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2. Incorporation of fluorinated phenylalanine generates highly specific inhibitor of proteasome's chymotrypsin-like sites. Geurink PP; Liu N; Spaans MP; Downey SL; van den Nieuwendijk AM; van der Marel GA; Kisselev AF; Florea BI; Overkleeft HS J Med Chem; 2010 Mar; 53(5):2319-23. PubMed ID: 20131905 [TBL] [Abstract][Full Text] [Related]
3. Selective inhibitor of proteasome's caspase-like sites sensitizes cells to specific inhibition of chymotrypsin-like sites. Britton M; Lucas MM; Downey SL; Screen M; Pletnev AA; Verdoes M; Tokhunts RA; Amir O; Goddard AL; Pelphrey PM; Wright DL; Overkleeft HS; Kisselev AF Chem Biol; 2009 Dec; 16(12):1278-89. PubMed ID: 20064438 [TBL] [Abstract][Full Text] [Related]
4. Kinetic characterization of the chymotryptic activity of the 20S proteasome. Stein RL; Melandri F; Dick L Biochemistry; 1996 Apr; 35(13):3899-908. PubMed ID: 8672420 [TBL] [Abstract][Full Text] [Related]
5. Activation of Chymotrypsin-Like Activity of the Proteasome during Ischemia Induces Myocardial Dysfunction and Death. Sanchez G; Berrios D; Olmedo I; Pezoa J; Riquelme JA; Montecinos L; Pedrozo Z; Donoso P PLoS One; 2016; 11(8):e0161068. PubMed ID: 27529620 [TBL] [Abstract][Full Text] [Related]
6. Methylation of green tea polyphenols affects their binding to and inhibitory poses of the proteasome beta5 subunit. Daniel KG; Landis-Piwowar KR; Chen D; Wan SB; Chan TH; Dou QP Int J Mol Med; 2006 Oct; 18(4):625-32. PubMed ID: 16964415 [TBL] [Abstract][Full Text] [Related]
7. Apigenin, chrysin, and luteolin selectively inhibit chymotrypsin-like and trypsin-like proteasome catalytic activities in tumor cells. Wu YX; Fang X Planta Med; 2010 Feb; 76(2):128-32. PubMed ID: 19653143 [TBL] [Abstract][Full Text] [Related]
8. Discovery of novel non-covalent inhibitors selective to the β5-subunit of the human 20S proteasome. Xu K; Wang K; Yang Y; Yan DA; Huang L; Chen CH; Xiao Z Eur J Med Chem; 2015 Jun; 98():61-8. PubMed ID: 26005024 [TBL] [Abstract][Full Text] [Related]
9. Cytoprotective effects of proteasome beta5 subunit overexpression in lens epithelial cells. Liu Y; Liu X; Zhang T; Luna C; Liton PB; Gonzalez P Mol Vis; 2007 Jan; 13():31-8. PubMed ID: 17262013 [TBL] [Abstract][Full Text] [Related]
10. Molecular modeling on porphyrin derivatives as β5 subunit inhibitor of 20S proteasome. Arba M; Nur-Hidayat A; Ruslin ; Yusuf M; Sumarlin ; Hertadi R; Wahyudi ST; Surantaadmaja SI; Tjahjono DH Comput Biol Chem; 2018 Jun; 74():230-238. PubMed ID: 29674291 [TBL] [Abstract][Full Text] [Related]
11. Inhibitors of the eukaryotic 20S proteasome core particle: a structural approach. Groll M; Huber R Biochim Biophys Acta; 2004 Nov; 1695(1-3):33-44. PubMed ID: 15571807 [TBL] [Abstract][Full Text] [Related]
12. Multicolor monitoring of the proteasome's catalytic signature. Priestman MA; Wang Q; Jernigan FE; Chowdhury R; Schmidt M; Lawrence DS ACS Chem Biol; 2015 Feb; 10(2):433-40. PubMed ID: 25347733 [TBL] [Abstract][Full Text] [Related]
13. Development of novel peptidomimetics containing a vinyl sulfone moiety as proteasome inhibitors. Ettari R; Bonaccorso C; Micale N; Heindl C; Schirmeister T; Calabrò ML; Grasso S; Zappalà M ChemMedChem; 2011 Jul; 6(7):1228-37. PubMed ID: 21506279 [TBL] [Abstract][Full Text] [Related]
14. Identification of noncovalent proteasome inhibitors with high selectivity for chymotrypsin-like activity by a multistep structure-based virtual screening. Di Giovanni C; Ettari R; Sarno S; Rotondo A; Bitto A; Squadrito F; Altavilla D; Schirmeister T; Novellino E; Grasso S; Zappalà M; Lavecchia A Eur J Med Chem; 2016 Oct; 121():578-591. PubMed ID: 27318981 [TBL] [Abstract][Full Text] [Related]
15. Bifunctional inhibitors of the trypsin-like activity of eukaryotic proteasomes. Loidl G; Groll M; Musiol HJ; Ditzel L; Huber R; Moroder L Chem Biol; 1999 Apr; 6(4):197-204. PubMed ID: 10099130 [TBL] [Abstract][Full Text] [Related]
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