245 related articles for article (PubMed ID: 26940860)
1. A continuous sirtuin activity assay without any coupling to enzymatic or chemical reactions.
Schuster S; Roessler C; Meleshin M; Zimmermann P; Simic Z; Kambach C; Schiene-Fischer C; Steegborn C; Hottiger MO; Schutkowski M
Sci Rep; 2016 Mar; 6():22643. PubMed ID: 26940860
[TBL] [Abstract][Full Text] [Related]
2. A Novel Continuous Assay for the Deacylase Sirtuin 5 and Other Deacetylases.
Roessler C; Tüting C; Meleshin M; Steegborn C; Schutkowski M
J Med Chem; 2015 Sep; 58(18):7217-23. PubMed ID: 26308971
[TBL] [Abstract][Full Text] [Related]
3. Continuous Fluorescent Sirtuin Activity Assay Based on Fatty Acylated Lysines.
Zessin M; Meleshin M; Hilscher S; Schiene-Fischer C; Barinka C; Jung M; Schutkowski M
Int J Mol Sci; 2023 Apr; 24(8):. PubMed ID: 37108579
[TBL] [Abstract][Full Text] [Related]
4. An improved fluorogenic assay for SIRT1, SIRT2, and SIRT3.
Chiang YL; Lin H
Org Biomol Chem; 2016 Feb; 14(7):2186-90. PubMed ID: 26796034
[TBL] [Abstract][Full Text] [Related]
5. High-throughput assays for sirtuin enzymes: a microfluidic mobility shift assay and a bioluminescence assay.
Liu Y; Gerber R; Wu J; Tsuruda T; McCarter JD
Anal Biochem; 2008 Jul; 378(1):53-9. PubMed ID: 18358225
[TBL] [Abstract][Full Text] [Related]
6. New chemical tools for probing activity and inhibition of the NAD
Swyter S; Schiedel M; Monaldi D; Szunyogh S; Lehotzky A; Rumpf T; Ovádi J; Sippl W; Jung M
Philos Trans R Soc Lond B Biol Sci; 2018 Jun; 373(1748):. PubMed ID: 29685963
[TBL] [Abstract][Full Text] [Related]
7. Identification and characterization of novel sirtuin inhibitor scaffolds.
Sanders BD; Jackson B; Brent M; Taylor AM; Dang W; Berger SL; Schreiber SL; Howitz K; Marmorstein R
Bioorg Med Chem; 2009 Oct; 17(19):7031-41. PubMed ID: 19734050
[TBL] [Abstract][Full Text] [Related]
8. New assays and approaches for discovery and design of Sirtuin modulators.
Schutkowski M; Fischer F; Roessler C; Steegborn C
Expert Opin Drug Discov; 2014 Feb; 9(2):183-99. PubMed ID: 24382304
[TBL] [Abstract][Full Text] [Related]
9. The mimics of N
Wang C; Wang F; Chen X; Zou Y; Zhu H; Zhao Q; Shen J; Li Y; Li Y; He B
Bioorg Med Chem Lett; 2018 Aug; 28(14):2375-2378. PubMed ID: 29921476
[TBL] [Abstract][Full Text] [Related]
10. Kinetic and Structural Basis for Acyl-Group Selectivity and NAD(+) Dependence in Sirtuin-Catalyzed Deacylation.
Feldman JL; Dittenhafer-Reed KE; Kudo N; Thelen JN; Ito A; Yoshida M; Denu JM
Biochemistry; 2015 May; 54(19):3037-3050. PubMed ID: 25897714
[TBL] [Abstract][Full Text] [Related]
11. Continuous Sirtuin/HDAC (histone deacetylase) activity assay using thioamides as PET (Photoinduced Electron Transfer)-based fluorescence quencher.
Zessin M; Meleshin M; Simic Z; Kalbas D; Arbach M; Gebhardt P; Melesina J; Liebscher S; Bordusa F; Sippl W; Barinka C; Schutkowski M
Bioorg Chem; 2021 Dec; 117():105425. PubMed ID: 34695733
[TBL] [Abstract][Full Text] [Related]
12. Identification of sirtuin 5 inhibitors by ultrafast microchip electrophoresis using nanoliter volume samples.
Guetschow ED; Kumar S; Lombard DB; Kennedy RT
Anal Bioanal Chem; 2016 Jan; 408(3):721-31. PubMed ID: 26635020
[TBL] [Abstract][Full Text] [Related]
13. HPLC-Based Enzyme Assays for Sirtuins.
Hong JY; Zhang X; Lin H
Methods Mol Biol; 2018; 1813():225-234. PubMed ID: 30097871
[TBL] [Abstract][Full Text] [Related]
14. Sensitive fluorogenic substrates for sirtuin deacylase inhibitor discovery.
Yang LL; Wang HL; Yan YH; Liu S; Yu ZJ; Huang MY; Luo Y; Zheng X; Yu Y; Li GB
Eur J Med Chem; 2020 Apr; 192():112201. PubMed ID: 32163813
[TBL] [Abstract][Full Text] [Related]
15. A Continuous, Fluorogenic Sirtuin 2 Deacylase Assay: Substrate Screening and Inhibitor Evaluation.
Galleano I; Schiedel M; Jung M; Madsen AS; Olsen CA
J Med Chem; 2016 Feb; 59(3):1021-31. PubMed ID: 26788965
[TBL] [Abstract][Full Text] [Related]
16. Potent and Selective Inhibitors of Human Sirtuin 5.
Kalbas D; Liebscher S; Nowak T; Meleshin M; Pannek M; Popp C; Alhalabi Z; Bordusa F; Sippl W; Steegborn C; Schutkowski M
J Med Chem; 2018 Mar; 61(6):2460-2471. PubMed ID: 29494161
[TBL] [Abstract][Full Text] [Related]
17. A FRET-based assay for screening SIRT6 modulators.
Li Y; You L; Huang W; Liu J; Zhu H; He B
Eur J Med Chem; 2015; 96():245-9. PubMed ID: 25884115
[TBL] [Abstract][Full Text] [Related]
18. Structure-based development of novel sirtuin inhibitors.
Schlicker C; Boanca G; Lakshminarasimhan M; Steegborn C
Aging (Albany NY); 2011 Sep; 3(9):852-72. PubMed ID: 21937767
[TBL] [Abstract][Full Text] [Related]
19. Sirtuin functions and modulation: from chemistry to the clinic.
Carafa V; Rotili D; Forgione M; Cuomo F; Serretiello E; Hailu GS; Jarho E; Lahtela-Kakkonen M; Mai A; Altucci L
Clin Epigenetics; 2016; 8():61. PubMed ID: 27226812
[TBL] [Abstract][Full Text] [Related]
20. The Current State of NAD
Schiedel M; Robaa D; Rumpf T; Sippl W; Jung M
Med Res Rev; 2018 Jan; 38(1):147-200. PubMed ID: 28094444
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]