BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

207 related articles for article (PubMed ID: 26280898)

  • 1. Synthesis and Biological Evaluation of Fluorinated 3-Phenylcoumarin-7-O-Sulfamate Derivatives as Steroid Sulfatase Inhibitors.
    Demkowicz S; Daśko M; Kozak W; Krawczyk K; Witt D; Masłyk M; Kubiński K; Rachon J
    Chem Biol Drug Des; 2016 Feb; 87(2):233-8. PubMed ID: 26280898
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and biological evaluation of fluorinated N-benzoyl and N-phenylacetoyl derivatives of 3-(4-aminophenyl)-coumarin-7-O-sulfamate as steroid sulfatase inhibitors.
    Daśko M; Przybyłowska M; Rachon J; Masłyk M; Kubiński K; Misiak M; Składanowski A; Demkowicz S
    Eur J Med Chem; 2017 Mar; 128():79-87. PubMed ID: 28152429
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and biological evaluation of N-acylated tyramine sulfamates containing C-F bonds as steroid sulfatase inhibitors.
    Daśko M; Rachon J; Masłyk M; Kubiński K; Demkowicz S
    Chem Biol Drug Des; 2017 Jul; 90(1):156-161. PubMed ID: 28032462
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase.
    Woo LW; Howarth NM; Purohit A; Hejaz HA; Reed MJ; Potter BV
    J Med Chem; 1998 Mar; 41(7):1068-83. PubMed ID: 9544207
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Design and synthesis of 3-benzylaminocoumarin-7-O-sulfamate derivatives as steroid sulfatase inhibitors.
    Hng Y; Lin MH; Lin TS; Liu IC; Lin IC; Lu YL; Chang CN; Chiu PF; Tsai KC; Chen MJ; Liang PH
    Bioorg Chem; 2020 Mar; 96():103618. PubMed ID: 32059152
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and biological evaluation of thiophosphate tricyclic coumarin derivatives as steroid sulfatase inhibitors.
    Kozak W; Daśko M; Masłyk M; Gielniewski B; Rachon J; Demkowicz S
    J Asian Nat Prod Res; 2015; 17(11):1091-6. PubMed ID: 26269086
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Novel steroid sulfatase inhibitors based on N-thiophosphorylated 3-(4-aminophenyl)-coumarin-7-O-sulfamates.
    Daśko M; Demkowicz S; Biernacki K; Harrous A; Rachon J; Kozak W; Martyna A; Masłyk M; Kubiński K; Boguszewska-Czubara A
    Drug Dev Res; 2019 Sep; 80(6):857-866. PubMed ID: 31301181
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Estrogen O-sulfamates and their analogues: Clinical steroid sulfatase inhibitors with broad potential.
    Thomas MP; Potter BV
    J Steroid Biochem Mol Biol; 2015 Sep; 153():160-9. PubMed ID: 25843211
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis of bicoumarin thiophosphate derivatives as steroid sulfatase inhibitors.
    Demkowicz S; Kozak W; Daśko M; Masłyk M; Gielniewski B; Rachon J
    Eur J Med Chem; 2015 Aug; 101():358-66. PubMed ID: 26163883
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Potent inhibition of steroid sulfatase activity by 3-O-sulfamate 17alpha-benzyl(or 4'-tert-butylbenzyl)estra-1,3,5(10)-trienes: combination of two substituents at positions C3 and c17alpha of estradiol.
    Ciobanu LC; Boivin RP; Luu-The V; Labrie F; Poirier D
    J Med Chem; 1999 Jun; 42(12):2280-6. PubMed ID: 10377235
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and evaluation of analogues of estrone-3-O-sulfamate as potent steroid sulfatase inhibitors.
    Lawrence Woo LW; Leblond B; Purohit A; Potter BV
    Bioorg Med Chem; 2012 Apr; 20(8):2506-19. PubMed ID: 22455789
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.
    Okada M; Nakagawa T; Iwashita S; Takegawa S; Fujii T; Koizumi N
    J Steroid Biochem Mol Biol; 2003 Nov; 87(2-3):141-8. PubMed ID: 14672734
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and structure-activity relationship studies of derivatives of the dual aromatase-sulfatase inhibitor 4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]methyl}phenyl sulfamate.
    Woo LW; Wood PM; Bubert C; Thomas MP; Purohit A; Potter BV
    ChemMedChem; 2013 May; 8(5):779-99. PubMed ID: 23495205
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design, synthesis, and biological evaluation of new arylamide derivatives possessing sulfonate or sulfamate moieties as steroid sulfatase enzyme inhibitors.
    El-Gamal MI; Semreen MH; Foster PA; Potter BV
    Bioorg Med Chem; 2016 Jun; 24(12):2762-7. PubMed ID: 27143133
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors.
    Moi D; Foster PA; Rimmer LG; Jaffri A; Deplano A; Balboni G; Onnis V; Potter BVL
    Eur J Med Chem; 2019 Nov; 182():111614. PubMed ID: 31422224
    [TBL] [Abstract][Full Text] [Related]  

  • 16. The design, synthesis, and biochemical evaluation of derivatives of biphenyl sulfamate-based compounds as novel inhibitors of estrone sulfatase.
    Ahmed S; James K; Owen CP
    Biochem Biophys Res Commun; 2002 May; 294(1):180-3. PubMed ID: 12054760
    [TBL] [Abstract][Full Text] [Related]  

  • 17. 2-phenylindole sulfamates: inhibitors of steroid sulfatase with antiproliferative activity in MCF-7 breast cancer cells.
    Walter G; Liebl R; von Angerer E
    J Steroid Biochem Mol Biol; 2004 Apr; 88(4-5):409-20. PubMed ID: 15145451
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Solid-phase parallel synthesis of 17alpha-substituted estradiol sulfamate and phenol libraries using the multidetachable sulfamate linker.
    Ciobanu LC; Poirier D
    J Comb Chem; 2003; 5(4):429-40. PubMed ID: 12857111
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Proton-in-flight mechanism for the spontaneous hydrolysis of N-methyl O-phenyl sulfamate: implications for the design of steroid sulfatase inhibitors.
    Edwards DR; Wolfenden R
    J Org Chem; 2012 May; 77(9):4450-3. PubMed ID: 22486328
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Steroid Sulfatase Inhibitors Based on Phosphate and Thiophosphate Flavone Analogs.
    Kozak W; Daśko M; Masłyk M; Kubiński K; Rachon J; Demkowicz S
    Drug Dev Res; 2015 Dec; 76(8):450-62. PubMed ID: 26415657
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.