BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

98 related articles for article (PubMed ID: 27100033)

  • 1. The combination of quinazoline and chalcone moieties leads to novel potent heterodimeric modulators of breast cancer resistance protein (BCRP/ABCG2).
    Kraege S; Stefan K; Juvale K; Ross T; Willmes T; Wiese M
    Eur J Med Chem; 2016 Jul; 117():212-29. PubMed ID: 27100033
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and biological investigation of 2,4-substituted quinazolines as highly potent inhibitors of breast cancer resistance protein (ABCG2).
    Krapf MK; Gallus J; Wiese M
    Eur J Med Chem; 2017 Oct; 139():587-611. PubMed ID: 28841513
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2).
    Juvale K; Gallus J; Wiese M
    Bioorg Med Chem; 2013 Dec; 21(24):7858-73. PubMed ID: 24184213
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and Biological Evaluation of 4-Anilino-quinazolines and -quinolines as Inhibitors of Breast Cancer Resistance Protein (ABCG2).
    Krapf MK; Wiese M
    J Med Chem; 2016 Jun; 59(11):5449-61. PubMed ID: 27148793
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Investigation of chalcones and benzochalcones as inhibitors of breast cancer resistance protein.
    Juvale K; Pape VF; Wiese M
    Bioorg Med Chem; 2012 Jan; 20(1):346-55. PubMed ID: 22112540
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design of inhibitors of BCRP/ABCG2.
    Juvale K; Wiese M
    Future Med Chem; 2015 Aug; 7(12):1521-7. PubMed ID: 26293476
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Functionalized chalcones as selective inhibitors of P-glycoprotein and breast cancer resistance protein.
    Liu XL; Tee HW; Go ML
    Bioorg Med Chem; 2008 Jan; 16(1):171-80. PubMed ID: 17964170
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Symmetric bis-chalcones as a new type of breast cancer resistance protein inhibitors with a mechanism different from that of chromones.
    Winter E; Devantier Neuenfeldt P; Chiaradia-Delatorre LD; Gauthier C; Yunes RA; Nunes RJ; Creczynski-Pasa TB; Di Pietro A
    J Med Chem; 2014 Apr; 57(7):2930-41. PubMed ID: 24611893
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel chalcone and flavone derivatives as selective and dual inhibitors of the transport proteins ABCB1 and ABCG2.
    Silbermann K; Shah CP; Sahu NU; Juvale K; Stefan SM; Kharkar PS; Wiese M
    Eur J Med Chem; 2019 Feb; 164():193-213. PubMed ID: 30594677
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Modulation of breast cancer resistance protein (BCRP/ABCG2) by non-basic chalcone analogues.
    Han Y; Riwanto M; Go ML; Ee PL
    Eur J Pharm Sci; 2008 Sep; 35(1-2):30-41. PubMed ID: 18598762
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Biological evaluation of non-basic chalcone CYB-2 as a dual ABCG2/ABCB1 inhibitor.
    Cai CY; Zhang W; Wang JQ; Lei ZN; Zhang YK; Wang YJ; Gupta P; Tan CP; Wang B; Chen ZS
    Biochem Pharmacol; 2020 May; 175():113848. PubMed ID: 32044354
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and biological evaluation of quinazoline derivatives - A SAR study of novel inhibitors of ABCG2.
    Krapf MK; Gallus J; Spindler A; Wiese M
    Eur J Med Chem; 2019 Jan; 161():506-525. PubMed ID: 30390439
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Structure activity relationships, multidrug resistance reversal and selectivity of heteroarylphenyl ABCG2 inhibitors.
    Köhler SC; Vahdati S; Scholz MS; Wiese M
    Eur J Med Chem; 2018 Feb; 146():483-500. PubMed ID: 29407974
    [TBL] [Abstract][Full Text] [Related]  

  • 14. New structure-activity relationships of chalcone inhibitors of breast cancer resistance protein: polyspecificity toward inhibition and critical substitutions against cytotoxicity.
    Rangel LP; Winter E; Gauthier C; Terreux R; Chiaradia-Delatorre LD; Mascarello A; Nunes RJ; Yunes RA; Creczynski-Pasa TB; Macalou S; Lorendeau D; Baubichon-Cortay H; Ferreira-Pereira A; Di Pietro A
    Drug Des Devel Ther; 2013; 7():1043-52. PubMed ID: 24109177
    [TBL] [Abstract][Full Text] [Related]  

  • 15. 2,4,6-Substituted Quinazolines with Extraordinary Inhibitory Potency toward ABCG2.
    Krapf MK; Gallus J; Namasivayam V; Wiese M
    J Med Chem; 2018 Sep; 61(17):7952-7976. PubMed ID: 30075623
    [TBL] [Abstract][Full Text] [Related]  

  • 16. 4-Anilino-2-pyridylquinazolines and -pyrimidines as Highly Potent and Nontoxic Inhibitors of Breast Cancer Resistance Protein (ABCG2).
    Krapf MK; Gallus J; Wiese M
    J Med Chem; 2017 May; 60(10):4474-4495. PubMed ID: 28471656
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and Investigation of Tetrahydro-β-carboline Derivatives as Inhibitors of the Breast Cancer Resistance Protein (ABCG2).
    Spindler A; Stefan K; Wiese M
    J Med Chem; 2016 Jul; 59(13):6121-35. PubMed ID: 27280693
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Investigation of chalcones as selective inhibitors of the breast cancer resistance protein: critical role of methoxylation in both inhibition potency and cytotoxicity.
    Valdameri G; Gauthier C; Terreux R; Kachadourian R; Day BJ; Winnischofer SM; Rocha ME; Frachet V; Ronot X; Di Pietro A; Boumendjel A
    J Med Chem; 2012 Apr; 55(7):3193-200. PubMed ID: 22449016
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Optimization of Acryloylphenylcarboxamides as Inhibitors of ABCG2 and Comparison with Acryloylphenylcarboxylates.
    Kraege S; Stefan K; Köhler SC; Wiese M
    ChemMedChem; 2016 Nov; 11(22):2547-2558. PubMed ID: 27785905
    [TBL] [Abstract][Full Text] [Related]  

  • 20. New, highly potent and non-toxic, chromone inhibitors of the human breast cancer resistance protein ABCG2.
    Pires ADRA; Lecerf-Schmidt F; Guragossian N; Pazinato J; Gozzi GJ; Winter E; Valdameri G; Veale A; Boumendjel A; Di Pietro A; Pérès B
    Eur J Med Chem; 2016 Oct; 122():291-301. PubMed ID: 27376492
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 5.