175 related articles for article (PubMed ID: 2709373)
1. Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors.
Jacobson KA; Barone S; Kammula U; Stiles GL
J Med Chem; 1989 May; 32(5):1043-51. PubMed ID: 2709373
[TBL] [Abstract][Full Text] [Related]
2. Trifunctional agents as a design strategy for tailoring ligand properties: irreversible inhibitors of A1 adenosine receptors.
Boring DL; Ji XD; Zimmet J; Taylor KE; Stiles GL; Jacobson KA
Bioconjug Chem; 1991; 2(2):77-88. PubMed ID: 1868116
[TBL] [Abstract][Full Text] [Related]
3. High affinity acylating antagonists for the A1 adenosine receptor: identification of binding subunit.
Stiles GL; Jacobson KA
Mol Pharmacol; 1988 Dec; 34(6):724-8. PubMed ID: 3200248
[TBL] [Abstract][Full Text] [Related]
4. Evidence of spare A1-adenosine receptors in guinea pig atrioventricular node.
Dennis D; Jacobson K; Belardinelli L
Am J Physiol; 1992 Mar; 262(3 Pt 2):H661-71. PubMed ID: 1558173
[TBL] [Abstract][Full Text] [Related]
5. 125I-labeled 8-phenylxanthine derivatives: antagonist radioligands for adenosine A1 receptors.
Linden J; Patel A; Earl CQ; Craig RH; Daluge SM
J Med Chem; 1988 Apr; 31(4):745-51. PubMed ID: 3351850
[TBL] [Abstract][Full Text] [Related]
6. 8-Substituted xanthines as antagonists at A1- and A2-adenosine receptors.
Jacobson KA; de la Cruz R; Schulick R; Kiriasis L; Padgett W; Pfleiderer W; Kirk KL; Neumeyer JL; Daly JW
Biochem Pharmacol; 1988 Oct; 37(19):3653-61. PubMed ID: 3178879
[TBL] [Abstract][Full Text] [Related]
7. A functionalized congener approach to adenosine receptor antagonists: amino acid conjugates of 1,3-dipropylxanthine.
Jacobson KA; Kirk KL; Padgett WL; Daly JW
Mol Pharmacol; 1986 Feb; 29(2):126-33. PubMed ID: 3005825
[TBL] [Abstract][Full Text] [Related]
8. Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.
Jacobson KA; Kiriasis L; Barone S; Bradbury BJ; Kammula U; Campagne JM; Secunda S; Daly JW; Neumeyer JL; Pfleiderer W
J Med Chem; 1989 Aug; 32(8):1873-9. PubMed ID: 2754711
[TBL] [Abstract][Full Text] [Related]
9. [3H]xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: an antagonist radioligand for adenosine receptors.
Jacobson KA; Ukena D; Kirk KL; Daly JW
Proc Natl Acad Sci U S A; 1986 Jun; 83(11):4089-93. PubMed ID: 3012550
[TBL] [Abstract][Full Text] [Related]
10. Structure-activity relationships of 8-styrylxanthines as A2-selective adenosine antagonists.
Jacobson KA; Gallo-Rodriguez C; Melman N; Fischer B; Maillard M; van Bergen A; van Galen PJ; Karton Y
J Med Chem; 1993 May; 36(10):1333-42. PubMed ID: 8496902
[TBL] [Abstract][Full Text] [Related]
11. Species differences in structure-activity relationships of adenosine agonists and xanthine antagonists at brain A1 adenosine receptors.
Ukena D; Jacobson KA; Padgett WL; Ayala C; Shamim MT; Kirk KL; Olsson RO; Daly JW
FEBS Lett; 1986 Dec; 209(1):122-8. PubMed ID: 3803571
[TBL] [Abstract][Full Text] [Related]
12. Analogues of 1,3-dipropyl-8-phenylxanthine: enhancement of selectivity at A1-adenosine receptors by aryl substituents.
Daly JW; Padgett WL; Shamim MT
J Med Chem; 1986 Aug; 29(8):1520-4. PubMed ID: 3016270
[TBL] [Abstract][Full Text] [Related]
13. Linear and proximal benzo-separated alkylated xanthines as adenosine-receptor antagonists.
Schneller SW; Ibay AC; Christ WJ; Bruns RF
J Med Chem; 1989 Oct; 32(10):2247-54. PubMed ID: 2795597
[TBL] [Abstract][Full Text] [Related]
14. Xanthine derivatives as antagonists at A1 and A2 adenosine receptors.
Schwabe U; Ukena D; Lohse MJ
Naunyn Schmiedebergs Arch Pharmacol; 1985 Sep; 330(3):212-21. PubMed ID: 2997628
[TBL] [Abstract][Full Text] [Related]
15. Functionalized congeners of 1,3-dipropyl-8-phenylxanthine: potent antagonists for adenosine receptors that modulate membrane adenylate cyclase in pheochromocytoma cells, platelets and fat cells.
Ukena D; Daly JW; Kirk KL; Jacobson KA
Life Sci; 1986 Mar; 38(9):797-807. PubMed ID: 3005794
[TBL] [Abstract][Full Text] [Related]
16. 8-Aryl-and 8-cycloalkyl-1,3-dipropylxanthines: further potent and selective antagonists for A1-adenosine receptors.
Shamim MT; Ukena D; Padgett WL; Hong O; Daly JW
J Med Chem; 1988 Mar; 31(3):613-7. PubMed ID: 3346878
[TBL] [Abstract][Full Text] [Related]
17. Potent adenosine receptor antagonists that are selective for the A1 receptor subtype.
Martinson EA; Johnson RA; Wells JN
Mol Pharmacol; 1987 Mar; 31(3):247-52. PubMed ID: 3561384
[TBL] [Abstract][Full Text] [Related]
18. Probing the adenosine receptor with adenosine and xanthine biotin conjugates.
Jacobson KA; Kirk KL; Padgett W; Daly JW
FEBS Lett; 1985 May; 184(1):30-5. PubMed ID: 2985445
[TBL] [Abstract][Full Text] [Related]
19. 8-Polycycloalkyl-1,3-dipropylxanthines as potent and selective antagonists for A1-adenosine receptors.
Shimada J; Suzuki F; Nonaka H; Ishii A
J Med Chem; 1992 Mar; 35(5):924-30. PubMed ID: 1548682
[TBL] [Abstract][Full Text] [Related]
20. Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions.
Kim SA; Marshall MA; Melman N; Kim HS; Müller CE; Linden J; Jacobson KA
J Med Chem; 2002 May; 45(11):2131-8. PubMed ID: 12014951
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
