170 related articles for article (PubMed ID: 26329912)
1. Nitrobenzoxadiazole-based GSTP1-1 inhibitors containing the full peptidyl moiety of (pseudo)glutathione.
Luisi G; Mollica A; Carradori S; Lenoci A; De Luca A; Caccuri AM
J Enzyme Inhib Med Chem; 2016 Dec; 31(6):924-30. PubMed ID: 26329912
[TBL] [Abstract][Full Text] [Related]
2. Potent isozyme-selective inhibition of human glutathione S-transferase A1-1 by a novel glutathione S-conjugate.
Cacciatore I; Caccuri AM; Cocco A; De Maria F; Di Stefano A; Luisi G; Pinnen F; Ricci G; Sozio P; Turella P
Amino Acids; 2005 Nov; 29(3):255-61. PubMed ID: 16082503
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis.
Di Paolo V; Fulci C; Rotili D; Sciarretta F; Lucidi A; Morozzo Della Rocca B; De Luca A; Rosato A; Quintieri L; Caccuri AM
J Enzyme Inhib Med Chem; 2019 Dec; 34(1):1131-1139. PubMed ID: 31169043
[TBL] [Abstract][Full Text] [Related]
4. Structural basis for the binding of the anticancer compound 6-(7-nitro-2,1,3-benzoxadiazol-4-ylthio)hexanol to human glutathione s-transferases.
Federici L; Lo Sterzo C; Pezzola S; Di Matteo A; Scaloni F; Federici G; Caccuri AM
Cancer Res; 2009 Oct; 69(20):8025-34. PubMed ID: 19808963
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and structure--activity relationship of new cytotoxic agents targeting human glutathione-S-transferases.
Rotili D; De Luca A; Tarantino D; Pezzola S; Forgione M; Morozzo Della Rocca B; Falconi M; Mai A; Caccuri AM
Eur J Med Chem; 2015 Jan; 89():156-71. PubMed ID: 25462236
[TBL] [Abstract][Full Text] [Related]
6. Selective inhibitors of glutathione transferase P1 with trioxane structure as anticancer agents.
Bräutigam M; Teusch N; Schenk T; Sheikh M; Aricioglu RZ; Borowski SH; Neudörfl JM; Baumann U; Griesbeck AG; Pietsch M
ChemMedChem; 2015 Apr; 10(4):629-39. PubMed ID: 25694385
[TBL] [Abstract][Full Text] [Related]
7. Peptide-bond modified glutathione conjugate analogs modulate GSTpi function in GSH-conjugation, drug sensitivity and JNK signaling.
Burg D; Riepsaame J; Pont C; Mulder G; van de Water B
Biochem Pharmacol; 2006 Jan; 71(3):268-77. PubMed ID: 16337611
[TBL] [Abstract][Full Text] [Related]
8. A covalent G-site inhibitor for glutathione S-transferase Pi (GSTP
Shishido Y; Tomoike F; Kimura Y; Kuwata K; Yano T; Fukui K; Fujikawa H; Sekido Y; Murakami-Tonami Y; Kameda T; Shuto S; Abe H
Chem Commun (Camb); 2017 Oct; 53(81):11138-11141. PubMed ID: 28848941
[TBL] [Abstract][Full Text] [Related]
9. Characterization of water-soluble esters of nitrobenzoxadiazole-based GSTP1-1 inhibitors for cancer treatment.
Di Paolo V; Fulci C; Rotili D; De Luca A; Tomassi S; Serra M; Scimeca M; Geroni C; Quintieri L; Caccuri AM
Biochem Pharmacol; 2020 Aug; 178():114060. PubMed ID: 32473836
[TBL] [Abstract][Full Text] [Related]
10. Identifying and characterizing binding sites on the irreversible inhibition of human glutathione S-transferase P1-1 by S-thiocarbamoylation.
Quesada-Soriano I; Primavera A; Casas-Solvas JM; Téllez-Sanz R; Barón C; Vargas-Berenguel A; Lo Bello M; García-Fuentes L
Chembiochem; 2012 Jul; 13(11):1594-604. PubMed ID: 22740430
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and biological evaluation of 2-substituted-5-(4-nitrophenylsulfonamido)benzoxazoles as human GST P1-1 inhibitors, and description of the binding site features.
Ertan-Bolelli T; Musdal Y; Bolelli K; Yilmaz S; Aksoy Y; Yildiz I; Aki-Yalcin E; Yalcin I
ChemMedChem; 2014 May; 9(5):984-92. PubMed ID: 24677708
[TBL] [Abstract][Full Text] [Related]
12. In Vitro Inhibition of Human Placental Glutathione S-Transferase by 3-Arylcoumarin Derivatives.
Alparslan MM; Danış Ö
Arch Pharm (Weinheim); 2015 Sep; 348(9):635-42. PubMed ID: 26205366
[TBL] [Abstract][Full Text] [Related]
13. A new nitrobenzoxadiazole-based GSTP1-1 inhibitor with a previously unheard of mechanism of action and high stability.
Fulci C; Rotili D; De Luca A; Stella L; Morozzo Della Rocca B; Forgione M; Di Paolo V; Mai A; Falconi M; Quintieri L; Caccuri AM
J Enzyme Inhib Med Chem; 2017 Dec; 32(1):240-247. PubMed ID: 28097896
[TBL] [Abstract][Full Text] [Related]
14. A Covalent Inhibitor for Glutathione S-Transferase Pi (GSTP
Shishido Y; Tomoike F; Kuwata K; Fujikawa H; Sekido Y; Murakami-Tonami Y; Kameda T; Abe N; Kimura Y; Shuto S; Abe H
Chembiochem; 2019 Apr; 20(7):900-905. PubMed ID: 30548113
[TBL] [Abstract][Full Text] [Related]
15. Ferrocene labelings as inhibitors and dual electrochemical sensors of human glutathione S-transferase P1-1.
Martos-Maldonado MC; Quesada-Soriano I; García-Maroto F; Vargas-Berenguel A; García-Fuentes L
Bioorg Med Chem Lett; 2012 Dec; 22(23):7256-60. PubMed ID: 23072868
[TBL] [Abstract][Full Text] [Related]
16. 7-Nitro-2,1,3-benzoxadiazole derivatives, a new class of suicide inhibitors for glutathione S-transferases. Mechanism of action of potential anticancer drugs.
Ricci G; De Maria F; Antonini G; Turella P; Bullo A; Stella L; Filomeni G; Federici G; Caccuri AM
J Biol Chem; 2005 Jul; 280(28):26397-405. PubMed ID: 15888444
[TBL] [Abstract][Full Text] [Related]
17. The evaluation of novel natural products as inhibitors of human glutathione transferase P1-1.
Mukanganyama S; Bezabih M; Robert M; Ngadjui BT; Kapche GF; Ngandeu F; Abegaz B
J Enzyme Inhib Med Chem; 2011 Aug; 26(4):460-7. PubMed ID: 21028940
[TBL] [Abstract][Full Text] [Related]
18. Enzymatic and nonenzymatic synthesis of glutathione conjugates: application to the understanding of a parasite's defense system and alternative to the discovery of potent glutathione S-transferase inhibitors.
Lo WJ; Chiou YC; Hsu YT; Lam WS; Chang MY; Jao SC; Li WS
Bioconjug Chem; 2007; 18(1):109-20. PubMed ID: 17226963
[TBL] [Abstract][Full Text] [Related]
19. Mechanistic studies of inactivation of glutathione S-transferase Pi isozyme by a haloenol lactone derivative.
Zheng J; Liu G; Tozkoparan B; Wen D
Med Chem; 2005 Mar; 1(2):191-8. PubMed ID: 16787314
[TBL] [Abstract][Full Text] [Related]
20. FDA-approved drugs and other compounds tested as inhibitors of human glutathione transferase P1-1.
Musdal Y; Hegazy UM; Aksoy Y; Mannervik B
Chem Biol Interact; 2013 Sep; 205(1):53-62. PubMed ID: 23769903
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]