These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

224 related articles for article (PubMed ID: 27688182)

  • 21. Substituted 1,3-dioxoisoindoline-4-aminoquinolines coupled via amide linkers: Synthesis, antiplasmodial and cytotoxic evaluation.
    Rani A; Legac J; Rosenthal PJ; Kumar V
    Bioorg Chem; 2019 Jul; 88():102912. PubMed ID: 30991190
    [TBL] [Abstract][Full Text] [Related]  

  • 22. 4-Aminoquinoline-β-lactam conjugates: synthesis, antimalarial, and antitubercular evaluation.
    Raj R; Biot C; Carrère-Kremer S; Kremer L; Guérardel Y; Gut J; Rosenthal PJ; Kumar V
    Chem Biol Drug Des; 2014 Feb; 83(2):191-7. PubMed ID: 24034147
    [TBL] [Abstract][Full Text] [Related]  

  • 23. 1H-1,2,3-Triazole-tethered isatin-7-chloroquinoline and 3-hydroxy-indole-7-chloroquinoline conjugates: synthesis and antimalarial evaluation.
    Raj R; Gut J; Rosenthal PJ; Kumar V
    Bioorg Med Chem Lett; 2014 Feb; 24(3):756-9. PubMed ID: 24424135
    [TBL] [Abstract][Full Text] [Related]  

  • 24. New compounds hybrids 1h-1,2,3-triazole-quinoline against Plasmodium falciparum.
    Boechat N; Ferreira Mde L; Pinheiro LC; Jesus AM; Leite MM; Júnior CC; Aguiar AC; de Andrade IM; Krettli AU
    Chem Biol Drug Des; 2014 Sep; 84(3):325-32. PubMed ID: 24803084
    [TBL] [Abstract][Full Text] [Related]  

  • 25. 1H-1,2,3-triazole tethered isatin-ferrocene conjugates: Synthesis and in vitro antimalarial evaluation.
    Kumar K; Pradines B; Madamet M; Amalvict R; Benoit N; Kumar V
    Eur J Med Chem; 2014 Nov; 87():801-4. PubMed ID: 25440881
    [TBL] [Abstract][Full Text] [Related]  

  • 26. Synthesis of ring-substituted 4-aminoquinolines and evaluation of their antimalarial activities.
    Madrid PB; Sherrill J; Liou AP; Weisman JL; Derisi JL; Guy RK
    Bioorg Med Chem Lett; 2005 Feb; 15(4):1015-8. PubMed ID: 15686903
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Design, synthesis and anti-plasmodial evaluation in vitro of new 4-aminoquinoline isatin derivatives.
    Chiyanzu I; Clarkson C; Smith PJ; Lehman J; Gut J; Rosenthal PJ; Chibale K
    Bioorg Med Chem; 2005 May; 13(9):3249-61. PubMed ID: 15809160
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Comparison of the antiplasmodial and falcipain-2 inhibitory activity of beta-amino alcohol thiolactone-chalcone and isatin-chalcone hybrids.
    Hans RH; Gut J; Rosenthal PJ; Chibale K
    Bioorg Med Chem Lett; 2010 Apr; 20(7):2234-7. PubMed ID: 20206517
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Antimalarial activity of ferrocenyl chalcones.
    Wu X; Wilairat P; Go ML
    Bioorg Med Chem Lett; 2002 Sep; 12(17):2299-302. PubMed ID: 12161120
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Metallocene-based antimalarials: an exploration into the influence of the ferrocenyl moiety on in vitro antimalarial activity in chloroquine-sensitive and chloroquine-resistant strains of Plasmodium falciparum.
    Blackie MA; Beagley P; Croft SL; Kendrick H; Moss JR; Chibale K
    Bioorg Med Chem; 2007 Oct; 15(20):6510-6. PubMed ID: 17693090
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Application of multicomponent reactions to antimalarial drug discovery. Part 3: discovery of aminoxazole 4-aminoquinolines with potent antiplasmodial activity in vitro.
    Musonda CC; Little S; Yardley V; Chibale K
    Bioorg Med Chem Lett; 2007 Sep; 17(17):4733-6. PubMed ID: 17644333
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Design, Synthesis, and Evaluation of Novel Ferroquine and Phenylequine Analogues as Potential Antiplasmodial Agents.
    Jacobs L; de Kock C; de Villiers KA; Smith PJ; Smith VJ; van Otterlo WA; Blackie MA
    ChemMedChem; 2015 Dec; 10(12):2099-110. PubMed ID: 26447782
    [TBL] [Abstract][Full Text] [Related]  

  • 33. Trioxaferroquines as new hybrid antimalarial drugs.
    Bellot F; Coslédan F; Vendier L; Brocard J; Meunier B; Robert A
    J Med Chem; 2010 May; 53(10):4103-9. PubMed ID: 20443628
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Synthesis, characterization, and antiplasmodial activity of polymer-incorporated aminoquinolines.
    Aderibigbe BA; Neuse EW; Sadiku ER; Ray SS; Smith PJ
    J Biomed Mater Res A; 2014 Jun; 102(6):1941-9. PubMed ID: 23853120
    [TBL] [Abstract][Full Text] [Related]  

  • 35. Probing the role of the covalent linkage of ferrocene into a chloroquine template.
    Biot C; Daher W; Ndiaye CM; Melnyk P; Pradines B; Chavain N; Pellet A; Fraisse L; Pelinski L; Jarry C; Brocard J; Khalife J; Forfar-Bares I; Dive D
    J Med Chem; 2006 Jul; 49(15):4707-14. PubMed ID: 16854077
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Synthesis, in vitro antimalarial activity and cytotoxicity of novel 4-aminoquinolinyl-chalcone amides.
    Smit FJ; N'da DD
    Bioorg Med Chem; 2014 Feb; 22(3):1128-38. PubMed ID: 24411478
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparum.
    Sashidhara KV; Avula SR; Palnati GR; Singh SV; Srivastava K; Puri SK; Saxena JK
    Bioorg Med Chem Lett; 2012 Sep; 22(17):5455-9. PubMed ID: 22850213
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Application of multicomponent reactions to antimalarial drug discovery. Part 2: New antiplasmodial and antitrypanosomal 4-aminoquinoline gamma- and delta-lactams via a 'catch and release' protocol.
    Musonda CC; Gut J; Rosenthal PJ; Yardley V; Carvalho de Souza RC; Chibale K
    Bioorg Med Chem; 2006 Aug; 14(16):5605-15. PubMed ID: 16690319
    [TBL] [Abstract][Full Text] [Related]  

  • 39. In vitro antimalarial activity, β-haematin inhibition and structure-activity relationships in a series of quinoline triazoles.
    Joshi MC; Wicht KJ; Taylor D; Hunter R; Smith PJ; Egan TJ
    Eur J Med Chem; 2013 Nov; 69():338-47. PubMed ID: 24077524
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Bioisosteric ferrocenyl aminoquinoline-benzimidazole hybrids: Antimicrobial evaluation and mechanistic insights.
    Baartzes N; Stringer T; Seldon R; Warner DF; Taylor D; Wittlin S; Chibale K; Smith GS
    Eur J Med Chem; 2019 Oct; 180():121-133. PubMed ID: 31301563
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 12.