These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

123 related articles for article (PubMed ID: 27078680)

  • 1. Identification of Drug-Like Inhibitors of Insulin-Regulated Aminopeptidase Through Small-Molecule Screening.
    Engen K; Rosenström U; Axelsson H; Konda V; Dahllund L; Otrocka M; Sigmundsson K; Nikolaou A; Vauquelin G; Hallberg M; Jenmalm Jensen A; Lundbäck T; Larhed M
    Assay Drug Dev Technol; 2016 Apr; 14(3):180-93. PubMed ID: 27078680
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Potent macrocyclic inhibitors of insulin-regulated aminopeptidase (IRAP) by olefin ring-closing metathesis.
    Andersson H; Demaegdt H; Johnsson A; Vauquelin G; Lindeberg G; Hallberg M; Erdelyi M; Karlen A; Hallberg A
    J Med Chem; 2011 Jun; 54(11):3779-92. PubMed ID: 21476495
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Virtual Screening for Transition State Analogue Inhibitors of IRAP Based on Quantum Mechanically Derived Reaction Coordinates.
    Svensson F; Engen K; Lundbäck T; Larhed M; Sköld C
    J Chem Inf Model; 2015 Sep; 55(9):1984-93. PubMed ID: 26252078
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Identification and characterization of a new cognitive enhancer based on inhibition of insulin-regulated aminopeptidase.
    Albiston AL; Morton CJ; Ng HL; Pham V; Yeatman HR; Ye S; Fernando RN; De Bundel D; Ascher DB; Mendelsohn FA; Parker MW; Chai SY
    FASEB J; 2008 Dec; 22(12):4209-17. PubMed ID: 18716029
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Binding to and Inhibition of Insulin-Regulated Aminopeptidase by Macrocyclic Disulfides Enhances Spine Density.
    Diwakarla S; Nylander E; Grönbladh A; Vanga SR; Khan YS; Gutiérrez-de-Terán H; Ng L; Pham V; Sävmarker J; Lundbäck T; Jenmalm-Jensen A; Andersson H; Engen K; Rosenström U; Larhed M; Åqvist J; Chai SY; Hallberg M
    Mol Pharmacol; 2016 Apr; 89(4):413-24. PubMed ID: 26769413
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Binding of "AT4 receptor" ligands to insulin regulated aminopeptidase (IRAP) in intact Chinese hamster ovary cells.
    Demaegdt H; Gard P; De Backer JP; Lukaszuk A; Szemenyei E; Tóth G; Tourwé D; Vauquelin G
    Mol Cell Endocrinol; 2011 Jun; 339(1-2):34-44. PubMed ID: 21457753
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Disulfide cyclized tripeptide analogues of angiotensin IV as potent and selective inhibitors of insulin-regulated aminopeptidase (IRAP).
    Andersson H; Demaegdt H; Vauquelin G; Lindeberg G; Karlén A; Hallberg M; Erdélyi M; Hallberg A
    J Med Chem; 2010 Nov; 53(22):8059-71. PubMed ID: 21047126
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Aryl Sulfonamide Inhibitors of Insulin-Regulated Aminopeptidase Enhance Spine Density in Primary Hippocampal Neuron Cultures.
    Diwakarla S; Nylander E; Grönbladh A; Vanga SR; Shamsudin Y; Gutiérrez-de-Terán H; Sävmarker J; Ng L; Pham V; Lundbäck T; Jenmalm-Jensen A; Svensson R; Artursson P; Zelleroth S; Engen K; Rosenström U; Larhed M; Åqvist J; Chai SY; Hallberg M
    ACS Chem Neurosci; 2016 Oct; 7(10):1383-1392. PubMed ID: 27501164
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Identification and development of specific inhibitors for insulin-regulated aminopeptidase as a new class of cognitive enhancers.
    Albiston AL; Diwakarla S; Fernando RN; Mountford SJ; Yeatman HR; Morgan B; Pham V; Holien JK; Parker MW; Thompson PE; Chai SY
    Br J Pharmacol; 2011 Sep; 164(1):37-47. PubMed ID: 21470200
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Selective labeling of IRAP by the tritiated AT(4) receptor ligand [3H]Angiotensin IV and its stable analog [3H]AL-11.
    Demaegdt H; Lukaszuk A; De Buyser E; De Backer JP; Szemenyei E; Tóth G; Chakravarthy S; Panicker M; Michotte Y; Tourwé D; Vauquelin G
    Mol Cell Endocrinol; 2009 Nov; 311(1-2):77-86. PubMed ID: 19643163
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Cyclic insulin-regulated aminopeptidase (IRAP)/AT4 receptor ligands.
    Axén A; Lindeberg G; Demaegdt H; Vauquelin G; Karlén A; Hallberg M
    J Pept Sci; 2006 Nov; 12(11):705-13. PubMed ID: 16967438
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors.
    Engen K; Vanga SR; Lundbäck T; Agalo F; Konda V; Jensen AJ; Åqvist J; Gutiérrez-de-Terán H; Hallberg M; Larhed M; Rosenström U
    ChemistryOpen; 2020 Mar; 9(3):325-337. PubMed ID: 32154052
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Small potent ligands to the insulin-regulated aminopeptidase (IRAP)/AT(4) receptor.
    Axén A; Andersson H; Lindeberg G; Rönnholm H; Kortesmaa J; Demaegdt H; Vauquelin G; Karlén A; Hallberg M
    J Pept Sci; 2007 Jul; 13(7):434-44. PubMed ID: 17559064
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Regulation of insulin-regulated membrane aminopeptidase activity by its C-terminal domain.
    Ascher DB; Cromer BA; Morton CJ; Volitakis I; Cherny RA; Albiston AL; Chai SY; Parker MW
    Biochemistry; 2011 Apr; 50(13):2611-22. PubMed ID: 21348480
    [TBL] [Abstract][Full Text] [Related]  

  • 15. The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds.
    Gising J; Honarnejad S; Bras M; Baillie GL; McElroy SP; Jones PS; Morrison A; Beveridge J; Hallberg M; Larhed M
    Int J Mol Sci; 2024 Apr; 25(7):. PubMed ID: 38612894
    [TBL] [Abstract][Full Text] [Related]  

  • 16. [3H]IVDE77, a novel radioligand with high affinity and selectivity for the insulin-regulated aminopeptidase.
    Nikolaou A; Van den Eynde I; Tourwé D; Vauquelin G; Tóth G; Mallareddy JR; Poglitsch M; Van Ginderachter JA; Vanderheyden PM
    Eur J Pharmacol; 2013 Feb; 702(1-3):93-102. PubMed ID: 23376157
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Angiotensin IV displays only low affinity for native insulin-regulated aminopeptidase (IRAP).
    Demaegdt H; De Backer JP; Lukaszuk A; Tóth G; Szemenyei E; Tourwé D; Vauquelin G
    Fundam Clin Pharmacol; 2012 Apr; 26(2):194-7. PubMed ID: 21477268
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Involvement of insulin-regulated aminopeptidase and/or aminopeptidase N in the angiotensin IV-induced effect on dopamine release in the striatum of the rat.
    Stragier B; Demaegdt H; De Bundel D; Smolders I; Sarre S; Vauquelin G; Ebinger G; Michotte Y; Vanderheyden P
    Brain Res; 2007 Feb; 1131(1):97-105. PubMed ID: 17169335
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Effects of ligands or substrate of insulin-regulated aminopeptidase (IRAP) on trophoblast invasion.
    Cohen M; Wuillemin C; Chai SY; Bischof P
    J Pept Sci; 2008 Jul; 14(7):883-7. PubMed ID: 18275097
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Inhibition of Insulin-Regulated Aminopeptidase (IRAP) by Arylsulfonamides.
    Borhade SR; Rosenström U; Sävmarker J; Lundbäck T; Jenmalm-Jensen A; Sigmundsson K; Axelsson H; Svensson F; Konda V; Sköld C; Larhed M; Hallberg M
    ChemistryOpen; 2014 Dec; 3(6):256-63. PubMed ID: 25558444
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.