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9. Small Molecule Inhibitors of DYRK1A Identified by Computational and Experimental Approaches. Yoon HR; Balupuri A; Choi KE; Kang NS Int J Mol Sci; 2020 Sep; 21(18):. PubMed ID: 32957634 [TBL] [Abstract][Full Text] [Related]
10. Identification of a DYRK1A Inhibitor that Induces Degradation of the Target Kinase using Co-chaperone CDC37 fused with Luciferase nanoKAZ. Sonamoto R; Kii I; Koike Y; Sumida Y; Kato-Sumida T; Okuno Y; Hosoya T; Hagiwara M Sci Rep; 2015 Aug; 5():12728. PubMed ID: 26234946 [TBL] [Abstract][Full Text] [Related]
11. Differential maturation and chaperone dependence of the paralogous protein kinases DYRK1A and DYRK1B. Papenfuss M; Lützow S; Wilms G; Babendreyer A; Flaßhoff M; Kunick C; Becker W Sci Rep; 2022 Feb; 12(1):2393. PubMed ID: 35165364 [TBL] [Abstract][Full Text] [Related]
12. Activation, regulation, and inhibition of DYRK1A. Becker W; Sippl W FEBS J; 2011 Jan; 278(2):246-56. PubMed ID: 21126318 [TBL] [Abstract][Full Text] [Related]
13. Harmine specifically inhibits protein kinase DYRK1A and interferes with neurite formation. Göckler N; Jofre G; Papadopoulos C; Soppa U; Tejedor FJ; Becker W FEBS J; 2009 Nov; 276(21):6324-37. PubMed ID: 19796173 [TBL] [Abstract][Full Text] [Related]
14. 10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acids are selective inhibitors of DYRK1A. Falke H; Chaikuad A; Becker A; Loaëc N; Lozach O; Abu Jhaisha S; Becker W; Jones PG; Preu L; Baumann K; Knapp S; Meijer L; Kunick C J Med Chem; 2015 Apr; 58(7):3131-43. PubMed ID: 25730262 [TBL] [Abstract][Full Text] [Related]
15. Systematic diversification of benzylidene heterocycles yields novel inhibitor scaffolds selective for Dyrk1A, Clk1 and CK2. Mariano M; Hartmann RW; Engel M Eur J Med Chem; 2016 Apr; 112():209-216. PubMed ID: 26896709 [TBL] [Abstract][Full Text] [Related]
16. Dual-Specificity Tyrosine Phosphorylation-Regulated Kinase 1A (DYRK1A) Inhibitors as Potential Therapeutics. Jarhad DB; Mashelkar KK; Kim HR; Noh M; Jeong LS J Med Chem; 2018 Nov; 61(22):9791-9810. PubMed ID: 29985601 [TBL] [Abstract][Full Text] [Related]
17. Synthesis and in vitro evaluation of diverse heterocyclic diphenolic compounds as inhibitors of DYRK1A. Zhou Q; Reekie TA; Abbassi RH; Indurthi Venkata D; Font JS; Ryan RM; Munoz L; Kassiou M Bioorg Med Chem; 2018 Dec; 26(22):5852-5869. PubMed ID: 30401502 [TBL] [Abstract][Full Text] [Related]
18. Dyrk1a is required for craniofacial development in Xenopus laevis. Johnson HK; Wahl SE; Sesay F; Litovchick L; Dickinson AJ Dev Biol; 2024 Jul; 511():63-75. PubMed ID: 38621649 [TBL] [Abstract][Full Text] [Related]
19. Down's-syndrome-related kinase Dyrk1A modulates the p120-catenin-Kaiso trajectory of the Wnt signaling pathway. Hong JY; Park JI; Lee M; Muñoz WA; Miller RK; Ji H; Gu D; Ezan J; Sokol SY; McCrea PD J Cell Sci; 2012 Feb; 125(Pt 3):561-9. PubMed ID: 22389395 [TBL] [Abstract][Full Text] [Related]
20. DYRK1A phosphorylates caspase 9 at an inhibitory site and is potently inhibited in human cells by harmine. Seifert A; Allan LA; Clarke PR FEBS J; 2008 Dec; 275(24):6268-80. PubMed ID: 19016842 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]