BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

163 related articles for article (PubMed ID: 26771593)

  • 1. Identification of Selective ERRγ Inverse Agonists.
    Kim J; Im CY; Yoo EK; Ma MJ; Kim SB; Hong E; Chin J; Hwang H; Lee S; Kim ND; Jeon JH; Lee IK; Jeon YH; Choi HS; Kim SH; Cho SJ
    Molecules; 2016 Jan; 21(1):80. PubMed ID: 26771593
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and biological evaluation of novel 4-hydroxytamoxifen analogs as estrogen-related receptor gamma inverse agonists.
    Kim J; Chin J; Im CY; Yoo EK; Woo S; Hwang HJ; Cho JH; Seo KA; Song J; Hwang H; Kim KH; Kim ND; Yoon SK; Jeon JH; Yoon SY; Jeon YH; Choi HS; Lee IK; Kim SH; Cho SJ
    Eur J Med Chem; 2016 Sep; 120():338-52. PubMed ID: 27236015
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Insights of a Lead Optimization Study and Biological Evaluation of Novel 4-Hydroxytamoxifen Analogs as Estrogen-Related Receptor γ (ERRγ) Inverse Agonists.
    Kim J; Woo SY; Im CY; Yoo EK; Lee S; Kim HJ; Hwang HJ; Cho JH; Lee WS; Yoon H; Kim S; Kwon OB; Hwang H; Kim KH; Jeon JH; Singh TD; Kim SW; Hwang SY; Choi HS; Lee IK; Kim SH; Jeon YH; Chin J; Cho SJ
    J Med Chem; 2016 Nov; 59(22):10209-10227. PubMed ID: 27805390
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Identification of novel inverse agonists of estrogen-related receptors ERRγ and ERRβ.
    Yu DD; Huss JM; Li H; Forman BM
    Bioorg Med Chem; 2017 Mar; 25(5):1585-1599. PubMed ID: 28189393
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Design, synthesis, and evaluation of simple phenol amides as ERRγ agonists.
    Lin H; Doebelin C; Patouret R; Garcia-Ordonez RD; Chang MR; Dharmarajan V; Bayona CR; Cameron MD; Griffin PR; Kamenecka TM
    Bioorg Med Chem Lett; 2018 May; 28(8):1313-1319. PubMed ID: 29548571
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Inverse agonist of ERRγ reduces cannabinoid receptor type 1-mediated induction of fibrinogen synthesis in mice with a high-fat diet-intoxicated liver.
    Zhang Y; Kim DK; Jung YS; Kim YH; Lee YS; Kim J; Jeong WI; Lee IK; Cho SJ; Dooley S; Lee CH; Choi HS
    Arch Toxicol; 2018 Sep; 92(9):2885-2896. PubMed ID: 30019168
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Efficient discovery of selective small molecule agonists of estrogen-related receptor gamma using combinatorial approach.
    Kim Y; Koh M; Kim DK; Choi HS; Park SB
    J Comb Chem; 2009; 11(5):928-37. PubMed ID: 19746993
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Inverse Agonist of Estrogen-Related Receptor γ Enhances Sodium Iodide Symporter Function Through Mitogen-Activated Protein Kinase Signaling in Anaplastic Thyroid Cancer Cells.
    Singh TD; Jeong SY; Lee SW; Ha JH; Lee IK; Kim SH; Kim J; Cho SJ; Ahn BC; Lee J; Jeon YH
    J Nucl Med; 2015 Nov; 56(11):1690-6. PubMed ID: 26338896
    [TBL] [Abstract][Full Text] [Related]  

  • 9. A Novel Orally Active Inverse Agonist of Estrogen-related Receptor Gamma (ERRγ), DN200434, A Booster of NIS in Anaplastic Thyroid Cancer.
    Singh TD; Song J; Kim J; Chin J; Ji HD; Lee JE; Lee SB; Yoon H; Yu JH; Kim SK; Yoon GS; Hwang H; Lee HW; Oh JM; Lee SW; Lee J; Choi HS; Na SY; Choi WI; Park YJ; Song YS; Kim YA; Lee IK; Cho SJ; Jeon YH
    Clin Cancer Res; 2019 Aug; 25(16):5069-5081. PubMed ID: 31010838
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Transcriptional corepressor SMILE recruits SIRT1 to inhibit nuclear receptor estrogen receptor-related receptor gamma transactivation.
    Xie YB; Park JH; Kim DK; Hwang JH; Oh S; Park SB; Shong M; Lee IK; Choi HS
    J Biol Chem; 2009 Oct; 284(42):28762-74. PubMed ID: 19690166
    [TBL] [Abstract][Full Text] [Related]  

  • 11. The Orphan Nuclear Receptor ERRγ Regulates Hepatic CB1 Receptor-Mediated Fibroblast Growth Factor 21 Gene Expression.
    Jung YS; Lee JM; Kim DK; Lee YS; Kim KS; Kim YH; Kim J; Lee MS; Lee IK; Kim SH; Cho SJ; Jeong WI; Lee CH; Harris RA; Choi HS
    PLoS One; 2016; 11(7):e0159425. PubMed ID: 27455076
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Discovery of Potent, Selective, and Orally Bioavailable Estrogen-Related Receptor-γ Inverse Agonists To Restore the Sodium Iodide Symporter Function in Anaplastic Thyroid Cancer.
    Kim J; Song J; Ji HD; Yoo EK; Lee JE; Lee SB; Oh JM; Lee S; Hwang JS; Yoon H; Kim DS; Lee SJ; Jeong M; Lee S; Kim KH; Choi HS; Lee SW; Park KG; Lee IK; Kim SH; Hwang H; Jeon YH; Chin J; Cho SJ
    J Med Chem; 2019 Feb; 62(4):1837-1858. PubMed ID: 30657313
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Orphan Nuclear Receptor ERRγ Is a Novel Transcriptional Regulator of IL-6 Mediated Hepatic BMP6 Gene Expression in Mice.
    Radhakrishnan K; Kim YH; Jung YS; Kim J; Kim DK; Cho SJ; Lee IK; Dooley S; Lee CH; Choi HS
    Int J Mol Sci; 2020 Sep; 21(19):. PubMed ID: 32998264
    [TBL] [Abstract][Full Text] [Related]  

  • 14. An inverse agonist of estrogen-related receptor γ regulates 2-arachidonoylglycerol synthesis by modulating diacylglycerol lipase expression in alcohol-intoxicated mice.
    Jung YS; Kim YH; Radhakrishnan K; Kim J; Kim DK; Lee JH; Oh H; Lee IK; Kim W; Cho SJ; Choi CS; Dooley S; Egan JM; Lee CH; Choi HS
    Arch Toxicol; 2020 Feb; 94(2):427-438. PubMed ID: 31912162
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Estrogen-Related Receptor γ Plays a Key Role in Vascular Calcification Through the Upregulation of BMP2 Expression.
    Kim JH; Choi YK; Do JY; Choi YK; Ha CM; Lee SJ; Jeon JH; Lee WK; Choi HS; Park KG; Lee IK
    Arterioscler Thromb Vasc Biol; 2015 Nov; 35(11):2384-90. PubMed ID: 26404484
    [TBL] [Abstract][Full Text] [Related]  

  • 16. A characteristic back support structure in the bisphenol A-binding pocket in the human nuclear receptor ERRγ.
    Liu X; Matsushima A; Shimohigashi M; Shimohigashi Y
    PLoS One; 2014; 9(6):e101252. PubMed ID: 24978476
    [TBL] [Abstract][Full Text] [Related]  

  • 17. In vitro metabolism of an estrogen-related receptor γ modulator, GSK5182, by human liver microsomes and recombinant cytochrome P450s.
    Joo J; Wu Z; Lee B; Shon JC; Lee T; Lee IK; Sim T; Kim KH; Kim ND; Kim SH; Liu KH
    Biopharm Drug Dispos; 2015 Apr; 36(3):163-73. PubMed ID: 25451157
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Requirements for transcriptional regulation by the orphan nuclear receptor ERRgamma.
    Huppunen J; Wohlfahrt G; Aarnisalo P
    Mol Cell Endocrinol; 2004 Apr; 219(1-2):151-60. PubMed ID: 15149736
    [TBL] [Abstract][Full Text] [Related]  

  • 19. A systematic methodology for large scale compound screening: A case study on the discovery of novel S1PL inhibitors.
    Deniz U; Ozkirimli E; Ulgen KO
    J Mol Graph Model; 2016 Jan; 63():110-24. PubMed ID: 26724452
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Structure-based discovery of pyrazolamides as novel ERRγ inverse agonists.
    Yang SH; Khadka DB; Han J; Na SY; Shin M; Kim DK; Oh BC; Kim EY; Choi HS; Cho WJ
    Eur J Med Chem; 2023 Mar; 250():115174. PubMed ID: 36805944
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.