138 related articles for article (PubMed ID: 26210158)
1. Novel fluorine-18 labeled 5-(1-pyrrolidinylsulfonyl)-7-azaisatin derivatives as potential PET tracers for in vivo imaging of activated caspases in apoptosis.
Waldmann CM; Hermann S; Faust A; Riemann B; Schober O; Schäfers M; Haufe G; Kopka K
Bioorg Med Chem; 2015 Sep; 23(17):5734-9. PubMed ID: 26210158
[TBL] [Abstract][Full Text] [Related]
2. The nonpeptidyl caspase binding radioligand (S)-1-(4-(2-[18F]Fluoroethoxy)-benzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin ([18F]CbR) as potential positron emission tomography-compatible apoptosis imaging agent.
Faust A; Wagner S; Law MP; Hermann S; Schnöckel U; Keul P; Schober O; Schäfers M; Levkau B; Kopka K
Q J Nucl Med Mol Imaging; 2007 Mar; 51(1):67-73. PubMed ID: 17372575
[TBL] [Abstract][Full Text] [Related]
3. Fluorinated isatin derivatives. Part 2. New N-substituted 5-pyrrolidinylsulfonyl isatins as potential tools for molecular imaging of caspases in apoptosis.
Podichetty AK; Wagner S; Schröer S; Faust A; Schäfers M; Schober O; Kopka K; Haufe G
J Med Chem; 2009 Jun; 52(11):3484-95. PubMed ID: 19445513
[TBL] [Abstract][Full Text] [Related]
4. 5-pyrrolidinylsulfonyl isatins as a potential tool for the molecular imaging of caspases in apoptosis.
Kopka K; Faust A; Keul P; Wagner S; Breyholz HJ; Höltke C; Schober O; Schäfers M; Levkau B
J Med Chem; 2006 Nov; 49(23):6704-15. PubMed ID: 17154501
[TBL] [Abstract][Full Text] [Related]
5. Synthesis, radiolabeling, and in vivo evaluation of an 18F-labeled isatin analog for imaging caspase-3 activation in apoptosis.
Zhou D; Chu W; Rothfuss J; Zeng C; Xu J; Jones L; Welch MJ; Mach RH
Bioorg Med Chem Lett; 2006 Oct; 16(19):5041-6. PubMed ID: 16891117
[TBL] [Abstract][Full Text] [Related]
6. Synthesis of new fluorinated, 2-substituted 5-pyrrolidinylsulfonyl isatin derivatives as caspase-3 and caspase-7 inhibitors: nonradioactive counterparts of putative PET-compatible apoptosis imaging agents.
Limpachayaporn P; Schäfers M; Schober O; Kopka K; Haufe G
Bioorg Med Chem; 2013 Apr; 21(7):2025-36. PubMed ID: 23411396
[TBL] [Abstract][Full Text] [Related]
7. Synthesis, 18F-radiolabeling, and in vivo biodistribution studies of N-fluorohydroxybutyl isatin sulfonamides using positron emission tomography.
Limpachayaporn P; Wagner S; Kopka K; Hermann S; Schäfers M; Haufe G
J Med Chem; 2013 Jun; 56(11):4509-20. PubMed ID: 23656488
[TBL] [Abstract][Full Text] [Related]
8. Fluorinated isatin derivatives. Part 3. New side-chain fluoro-functionalized pyrrolidinyl sulfonyl isatins as potent caspase-3 and -7 inhibitors.
Podichetty AK; Wagner S; Faust A; Schäfers M; Schober O; Kopka K; Haufe G
Future Med Chem; 2009 Aug; 1(5):969-89. PubMed ID: 21426092
[TBL] [Abstract][Full Text] [Related]
9. [18F]- and [11C]-labeled N-benzyl-isatin sulfonamide analogues as PET tracers for apoptosis: synthesis, radiolabeling mechanism, and in vivo imaging study of apoptosis in Fas-treated mice using [11C]WC-98.
Zhou D; Chu W; Chen DL; Wang Q; Reichert DE; Rothfuss J; D'Avignon A; Welch MJ; Mach RH
Org Biomol Chem; 2009 Apr; 7(7):1337-48. PubMed ID: 19300818
[TBL] [Abstract][Full Text] [Related]
10. Design, synthesis, and biological characterization of a caspase 3/7 selective isatin labeled with 2-[18F]fluoroethylazide.
Smith G; Glaser M; Perumal M; Nguyen QD; Shan B; Arstad E; Aboagye EO
J Med Chem; 2008 Dec; 51(24):8057-67. PubMed ID: 19049429
[TBL] [Abstract][Full Text] [Related]
11. One-pot multi-tracer synthesis of novel (18)F-labeled PET imaging agents.
Haslop A; Wells L; Gee A; Plisson C; Long N
Mol Pharm; 2014 Nov; 11(11):3818-22. PubMed ID: 25158244
[TBL] [Abstract][Full Text] [Related]
12. Fluorine-18 click radiosynthesis and preclinical evaluation of a new 18F-labeled folic acid derivative.
Ross TL; Honer M; Lam PY; Mindt TL; Groehn V; Schibli R; Schubiger PA; Ametamey SM
Bioconjug Chem; 2008 Dec; 19(12):2462-70. PubMed ID: 19053298
[TBL] [Abstract][Full Text] [Related]
13. Influence of 4- or 5-substituents on the pyrrolidine ring of 5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin derivatives on their inhibitory activities towards caspases-3 and -7.
Limpachayaporn P; Riemann B; Kopka K; Schober O; Schäfers M; Haufe G
Eur J Med Chem; 2013 Jun; 64():562-78. PubMed ID: 23685941
[TBL] [Abstract][Full Text] [Related]
14. An efficient bioorthogonal strategy using CuAAC click chemistry for radiofluorinations of SNEW peptides and the role of copper depletion.
Pretze M; Kuchar M; Bergmann R; Steinbach J; Pietzsch J; Mamat C
ChemMedChem; 2013 Jun; 8(6):935-45. PubMed ID: 23559494
[TBL] [Abstract][Full Text] [Related]
15. Isatin sulfonamides: potent caspases-3 and -7 inhibitors, and promising PET and SPECT radiotracers for apoptosis imaging.
Limpachayaporn P; Schäfers M; Haufe G
Future Med Chem; 2015; 7(9):1173-96. PubMed ID: 26132525
[TBL] [Abstract][Full Text] [Related]
16. A novel versatile precursor suitable for
Lugato B; Stucchi S; Ciceri S; Iannone MN; Turolla EA; Giuliano L; Chinello C; Todde S; Ferraboschi P
J Labelled Comp Radiopharm; 2017 Aug; 60(10):466-480. PubMed ID: 28600889
[TBL] [Abstract][Full Text] [Related]
17. A fluorous and click approach for screening potential PET probes: Evaluation of potential hypoxia biomarkers.
Bejot R; Carroll L; Bhakoo K; Declerck J; Gouverneur V
Bioorg Med Chem; 2012 Jan; 20(1):324-9. PubMed ID: 22130421
[TBL] [Abstract][Full Text] [Related]
18. Fluorine-18 labeling by click chemistry: multiple probes in one pot.
Jia L; Cheng Z; Shi L; Li J; Wang C; Jiang D; Zhou W; Meng H; Qi Y; Cheng D; Zhang L
Appl Radiat Isot; 2013 May; 75():64-70. PubMed ID: 23455406
[TBL] [Abstract][Full Text] [Related]
19. General method for labeling siRNA by click chemistry with fluorine-18 for the purpose of PET imaging.
Mercier F; Paris J; Kaisin G; Thonon D; Flagothier J; Teller N; Lemaire C; Luxen A
Bioconjug Chem; 2011 Jan; 22(1):108-14. PubMed ID: 21174402
[TBL] [Abstract][Full Text] [Related]
20. Development of indazolylpyrimidine derivatives as high-affine EphB4 receptor ligands and potential PET radiotracers.
Ebert K; Wiemer J; Caballero J; Köckerling M; Steinbach J; Pietzsch J; Mamat C
Bioorg Med Chem; 2015 Sep; 23(17):6025-35. PubMed ID: 26189032
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
