123 related articles for article (PubMed ID: 26216015)
1. Synthesis of CNS active thyrotropin-releasing hormone (TRH)-like peptides: Biological evaluation and effect on cognitive impairment induced by cerebral ischemia in mice.
Meena CL; Thakur A; Nandekar PP; Sangamwar AT; Sharma SS; Jain R
Bioorg Med Chem; 2015 Sep; 23(17):5641-53. PubMed ID: 26216015
[TBL] [Abstract][Full Text] [Related]
2. Modifications of the pyroglutamic acid and histidine residues in thyrotropin-releasing hormone (TRH) yield analogs with selectivity for TRH receptor type 2 over type 1.
Kaur N; Monga V; Lu X; Gershengorn MC; Jain R
Bioorg Med Chem; 2007 Jan; 15(1):433-43. PubMed ID: 17035026
[TBL] [Abstract][Full Text] [Related]
3. Synthesis, receptor binding, and CNS pharmacological studies of new thyrotropin-releasing hormone (TRH) analogues.
Monga V; Meena CL; Rajput S; Pawar C; Sharma SS; Lu X; Gershengorn MC; Jain R
ChemMedChem; 2011 Mar; 6(3):531-43. PubMed ID: 21302359
[TBL] [Abstract][Full Text] [Related]
4. Synthesis and biology of ring-modified l-Histidine containing thyrotropin-releasing hormone (TRH) analogues.
Meena CL; Thakur A; Nandekar PP; Sharma SS; Sangamwar AT; Jain R
Eur J Med Chem; 2016 Mar; 111():72-83. PubMed ID: 26854379
[TBL] [Abstract][Full Text] [Related]
5. Thyrotropin-releasing hormone (TRH) analogues that exhibit selectivity to TRH receptor subtype 2.
Kaur N; Lu X; Gershengorn MC; Jain R
J Med Chem; 2005 Sep; 48(19):6162-5. PubMed ID: 16162016
[TBL] [Abstract][Full Text] [Related]
6. Synthesis, receptor binding, and activation studies of N(1)-alkyl-L-histidine containing thyrotropin-releasing hormone (TRH) analogues.
Kaur N; Monga V; Josan JS; Lu X; Gershengorn MC; Jain R
Bioorg Med Chem; 2006 Sep; 14(17):5981-8. PubMed ID: 16735122
[TBL] [Abstract][Full Text] [Related]
7. Discovery of a low affinity thyrotropin-releasing hormone (TRH)-like peptide that exhibits potent inhibition of scopolamine-induced memory impairment in mice.
Meena CL; Ingole S; Rajpoot S; Thakur A; Nandeker PP; Sangamwar AT; Sharma SS; Jain R
RSC Adv; 2015 Jun; 5():56872-56884. PubMed ID: 26191403
[TBL] [Abstract][Full Text] [Related]
8. Selectivity-based QSAR approach for screening and evaluation of TRH analogs for TRH-R1 and TRH-R2 receptors subtypes.
Kadam RU; Chavan AG; Monga V; Kaur N; Jain R; Roy N
J Mol Graph Model; 2008 Oct; 27(3):309-20. PubMed ID: 18595758
[TBL] [Abstract][Full Text] [Related]
9. Thyrotropin-releasing hormone receptor type 1 (TRH-R1), not TRH-R2, primarily mediates taltirelin actions in the CNS of mice.
Thirunarayanan N; Nir EA; Raaka BM; Gershengorn MC
Neuropsychopharmacology; 2013 May; 38(6):950-6. PubMed ID: 23303050
[TBL] [Abstract][Full Text] [Related]
10. Discovery of a dual action first-in-class peptide that mimics and enhances CNS-mediated actions of thyrotropin-releasing hormone.
Scalabrino GA; Hogan N; O'Boyle KM; Slator GR; Gregg DJ; Fitchett CM; Draper SM; Bennett GW; Hinkle PM; Bauer K; Williams CH; Tipton KF; Kelly JA
Neuropharmacology; 2007 Jun; 52(7):1472-81. PubMed ID: 17418282
[TBL] [Abstract][Full Text] [Related]
11. First-in-class thyrotropin-releasing hormone (TRH)-based compound binds to a pharmacologically distinct TRH receptor subtype in human brain and is effective in neurodegenerative models.
Kelly JA; Boyle NT; Cole N; Slator GR; Colivicchi MA; Stefanini C; Gobbo OL; Scalabrino GA; Ryan SM; Elamin M; Walsh C; Vajda A; Goggin MM; Campbell M; Mash DC; O'Mara SM; Brayden DJ; Callanan JJ; Tipton KF; Della Corte L; Hunter J; O'Boyle KM; Williams CH; Hardiman O
Neuropharmacology; 2015 Feb; 89():193-203. PubMed ID: 25281210
[TBL] [Abstract][Full Text] [Related]
12. Antiepileptic potential and behavioral profile of L-pGlu-(2-propyl)-L-His-L-ProNH2, a newer thyrotropin-releasing hormone analog.
Rajput SK; Krishnamoorthy S; Pawar C; Kaur N; Monga V; Meena CL; Jain R; Sharma SS
Epilepsy Behav; 2009 Jan; 14(1):48-53. PubMed ID: 18952198
[TBL] [Abstract][Full Text] [Related]
13. Thyrotropin-releasing hormone receptors -- similarities and differences.
Sun Y; Lu X; Gershengorn MC
J Mol Endocrinol; 2003 Apr; 30(2):87-97. PubMed ID: 12683933
[TBL] [Abstract][Full Text] [Related]
14. Regulator of G protein signaling 4 suppresses basal and thyrotropin releasing-hormone (TRH)-stimulated signaling by two mouse TRH receptors, TRH-R(1) and TRH-R(2).
Harder S; Lu X; Wang W; Buck F; Gershengorn MC; Bruhn TO
Endocrinology; 2001 Mar; 142(3):1188-94. PubMed ID: 11181534
[TBL] [Abstract][Full Text] [Related]
15. Effect of L-pGlu-(1-benzyl)-l-His-l-Pro-NH
Rajput SK; Sharma AK; Meena CL; Pant AB; Jain R; Sharma SS
Biomed Pharmacother; 2016 Dec; 84():1256-1265. PubMed ID: 27810782
[TBL] [Abstract][Full Text] [Related]
16. Pyroglutamyl peptidase II inhibition enhances the analeptic effect of thyrotropin-releasing hormone in the rat medial septum.
Lazcano I; Uribe RM; Martínez-Chávez E; Vargas MA; Matziari M; Joseph-Bravo P; Charli JL
J Pharmacol Exp Ther; 2012 Jul; 342(1):222-31. PubMed ID: 22532627
[TBL] [Abstract][Full Text] [Related]
17. Expression of thyrotropin-releasing hormone receptor 2 (TRH-R2) in the central nervous system of rats.
Heuer H; Schäfer MK; O'Donnell D; Walker P; Bauer K
J Comp Neurol; 2000 Dec; 428(2):319-36. PubMed ID: 11064370
[TBL] [Abstract][Full Text] [Related]
18. Understanding the structural and functional differences between mouse thyrotropin-releasing hormone receptors 1 and 2.
Deflorian F; Engel S; Colson AO; Raaka BM; Gershengorn MC; Costanzi S
Proteins; 2008 May; 71(2):783-94. PubMed ID: 17979196
[TBL] [Abstract][Full Text] [Related]
19. Centrally acting and metabolically stable thyrotropin-releasing hormone analogues by replacement of histidine with substituted pyridinium.
Prokai L; Prokai-Tatrai K; Zharikova AD; Nguyen V; Perjesi P; Stevens SM
J Med Chem; 2004 Nov; 47(24):6025-33. PubMed ID: 15537357
[TBL] [Abstract][Full Text] [Related]
20. Role of the extracellular loops of the thyrotropin-releasing hormone receptor: evidence for an initial interaction with thyrotropin-releasing hormone.
Perlman JH; Colson AO; Jain R; Czyzewski B; Cohen LA; Osman R; Gershengorn MC
Biochemistry; 1997 Dec; 36(50):15670-6. PubMed ID: 9398295
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
