioorg Med Chem; 2013 Jan; 21(1):269-77. PubMed ID: 23168082
    [TBL] [Abstract][Full Text] [Related]  

  • 7. 4-Aminoquinoline-pyrimidine hybrids: synthesis, antimalarial activity, heme binding and docking studies.
    Kumar D; Khan SI; Tekwani BL; Ponnan P; Rawat DS
    Eur J Med Chem; 2015 Jan; 89():490-502. PubMed ID: 25462261
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis of 4-aminoquinoline-pyrimidine hybrids as potent antimalarials and their mode of action studies.
    Singh K; Kaur H; Chibale K; Balzarini J
    Eur J Med Chem; 2013 Aug; 66():314-23. PubMed ID: 23811093
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and evaluation of the antiplasmodial activity of novel indeno[2,1-c]quinoline derivatives.
    Barteselli A; Parapini S; Basilico N; Mommo D; Sparatore A
    Bioorg Med Chem; 2014 Nov; 22(21):5757-65. PubMed ID: 25311562
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Ferrocene-pyrimidine conjugates: Synthesis, electrochemistry, physicochemical properties and antiplasmodial activities.
    Chopra R; de Kock C; Smith P; Chibale K; Singh K
    Eur J Med Chem; 2015 Jul; 100():1-9. PubMed ID: 26057222
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Primaquine-pyrimidine hybrids: synthesis and dual-stage antiplasmodial activity.
    Kaur H; Machado M; de Kock C; Smith P; Chibale K; Prudêncio M; Singh K
    Eur J Med Chem; 2015 Aug; 101():266-73. PubMed ID: 26142491
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and evaluation of new diaryl ether and quinoline hybrids as potential antiplasmodial and antimicrobial agents.
    Mishra A; Batchu H; Srivastava K; Singh P; Shukla PK; Batra S
    Bioorg Med Chem Lett; 2014 Apr; 24(7):1719-23. PubMed ID: 24630564
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and antimalarial testing of neocryptolepine analogues: addition of ester function in SAR study of 2,11-disubstituted indolo[2,3-b]quinolines.
    Lu WJ; Wicht KJ; Wang L; Imai K; Mei ZW; Kaiser M; El Sayed Iel T; Egan TJ; Inokuchi T
    Eur J Med Chem; 2013 Jun; 64():498-511. PubMed ID: 23685569
    [TBL] [Abstract][Full Text] [Related]  

  • 14. New pentasubstituted pyrrole hybrid atorvastatin-quinoline derivatives with antiplasmodial activity.
    Carvalho RC; Martins WA; Silva TP; Kaiser CR; Bastos MM; Pinheiro LC; Krettli AU; Boechat N
    Bioorg Med Chem Lett; 2016 Apr; 26(8):1881-4. PubMed ID: 26988303
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Bioisosteric ferrocenyl aminoquinoline-benzimidazole hybrids: Antimicrobial evaluation and mechanistic insights.
    Baartzes N; Stringer T; Seldon R; Warner DF; Taylor D; Wittlin S; Chibale K; Smith GS
    Eur J Med Chem; 2019 Oct; 180():121-133. PubMed ID: 31301563
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Novel Quinolinyl-pyrrolo[3,4-d]pyrimidine-2,5-dione Derivatives Against Chloroquine-resistant Plasmodium falciparum.
    Rogerio KR; Graebin CS; Pinto Domingues LH; Oliveira LS; de Souza Fernandes da Silva V; Daniel-Ribeiro CT; Carvalho LJM; Boechat N
    Curr Top Med Chem; 2020; 20(2):99-110. PubMed ID: 31648638
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Quinoline hybrids and their antiplasmodial and antimalarial activities.
    Hu YQ; Gao C; Zhang S; Xu L; Xu Z; Feng LS; Wu X; Zhao F
    Eur J Med Chem; 2017 Oct; 139():22-47. PubMed ID: 28800458
    [TBL] [Abstract][Full Text] [Related]  

  • 18. New derivatives of quinoline-4-carboxylic acid with antiplasmodial activity.
    Hochegger P; Faist J; Seebacher W; Saf R; Mäser P; Kaiser M; Weis R
    Bioorg Med Chem; 2017 Apr; 25(7):2251-2259. PubMed ID: 28279559
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Evaluation of Antiplasmodial Potential of C2 and C8 Modified Quinolines: in vitro and in silico Study.
    Kumar R; Sharma R; Kumar I; Upadhyay P; Dhiman AK; Kumar R; Kumar R; Purohit R; Sahal D; Sharma U
    Med Chem; 2019; 15(7):790-800. PubMed ID: 30324888
    [TBL] [Abstract][Full Text] [Related]  

  • 20. 4-Aminoquinoline-chalcone/-N-acetylpyrazoline conjugates: Synthesis and antiplasmodial evaluation.
    Kumar S; Saini A; Gut J; Rosenthal PJ; Raj R; Kumar V
    Eur J Med Chem; 2017 Sep; 138():993-1001. PubMed ID: 28756265
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 14.