BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

128 related articles for article (PubMed ID: 26288111)

  • 1. Structure-Activity Relationships and Anti-inflammatory Activities of N-Carbamothioylformamide Analogues as MIF Tautomerase Inhibitors.
    Zhang Y; Xu L; Zhang Z; Zhang Z; Zheng L; Li D; Li Y; Liu F; Yu K; Hou T; Zhen X
    J Chem Inf Model; 2015 Sep; 55(9):1994-2004. PubMed ID: 26288111
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Inhibition of macrophage migration inhibitory factor (MIF) tautomerase activity suppresses microglia-mediated inflammatory responses.
    Zhang Y; Gu R; Jia J; Hou T; Zheng LT; Zhen X
    Clin Exp Pharmacol Physiol; 2016 Nov; 43(11):1134-1144. PubMed ID: 27543936
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Macrophage migration inhibitory factor (MIF) inhibitor, Z-590 suppresses cartilage destruction in adjuvant-induced arthritis via inhibition of macrophage inflammatory activation.
    Zhang Z; Zhang R; Li L; Zhu L; Gao S; Lu Q; Gu Y; Zhang Y; Yang H; Hou T; Zhen X; Zheng LT
    Immunopharmacol Immunotoxicol; 2018 Apr; 40(2):149-157. PubMed ID: 29447014
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Macrophage migration inhibitory factor (MIF) tautomerase inhibitors as potential novel anti-inflammatory agents: current developments.
    Garai J; Lóránd T
    Curr Med Chem; 2009; 16(9):1091-114. PubMed ID: 19275614
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Macrophage migration inhibitory factor and the discovery of tautomerase inhibitors.
    Orita M; Yamamoto S; Katayama N; Fujita S
    Curr Pharm Des; 2002; 8(14):1297-317. PubMed ID: 12052220
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Critical modifications of the ISO-1 scaffold improve its potent inhibition of macrophage migration inhibitory factor (MIF) tautomerase activity.
    Cheng KF; Al-Abed Y
    Bioorg Med Chem Lett; 2006 Jul; 16(13):3376-9. PubMed ID: 16682188
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Coumarin and chromen-4-one analogues as tautomerase inhibitors of macrophage migration inhibitory factor: discovery and X-ray crystallography.
    Orita M; Yamamoto S; Katayama N; Aoki M; Takayama K; Yamagiwa Y; Seki N; Suzuki H; Kurihara H; Sakashita H; Takeuchi M; Fujita S; Yamada T; Tanaka A
    J Med Chem; 2001 Feb; 44(4):540-7. PubMed ID: 11170644
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening.
    McLean LR; Zhang Y; Li H; Li Z; Lukasczyk U; Choi YM; Han Z; Prisco J; Fordham J; Tsay JT; Reiling S; Vaz RJ; Li Y
    Bioorg Med Chem Lett; 2009 Dec; 19(23):6717-20. PubMed ID: 19836948
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Multiple binding modes of isothiocyanates that inhibit macrophage migration inhibitory factor.
    Spencer ES; Dale EJ; Gommans AL; Rutledge MT; Vo CT; Nakatani Y; Gamble AB; Smith RA; Wilbanks SM; Hampton MB; Tyndall JD
    Eur J Med Chem; 2015 Mar; 93():501-10. PubMed ID: 25743213
    [TBL] [Abstract][Full Text] [Related]  

  • 10. MIF tautomerase inhibitor potency of alpha,beta-unsaturated cyclic ketones.
    Garai J; Molnár V; Eros D; Orfi L; Lóránd T
    Int Immunopharmacol; 2007 Dec; 7(13):1741-6. PubMed ID: 17996684
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Inhibition of MIF bioactivity by rational design of pharmacological inhibitors of MIF tautomerase activity.
    Dios A; Mitchell RA; Aljabari B; Lubetsky J; O'Connor K; Liao H; Senter PD; Manogue KR; Lolis E; Metz C; Bucala R; Callaway DJ; Al-Abed Y
    J Med Chem; 2002 Jun; 45(12):2410-6. PubMed ID: 12036350
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Novel arylazoarylmethane as potential inhibitor of macrophage migration inhibitory factor.
    He M; Metz C; Cheng KF; Ling J; Coleman T; VanPatten S; Al-Abed Y
    Arch Pharm (Weinheim); 2014 Feb; 347(2):104-7. PubMed ID: 24243226
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Ellagic Acid, a Dietary Polyphenol, Inhibits Tautomerase Activity of Human Macrophage Migration Inhibitory Factor and Its Pro-inflammatory Responses in Human Peripheral Blood Mononuclear Cells.
    Sarkar S; Siddiqui AA; Mazumder S; De R; Saha SJ; Banerjee C; Iqbal MS; Adhikari S; Alam A; Roy S; Bandyopadhyay U
    J Agric Food Chem; 2015 May; 63(20):4988-98. PubMed ID: 25929447
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and bio-evaluation of human macrophage migration inhibitory factor inhibitor to develop anti-inflammatory agent.
    Alam A; Pal C; Goyal M; Kundu MK; Kumar R; Iqbal MS; Dey S; Bindu S; Sarkar S; Pal U; Maiti NC; Adhikari S; Bandyopadhyay U
    Bioorg Med Chem; 2011 Dec; 19(24):7365-73. PubMed ID: 22088307
    [TBL] [Abstract][Full Text] [Related]  

  • 15. A fluorinated analog of ISO-1 blocks the recognition and biological function of MIF and is orally efficacious in a murine model of colitis.
    Dagia NM; Kamath DV; Bhatt P; Gupte RD; Dadarkar SS; Fonseca L; Agarwal G; Chetrapal-Kunwar A; Balachandran S; Srinivasan S; Bose J; Pari K; B-Rao C; Parkale SS; Gadekar PK; Rodge AH; Mandrekar N; Vishwakarma RA; Sharma S
    Eur J Pharmacol; 2009 Apr; 607(1-3):201-12. PubMed ID: 19239912
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Virtual Screening of Some Active Human Macrophage Migration Inhibitory Factor Antagonists.
    Tsai TL; Lin TH
    J Biomol Screen; 2014 Aug; 19(7):1116-23. PubMed ID: 24554444
    [TBL] [Abstract][Full Text] [Related]  

  • 17. The tautomerase active site of macrophage migration inhibitory factor is a potential target for discovery of novel anti-inflammatory agents.
    Lubetsky JB; Dios A; Han J; Aljabari B; Ruzsicska B; Mitchell R; Lolis E; Al-Abed Y
    J Biol Chem; 2002 Jul; 277(28):24976-82. PubMed ID: 11997397
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design, synthesis, and protein crystallography of biaryltriazoles as potent tautomerase inhibitors of macrophage migration inhibitory factor.
    Dziedzic P; Cisneros JA; Robertson MJ; Hare AA; Danford NE; Baxter RH; Jorgensen WL
    J Am Chem Soc; 2015 Mar; 137(8):2996-3003. PubMed ID: 25697265
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Novel inhibitors of macrophage migration inhibitory factor prevent cytokine-induced beta cell death.
    Vujicic M; Nikolic I; Krajnovic T; Cheng KF; VanPatten S; He M; Stosic-Grujicic S; Stojanovic I; Al-Abed Y; Saksida T
    Eur J Pharmacol; 2014 Oct; 740():683-9. PubMed ID: 24967533
    [TBL] [Abstract][Full Text] [Related]  

  • 20. An integrative in silico methodology for the identification of modulators of macrophage migration inhibitory factor (MIF) tautomerase activity.
    El Turk F; Fauvet B; Ouertatani-Sakouhi H; Lugari A; Betzi S; Roche P; Morelli X; Lashuel HA
    Bioorg Med Chem; 2010 Jul; 18(14):5425-40. PubMed ID: 20639113
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.