BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

193 related articles for article (PubMed ID: 26329281)

  • 1. Synthesis and characterization of a new fluorogenic substrate for monoacylglycerol lipase and application to inhibition studies.
    Lauria S; Casati S; Ciuffreda P
    Anal Bioanal Chem; 2015 Oct; 407(26):8163-7. PubMed ID: 26329281
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A fluorescence-based assay for monoacylglycerol lipase compatible with inhibitor screening.
    Wang Y; Chanda P; Jones PG; Kennedy JD
    Assay Drug Dev Technol; 2008 Jun; 6(3):387-93. PubMed ID: 18452392
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Set-Up and Validation of a High Throughput Screening Method for Human Monoacylglycerol Lipase (MAGL) Based on a New Red Fluorescent Probe.
    Miceli M; Casati S; Ottria R; Di Leo S; Eberini I; Palazzolo L; Parravicini C; Ciuffreda P
    Molecules; 2019 Jun; 24(12):. PubMed ID: 31208066
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Cross-validated stable-isotope dilution GC-MS and LC-MS/MS assays for monoacylglycerol lipase (MAGL) activity by measuring arachidonic acid released from the endocannabinoid 2-arachidonoyl glycerol.
    Kayacelebi AA; Schauerte C; Kling K; Herbers J; Beckmann B; Engeli S; Jordan J; Zoerner AA; Tsikas D
    J Chromatogr B Analyt Technol Biomed Life Sci; 2017 Mar; 1047():151-159. PubMed ID: 27511795
    [TBL] [Abstract][Full Text] [Related]  

  • 5. A Sensitive and Versatile Fluorescent Activity Assay for ABHD6.
    Savinainen JR; Navia-Paldanius D; Laitinen JT
    Methods Mol Biol; 2016; 1412():169-78. PubMed ID: 27245903
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Characterization of binding properties of monoglyceride lipase inhibitors by a versatile fluorescence-based technique.
    Savinainen JR; Yoshino M; Minkkilä A; Nevalainen T; Laitinen JT
    Anal Biochem; 2010 Apr; 399(1):132-4. PubMed ID: 20005861
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Development of an HPLC/UV assay for the evaluation of inhibitors of human recombinant monoacylglycerol lipase.
    Del Carlo S; Manera C; Chicca A; Arena C; Bertini S; Burgalassi S; Tampucci S; Gertsch J; Macchia M; Saccomanni G
    J Pharm Biomed Anal; 2015 Apr; 108():113-21. PubMed ID: 25743577
    [TBL] [Abstract][Full Text] [Related]  

  • 8. High-performance liquid chromatography assay with fluorescence detection for the evaluation of inhibitors against human recombinant monoacylglycerol lipase.
    Holtfrerich A; Makharadze T; Lehr M
    Anal Biochem; 2010 Apr; 399(2):218-24. PubMed ID: 20015447
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Comparative biochemical characterization of the monoacylglycerol lipase inhibitor KML29 in brain, spinal cord, liver, spleen, fat and muscle tissue.
    Pasquarelli N; Porazik C; Hanselmann J; Weydt P; Ferger B; Witting A
    Neuropharmacology; 2015 Apr; 91():148-56. PubMed ID: 25497453
    [TBL] [Abstract][Full Text] [Related]  

  • 10. A Sensitive and Versatile Fluorescent Activity Assay for ABHD12.
    Savinainen JR; Navia-Paldanius D; Laitinen JT
    Methods Mol Biol; 2016; 1412():179-89. PubMed ID: 27245904
    [TBL] [Abstract][Full Text] [Related]  

  • 11. A New Ultrasensitive Bioluminescence-Based Method for Assaying Monoacylglycerol Lipase.
    Miceli M; Casati S; Allevi P; Berra S; Ottria R; Rota P; Branchini BR; Ciuffreda P
    Int J Mol Sci; 2021 Jun; 22(11):. PubMed ID: 34200322
    [TBL] [Abstract][Full Text] [Related]  

  • 12. The design, synthesis and biological evaluation of novel URB602 analogues as potential monoacylglycerol lipase inhibitors.
    Szabo M; Agostino M; Malone DT; Yuriev E; Capuano B
    Bioorg Med Chem Lett; 2011 Nov; 21(22):6782-7. PubMed ID: 21982493
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Identification and characterization of a new reversible MAGL inhibitor.
    Tuccinardi T; Granchi C; Rizzolio F; Caligiuri I; Battistello V; Toffoli G; Minutolo F; Macchia M; Martinelli A
    Bioorg Med Chem; 2014 Jul; 22(13):3285-91. PubMed ID: 24853323
    [TBL] [Abstract][Full Text] [Related]  

  • 14. The discovery of diazetidinyl diamides as potent and reversible inhibitors of monoacylglycerol lipase (MAGL).
    Zhu B; Connolly PJ; Zhang SP; Chevalier KM; Milligan CM; Flores CM; Macielag MJ
    Bioorg Med Chem Lett; 2020 Jun; 30(12):127198. PubMed ID: 32334914
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Discovery of long-chain salicylketoxime derivatives as monoacylglycerol lipase (MAGL) inhibitors.
    Bononi G; Granchi C; Lapillo M; Giannotti M; Nieri D; Fortunato S; Boustani ME; Caligiuri I; Poli G; Carlson KE; Kim SH; Macchia M; Martinelli A; Rizzolio F; Chicca A; Katzenellenbogen JA; Minutolo F; Tuccinardi T
    Eur J Med Chem; 2018 Sep; 157():817-836. PubMed ID: 30144699
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors.
    Aghazadeh Tabrizi M; Baraldi PG; Baraldi S; Ruggiero E; De Stefano L; Rizzolio F; Di Cesare Mannelli L; Ghelardini C; Chicca A; Lapillo M; Gertsch J; Manera C; Macchia M; Martinelli A; Granchi C; Minutolo F; Tuccinardi T
    J Med Chem; 2018 Feb; 61(3):1340-1354. PubMed ID: 29309142
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Robust hydrolysis of prostaglandin glycerol esters by human monoacylglycerol lipase (MAGL).
    Savinainen JR; Kansanen E; Pantsar T; Navia-Paldanius D; Parkkari T; Lehtonen M; Laitinen T; Nevalainen T; Poso A; Levonen AL; Laitinen JT
    Mol Pharmacol; 2014 Nov; 86(5):522-35. PubMed ID: 25140003
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Loratadine analogues as MAGL inhibitors.
    Patel JZ; Ahenkorah S; Vaara M; Staszewski M; Adams Y; Laitinen T; Navia-Paldanius D; Parkkari T; Savinainen JR; Walczyński K; Laitinen JT; Nevalainen TJ
    Bioorg Med Chem Lett; 2015 Apr; 25(7):1436-42. PubMed ID: 25752982
    [TBL] [Abstract][Full Text] [Related]  

  • 19. (4-Phenoxyphenyl)tetrazolecarboxamides and related compounds as dual inhibitors of fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL).
    Holtfrerich A; Hanekamp W; Lehr M
    Eur J Med Chem; 2013 May; 63():64-75. PubMed ID: 23455058
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Docking based virtual screening and molecular dynamics study to identify potential monoacylglycerol lipase inhibitors.
    Afzal O; Kumar S; Kumar R; Firoz A; Jaggi M; Bawa S
    Bioorg Med Chem Lett; 2014 Aug; 24(16):3986-96. PubMed ID: 25011912
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.