107 related articles for article (PubMed ID: 26394987)
1. Novel dehydroepiandrosterone benzimidazolyl derivatives as 5α-reductase isozymes inhibitors.
Arellano Y; Bratoeff E; Segura T; Mendoza ME; Sánchez-Márquez A; Medina Y; Heuze Y; Soriano J; Cabeza M
J Enzyme Inhib Med Chem; 2016 Dec; 31(6):908-14. PubMed ID: 26394987
[TBL] [Abstract][Full Text] [Related]
2. Activity of steroid 4 and derivatives 4a-4f as inhibitors of the enzyme 5α-reductase 1.
Arellano Y; Bratoeff E; Heuze Y; Bravo M; Soriano J; Cabeza M
Bioorg Med Chem; 2018 Aug; 26(14):4058-4064. PubMed ID: 30007568
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and biological evaluation of esters of 16-formyl-17-methoxy-dehydroepiandrosterone derivatives as inhibitors of 5α-reductase type 2.
Sánchez-Márquez A; Arellano Y; Bratoeff E; Heuze Y; Córdova K; Nieves G; Soriano J; Cabeza M
J Enzyme Inhib Med Chem; 2016 Dec; 31(6):1170-6. PubMed ID: 26526826
[TBL] [Abstract][Full Text] [Related]
4. In vivo and in vitro effect of androstene derivatives as 5α-reductase type 1 enzyme inhibitors.
Bratoeff E; Sánchez A; Arellano Y; Heuze Y; Soriano J; Cabeza M
J Enzyme Inhib Med Chem; 2013 Dec; 28(6):1247-54. PubMed ID: 23051174
[TBL] [Abstract][Full Text] [Related]
5. Effect of dehydroepiandrosterone derivatives on the activity of 5α-reductase isoenzymes and on cancer cell line PC-3.
Bratoeff E; Garrido M; Ramírez-Apan T; Heuze Y; Sánchez A; Soriano J; Cabeza M
Bioorg Med Chem; 2014 Nov; 22(21):6233-41. PubMed ID: 25261928
[TBL] [Abstract][Full Text] [Related]
6. New ester derivatives of dehydroepiandrosterone as 5α-reductase inhibitors.
Arellano Y; Bratoeff E; Garrido M; Soriano J; Heuze Y; Cabeza M
Steroids; 2011 Nov; 76(12):1241-6. PubMed ID: 21729714
[TBL] [Abstract][Full Text] [Related]
7. Novel C-6 substituted and unsubstituted pregnane derivatives as 5alpha-reductase inhibitors and their effect on hamster flank organs diameter size.
Cabeza M; Zambrano A; Heuze I; Carrizales E; Palacios A; Segura T; Valencia N; Bratoeff E
Steroids; 2009 Oct; 74(10-11):793-802. PubMed ID: 19406144
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and activity of novel 16-dehydropregnenolone acetate derivatives as inhibitors of type 1 5α-reductase and on cancer cell line SK-LU-1.
Silva-Ortiz AV; Bratoeff E; Ramírez-Apan T; Heuze Y; Sánchez A; Soriano J; Cabeza M
Bioorg Med Chem; 2015 Dec; 23(24):7535-42. PubMed ID: 26631442
[TBL] [Abstract][Full Text] [Related]
9. Design, synthesis and biological evaluation of novel androst-3,5-diene-3-carboxylic acid derivatives as inhibitors of 5α-reductase type 1 and 2.
Lao K; Sun J; Wang C; Lyu W; Zhou B; Zhao R; Xu Q; You Q; Xiang H
Steroids; 2017 Aug; 124():29-34. PubMed ID: 28549802
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and biological evaluation of 3-tetrazolo steroidal analogs: Novel class of 5α-reductase inhibitors.
Aggarwal S; Mahapatra MK; Kumar R; Bhardwaj TR; Hartmann RW; Haupenthal J; Kumar M
Bioorg Med Chem; 2016 Feb; 24(4):779-88. PubMed ID: 26780831
[TBL] [Abstract][Full Text] [Related]
11. New steroidal 17β-carboxy derivatives present anti-5α-reductase activity and anti-proliferative effects in a human androgen-responsive prostate cancer cell line.
Amaral C; Varela C; Correia-da-Silva G; Tavares da Silva E; Carvalho RA; Costa SC; Cunha SC; Fernandes JO; Teixeira N; Roleira FM
Biochimie; 2013 Nov; 95(11):2097-106. PubMed ID: 23933094
[TBL] [Abstract][Full Text] [Related]
12. Synthesis and biological evaluation of novel unsaturated carboxysteroids as human 5α-reductase inhibitors: a legitimate approach.
Aggarwal S; Thareja S; Bhardwaj TR; Haupenthal J; Hartmann RW; Kumar M
Eur J Med Chem; 2012 Aug; 54():728-39. PubMed ID: 22776417
[TBL] [Abstract][Full Text] [Related]
13. Biological activity of pyrazole and imidazole-dehydroepiandrosterone derivatives on the activity of 17β-hydroxysteroid dehydrogenase.
Cabeza M; Posada A; Sánchez-Márquez A; Heuze Y; Moreno I; Soriano J; Garrido M; Cortés F; Bratoeff E
J Enzyme Inhib Med Chem; 2016; 31(1):53-62. PubMed ID: 25690043
[TBL] [Abstract][Full Text] [Related]
14. Synthesis of new derivatives of 21-imidazolyl-16-dehydropregnenolone as inhibitors of 5α-reductase 2 and with cytotoxic activity in cancer cells.
Silva-Ortiz AV; Bratoeff E; Ramírez-Apan T; Heuze Y; Soriano J; Moreno I; Bravo M; Bautista L; Cabeza M
Bioorg Med Chem; 2017 Mar; 25(5):1600-1607. PubMed ID: 28174065
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and Identification of Pregnenolone Derivatives as Inhibitors of Isozymes of 5α-Reductase.
Chávez-Riveros A; Bratoeff E; Heuze Y; Soriano J; Moreno I; Sánchez-Márquez A; Cabeza M
Arch Pharm (Weinheim); 2015 Nov; 348(11):808-816. PubMed ID: 26377677
[TBL] [Abstract][Full Text] [Related]
16. Bisphenol A modifies the regulation exerted by testosterone on 5 α -reductase isozymes in ventral prostate of adult rats.
Sánchez P; Castro B; Torres JM; Olmo A; del Moral RG; Ortega E
Biomed Res Int; 2013; 2013():629235. PubMed ID: 23984391
[TBL] [Abstract][Full Text] [Related]
17. New 5alpha-reductase inhibitors: in vitro and in vivo effects.
Pérez-Ornelas V; Cabeza M; Bratoeff E; Heuze I; Sánchez M; Ramírez E; Naranjo-Rodríguez E
Steroids; 2005 Mar; 70(3):217-24. PubMed ID: 15763601
[TBL] [Abstract][Full Text] [Related]
18. Activity of 17beta-(N-alkyl/arylformamido) and 17beta-[(N-alkyl/aryl) alkyl/arylamido]-4-methyl-4-aza-5alpha-androstan-3-ones as 5alpha-reductase inhibitors in the hamster flank organ and ear.
Chen C; Li X; Singh SM; Labrie F
J Invest Dermatol; 1998 Aug; 111(2):273-8. PubMed ID: 9699729
[TBL] [Abstract][Full Text] [Related]
19. Design, synthesis, and biological evaluation of novel androst-17β-amide structurally related compounds as dual 5α-reductase inhibitors and androgen receptor antagonists.
Lao K; Xun G; Gou X; Xiang H
J Enzyme Inhib Med Chem; 2019 Dec; 34(1):1597-1606. PubMed ID: 31469015
[TBL] [Abstract][Full Text] [Related]
20. Effects of perinatal exposure to bisphenol A on the intraprostatic levels of aromatase and 5α-reductase isozymes in juvenile rats.
Castro B; Sánchez P; Torres JM; Ortega E
Food Chem Toxicol; 2018 May; 115():20-25. PubMed ID: 29501275
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
