BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

306 related articles for article (PubMed ID: 27138243)

  • 1. Synthesis and in-vitro reactivation screening of imidazolium aldoximes as reactivators of sarin and VX-inhibited human acetylcholinesterase (hAChE).
    Sharma R; Gupta B; Sahu AK; Acharya J; Satnami ML; Ghosh KK
    Chem Biol Interact; 2016 Nov; 259(Pt B):85-92. PubMed ID: 27138243
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and in vitro kinetic evaluation of N-thiazolylacetamido monoquaternary pyridinium oximes as reactivators of sarin, O-ethylsarin and VX inhibited human acetylcholinesterase (hAChE).
    Valiveti AK; Bhalerao UM; Acharya J; Karade HN; Acharya BN; Raviraju G; Halve AK; Kaushik MP
    Bioorg Med Chem; 2015 Aug; 23(15):4899-4910. PubMed ID: 26043948
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and in vitro evaluation of bis-quaternary 2-(hydroxyimino)-N-(pyridin-3-yl)acetamide derivatives as reactivators against sarin and VX inhibited human acetylcholinesterase (hAChE).
    Karade HN; Valiveti AK; Acharya J; Kaushik MP
    Bioorg Med Chem; 2014 May; 22(9):2684-91. PubMed ID: 24721830
    [TBL] [Abstract][Full Text] [Related]  

  • 4. In vitro reactivation of acetylcholinesterase using the oxime K027.
    Kuca K; Kassa J
    Vet Hum Toxicol; 2004 Feb; 46(1):15-8. PubMed ID: 14748409
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and in vitro reactivation study of isonicotinamide derivatives of 2-(hydroxyimino)-N-(pyridin-3-yl)acetamide as reactivators of Sarin and VX inhibited human acetylcholinesterase (hAChE).
    Karade HN; Raviraju G; Acharya BN; Valiveti AK; Bhalerao U; Acharya J
    Bioorg Med Chem; 2016 Sep; 24(18):4171-4176. PubMed ID: 27450532
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Interactions between xylene-linked carbamoyl bis-pyridinium mono-oximes and organophosphates inhibited-AChE: a kinetic study.
    Sharma R; Gupta B; Acharya J; Kaushik MP; Ghosh KK
    Toxicology; 2014 Feb; 316():1-8. PubMed ID: 24345352
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and in vitro kinetic study of novel mono-pyridinium oximes as reactivators of organophosphorus (OP) inhibited human acetylcholinesterase (hAChE).
    Valiveti AK; Bhalerao UM; Acharya J; Karade HN; Gundapu R; Halve AK; Kaushik MP
    Chem Biol Interact; 2015 Jul; 237():125-32. PubMed ID: 26070418
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Rational design, synthesis, and evaluation of uncharged, "smart" bis-oxime antidotes of organophosphate-inhibited human acetylcholinesterase.
    Gorecki L; Gerlits O; Kong X; Cheng X; Blumenthal DK; Taylor P; Ballatore C; Kovalevsky A; Radić Z
    J Biol Chem; 2020 Mar; 295(13):4079-4092. PubMed ID: 32019865
    [TBL] [Abstract][Full Text] [Related]  

  • 9. In vitro reactivation of sarin-inhibited human acetylcholinesterase (AChE) by bis-pyridinium oximes connected by xylene linkers.
    Acharya J; Dubey DK; Srivastava AK; Raza SK
    Toxicol In Vitro; 2011 Feb; 25(1):251-6. PubMed ID: 20688148
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and in vitro evaluation of neutral aryloximes as reactivators of Electrophorus eel acetylcholinesterase inhibited by NEMP, a VX surrogate.
    Cavalcante SFA; Kitagawa DAS; Rodrigues RB; Bernardo LB; da Silva TN; Dos Santos WV; Correa ABA; de Almeida JSFD; França TCC; Kuča K; Simas ABC
    Chem Biol Interact; 2019 Aug; 309():108682. PubMed ID: 31163137
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Efficacy of novel phenoxyalkyl pyridinium oximes as brain-penetrating reactivators of cholinesterase inhibited by surrogates of sarin and VX.
    Chambers JE; Chambers HW; Funck KE; Meek EC; Pringle RB; Ross MK
    Chem Biol Interact; 2016 Nov; 259(Pt B):154-159. PubMed ID: 27387540
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Productive reorientation of a bound oxime reactivator revealed in room temperature X-ray structures of native and VX-inhibited human acetylcholinesterase.
    Gerlits O; Kong X; Cheng X; Wymore T; Blumenthal DK; Taylor P; Radić Z; Kovalevsky A
    J Biol Chem; 2019 Jul; 294(27):10607-10618. PubMed ID: 31138650
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Reactivating potency of obidoxime, pralidoxime, HI 6 and HLö 7 in human erythrocyte acetylcholinesterase inhibited by highly toxic organophosphorus compounds.
    Worek F; Widmann R; Knopff O; Szinicz L
    Arch Toxicol; 1998 Mar; 72(4):237-43. PubMed ID: 9587020
    [TBL] [Abstract][Full Text] [Related]  

  • 14. HI-6 assisted catalytic scavenging of VX by acetylcholinesterase choline binding site mutants.
    Maček Hrvat N; Žunec S; Taylor P; Radić Z; Kovarik Z
    Chem Biol Interact; 2016 Nov; 259(Pt B):148-153. PubMed ID: 27083141
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Oxime-mediated in vitro reactivation kinetic analysis of organophosphates-inhibited human and electric eel acetylcholinesterase.
    Sahu AK; Sharma R; Gupta B; Musilek K; Kuca K; Acharya J; Ghosh KK
    Toxicol Mech Methods; 2016 Jun; 26(5):319-26. PubMed ID: 27101948
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Centrally acting oximes in reactivation of tabun-phosphoramidated AChE.
    Kovarik Z; Maček N; Sit RK; Radić Z; Fokin VV; Barry Sharpless K; Taylor P
    Chem Biol Interact; 2013 Mar; 203(1):77-80. PubMed ID: 22960624
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Enzyme-kinetic investigation of different sarin analogues reacting with human acetylcholinesterase and butyrylcholinesterase.
    Bartling A; Worek F; Szinicz L; Thiermann H
    Toxicology; 2007 Apr; 233(1-3):166-72. PubMed ID: 16904809
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Reactivation of organophosphate-inhibited human AChE by combinations of obidoxime and HI 6 in vitro.
    Worek F; Aurbek N; Thiermann H
    J Appl Toxicol; 2007; 27(6):582-8. PubMed ID: 17370251
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Design, synthesis and evaluation of novel nonquaternary and 3 non-oxime reactivators for acetylcholinesterase inhibited by organophosphates.
    Bi H; Ouyang Q; Wei Z; Zheng Z
    Bioorg Chem; 2020 Jul; 100():103902. PubMed ID: 32388435
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Mechanism of interaction of novel uncharged, centrally active reactivators with OP-hAChE conjugates.
    Radić Z; Sit RK; Garcia E; Zhang L; Berend S; Kovarik Z; Amitai G; Fokin VV; Barry Sharpless K; Taylor P
    Chem Biol Interact; 2013 Mar; 203(1):67-71. PubMed ID: 22975155
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 16.