BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

337 related articles for article (PubMed ID: 27526040)

  • 1. Design and synthesis of new potent PTP1B inhibitors with the skeleton of 2-substituted imino-3-substituted-5-heteroarylidene-1,3-thiazolidine-4-one: Part I.
    Meng G; Zheng M; Wang M; Tong J; Ge W; Zhang J; Zheng A; Li J; Gao L; Li J
    Eur J Med Chem; 2016 Oct; 122():756-769. PubMed ID: 27526040
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design, synthesis and docking study of 5-(substituted benzylidene)thiazolidine-2,4-dione derivatives as inhibitors of protein tyrosine phosphatase 1B.
    Wang Z; Liu Z; Lee W; Kim SN; Yoon G; Cheon SH
    Bioorg Med Chem Lett; 2014 Aug; 24(15):3337-40. PubMed ID: 24953600
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and biological evaluation of novel thiadiazole amides as potent Cdc25B and PTP1B inhibitors.
    Li Y; Yu Y; Jin K; Gao L; Luo T; Sheng L; Shao X; Li J
    Bioorg Med Chem Lett; 2014 Sep; 24(17):4125-8. PubMed ID: 25124112
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis, biological evaluation and in silico studies of 5-(3-methoxybenzylidene)thiazolidine-2,4-dione analogues as PTP1B inhibitors.
    Mahapatra MK; Kumar R; Kumar M
    Bioorg Chem; 2017 Apr; 71():1-9. PubMed ID: 28126289
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Identification of 2-substituted ethenesulfonic acid ester derivatives as novel, potent and selective inhibitors of protein tyrosine phosphatase 1B.
    Deng X; Liu J; Jin Y; Zhang Y; He W; Bao J; Liu W; Jiang F; Fu L
    Pharmazie; 2015 Dec; 70(12):777-83. PubMed ID: 26817274
    [TBL] [Abstract][Full Text] [Related]  

  • 6. A Library of Thiazolidin-4-one Derivatives as Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitors: An Attempt To Discover Novel Antidiabetic Agents.
    Patel AD; Pasha TY; Lunagariya P; Shah U; Bhambharoliya T; Tripathi RKP
    ChemMedChem; 2020 Jul; 15(13):1229-1242. PubMed ID: 32390300
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design and synthesis of 2-substituted benzoxazoles as novel PTP1B inhibitors.
    Chandrasekharappa AP; Badiger SE; Dubey PK; Panigrahi SK; Manukonda SR
    Bioorg Med Chem Lett; 2013 May; 23(9):2579-84. PubMed ID: 23528300
    [TBL] [Abstract][Full Text] [Related]  

  • 8. New chromone derivatives bearing thiazolidine-2,4-dione moiety as potent PTP1B inhibitors: Synthesis and biological activity evaluation.
    Zheng Y; Lu L; Li M; Xu D; Zhang L; Xiong Z; Zhou Y; Li J; Xu X; Zhang K; Xu L
    Bioorg Chem; 2024 Feb; 143():106985. PubMed ID: 38007892
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design, synthesis, and biological evaluation of 2-substituted ethenesulfonic acid ester derivatives as selective PTP1B inhibitors.
    Liu J; Deng X; Jin Y; Xu B; Liu W; Jiang F; Fu L
    Pharmazie; 2015 Jul; 70(7):446-51. PubMed ID: 26373204
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design, synthesis and insulin-sensitising effects of novel PTP1B inhibitors.
    Tang YB; Lu D; Chen Z; Hu C; Yang Y; Tian JY; Ye F; Wu L; Zhang ZY; Xiao Z
    Bioorg Med Chem Lett; 2013 Apr; 23(8):2313-8. PubMed ID: 23499238
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of small peptide compounds, molecular docking, and inhibitory activity evaluation against phosphatases PTP1B and SHP2.
    Kostrzewa T; Sahu KK; Gorska-Ponikowska M; Tuszynski JA; Kuban-Jankowska A
    Drug Des Devel Ther; 2018; 12():4139-4147. PubMed ID: 30584278
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Potent protein tyrosine phosphatase 1B (PTP1B) inhibiting constituents from Anoectochilus chapaensis and molecular docking studies.
    Cai J; Zhao L; Tao W
    Pharm Biol; 2015 Jul; 53(7):1030-4. PubMed ID: 25609152
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Discovery of novel, high potent, ABC type PTP1B inhibitors with TCPTP selectivity and cellular activity.
    Liu P; Du Y; Song L; Shen J; Li Q
    Eur J Med Chem; 2016 Aug; 118():27-33. PubMed ID: 27123900
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Toward a treatment of diabesity: Rational design, synthesis and biological evaluation of benzene-sulfonamide derivatives as a new class of PTP-1B inhibitors.
    Ghareb N; El-Sayed NM; Abdelhameed R; Yamada K; Elgawish MS
    Bioorg Chem; 2019 May; 86():322-338. PubMed ID: 30743173
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and biological evaluation of 2,4,6-trihydroxychalcone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
    Sun LP; Gao LX; Ma WP; Nan FJ; Li J; Piao HR
    Chem Biol Drug Des; 2012 Oct; 80(4):584-90. PubMed ID: 22805439
    [TBL] [Abstract][Full Text] [Related]  

  • 16. 5-Arylidene-2-phenylimino-4-thiazolidinones as PTP1B and LMW-PTP inhibitors.
    Ottanà R; Maccari R; Ciurleo R; Paoli P; Jacomelli M; Manao G; Camici G; Laggner C; Langer T
    Bioorg Med Chem; 2009 Mar; 17(5):1928-37. PubMed ID: 19217304
    [TBL] [Abstract][Full Text] [Related]  

  • 17. In silico modelling and molecular dynamics simulation studies of thiazolidine based PTP1B inhibitors.
    Mahapatra MK; Bera K; Singh DV; Kumar R; Kumar M
    J Biomol Struct Dyn; 2018 Apr; 36(5):1195-1211. PubMed ID: 28393626
    [TBL] [Abstract][Full Text] [Related]  

  • 18. [Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].
    Du X; Zhang SE; Liu JZ; Nie FL; Ye F; Tian JY; Xiao ZY
    Yao Xue Xue Bao; 2012 Mar; 47(3):367-73. PubMed ID: 22645761
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and biological evaluation of heterocyclic ring-substituted maslinic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.
    Qiu WW; Shen Q; Yang F; Wang B; Zou H; Li JY; Li J; Tang J
    Bioorg Med Chem Lett; 2009 Dec; 19(23):6618-22. PubMed ID: 19846303
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B.
    Li XQ; Xu Q; Luo J; Wang LJ; Jiang B; Zhang RS; Shi DY
    Eur J Med Chem; 2017 Aug; 136():348-359. PubMed ID: 28511130
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 17.