179 related articles for article (PubMed ID: 27041552)
1. Synthesis of 1,4-disubstituted 1,2,3-triazole Derivatives Using Click Chemistry and their Src Kinase Activities.
Lebeau A; Abrioux C; Bénimèlis D; Benfodda Z; Meffre P
Med Chem; 2016; 13(1):40-48. PubMed ID: 27041552
[TBL] [Abstract][Full Text] [Related]
2. Click chemistry inspired one-pot synthesis of 1,4-disubstituted 1,2,3-triazoles and their Src kinase inhibitory activity.
Kumar D; Reddy VB; Kumar A; Mandal D; Tiwari R; Parang K
Bioorg Med Chem Lett; 2011 Jan; 21(1):449-52. PubMed ID: 21084189
[TBL] [Abstract][Full Text] [Related]
3. ZINClick: a database of 16 million novel, patentable, and readily synthesizable 1,4-disubstituted triazoles.
Massarotti A; Brunco A; Sorba G; Tron GC
J Chem Inf Model; 2014 Feb; 54(2):396-406. PubMed ID: 24451008
[TBL] [Abstract][Full Text] [Related]
4. 'Click' synthesis of a triazole-based inhibitor of Met functions in cancer cells.
Colombo F; Tintori C; Furlan A; Borrelli S; Christodoulou MS; Dono R; Maina F; Botta M; Amat M; Bosch J; Passarella D
Bioorg Med Chem Lett; 2012 Jul; 22(14):4693-6. PubMed ID: 22738633
[TBL] [Abstract][Full Text] [Related]
5. Click chemistry based synthesis, cytotoxic activity and molecular docking of novel triazole-thienopyrimidine hybrid glycosides targeting EGFR.
Khattab RR; Alshamari AK; Hassan AA; Elganzory HH; El-Sayed WA; Awad HM; Nossier ES; Hassan NA
J Enzyme Inhib Med Chem; 2021 Dec; 36(1):504-516. PubMed ID: 33504239
[TBL] [Abstract][Full Text] [Related]
6. Click-chemistry mediated synthesis of OTBN-1,2,3-Triazole derivatives exhibiting STK33 inhibition with diverse anti-cancer activities.
Vala DP; Dunne Miller A; Atmasidha A; Parmar MP; Patel CD; Upadhyay DB; Bhalodiya SS; González-Bakker A; Khan AN; Nogales J; Padrón JM; Banerjee S; Patel HM
Bioorg Chem; 2024 Aug; 149():107485. PubMed ID: 38824700
[TBL] [Abstract][Full Text] [Related]
7. Synthesis, biological evaluation and docking studies of new pyrrolo[2,3-d] pyrimidine derivatives as Src family-selective tyrosine kinase inhibitors.
Dincer S; Cetin KT; Onay-Besikci A; Ölgen S
J Enzyme Inhib Med Chem; 2013 Oct; 28(5):1080-7. PubMed ID: 22957720
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and biological evaluation of 1-(6-methylpyridin-2-yl)-5-(quinoxalin-6-yl)-1,2,3-triazoles as transforming growth factor-β type 1 receptor kinase inhibitors.
Li F; Park Y; Hah JM; Ryu JS
Bioorg Med Chem Lett; 2013 Feb; 23(4):1083-6. PubMed ID: 23294702
[TBL] [Abstract][Full Text] [Related]
9. 4-Aryl-4H-chromene-3-carbonitrile derivatives: evaluation of Src kinase inhibitory and anticancer activities.
Fallah-Tafti A; Tiwari R; Shirazi AN; Akbarzadeh T; Mandal D; Shafiee A; Parang K; Foroumadi A
Med Chem; 2011 Sep; 7(5):466-72. PubMed ID: 21801146
[TBL] [Abstract][Full Text] [Related]
10. Discovery of novel purine derivatives with potent and selective inhibitory activity against c-Src tyrosine kinase.
Huang H; Ma J; Shi J; Meng L; Jiang H; Ding J; Liu H
Bioorg Med Chem; 2010 Jul; 18(13):4615-24. PubMed ID: 20570525
[TBL] [Abstract][Full Text] [Related]
11. N-[2-Methyl-5-(triazol-1-yl)phenyl]pyrimidin-2-amine as a scaffold for the synthesis of inhibitors of Bcr-Abl.
Arioli F; Borrelli S; Colombo F; Falchi F; Filippi I; Crespan E; Naldini A; Scalia G; Silvani A; Maga G; Carraro F; Botta M; Passarella D
ChemMedChem; 2011 Nov; 6(11):2009-18. PubMed ID: 21990039
[TBL] [Abstract][Full Text] [Related]
12. 7-Chloroquinolinotriazoles: synthesis by the azide-alkyne cycloaddition click chemistry, antimalarial activity, cytotoxicity and SAR studies.
Pereira GR; Brandão GC; Arantes LM; de Oliveira HA; de Paula RC; do Nascimento MF; dos Santos FM; da Rocha RK; Lopes JC; de Oliveira AB
Eur J Med Chem; 2014 Feb; 73():295-309. PubMed ID: 24469080
[TBL] [Abstract][Full Text] [Related]
13. Structure-based virtual screening of Src kinase inhibitors.
Lee K; Kim J; Jeong KW; Lee KW; Lee Y; Song JY; Kim MS; Lee GS; Kim Y
Bioorg Med Chem; 2009 Apr; 17(8):3152-61. PubMed ID: 19321350
[TBL] [Abstract][Full Text] [Related]
14. Novel oxazolo[4,5-g]quinazolin-2(1H)-ones: dual inhibitors of EGFR and Src protein tyrosine kinases.
Lin J; Shen W; Xue J; Sun J; Zhang X; Zhang C
Eur J Med Chem; 2012 Sep; 55():39-48. PubMed ID: 22818848
[TBL] [Abstract][Full Text] [Related]
15. Synthesis, biological evaluation, and molecular docking studies of novel 1,3,4-oxadiazole derivatives possessing benzotriazole moiety as FAK inhibitors with anticancer activity.
Zhang S; Luo Y; He LQ; Liu ZJ; Jiang AQ; Yang YH; Zhu HL
Bioorg Med Chem; 2013 Jul; 21(13):3723-9. PubMed ID: 23673215
[TBL] [Abstract][Full Text] [Related]
16. Novel purine-based fluoroaryl-1,2,3-triazoles as neuroprotecting agents: synthesis, neuronal cell culture investigations, and CDK5 docking studies.
Nair N; Kudo W; Smith MA; Abrol R; Goddard WA; Reddy VP
Bioorg Med Chem Lett; 2011 Jul; 21(13):3957-61. PubMed ID: 21641213
[TBL] [Abstract][Full Text] [Related]
17. Exploration of acridine scaffold as a potentially interesting scaffold for discovering novel multi-target VEGFR-2 and Src kinase inhibitors.
Luan X; Gao C; Zhang N; Chen Y; Sun Q; Tan C; Liu H; Jin Y; Jiang Y
Bioorg Med Chem; 2011 Jun; 19(11):3312-9. PubMed ID: 21576023
[TBL] [Abstract][Full Text] [Related]
18. 1,2,3-Triazole-totarol conjugates as potent PIP5K1α lipid kinase inhibitors.
Haidar S; Amesty Á; Oramas-Royo S; Götz C; El-Awaad E; Kaiser J; Bödecker S; Arnold A; Aichele D; Amaro-Luis JM; Estévez-Braun A; Jose J
Bioorg Med Chem; 2024 May; 105():117727. PubMed ID: 38669736
[TBL] [Abstract][Full Text] [Related]
19. New triazole derivatives as antifungal agents: synthesis via click reaction, in vitro evaluation and molecular docking studies.
Zou Y; Zhao Q; Liao J; Hu H; Yu S; Chai X; Xu M; Wu Q
Bioorg Med Chem Lett; 2012 Apr; 22(8):2959-62. PubMed ID: 22437114
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and biological evaluation of a triazole-based library of pyrido[2,3-d]pyrimidines as FGFR3 tyrosine kinase inhibitors.
Le Corre L; Girard AL; Aubertin J; Radvanyi F; Benoist-Lasselin C; Jonquoy A; Mugniery E; Legeai-Mallet L; Busca P; Le Merrer Y
Org Biomol Chem; 2010 May; 8(9):2164-73. PubMed ID: 20401393
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]