BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

157 related articles for article (PubMed ID: 27731647)

  • 21. Rational design, chemical synthesis and biological evaluation of novel biguanides exploring species-specificity responsiveness of TAAR1 agonists.
    Guariento S; Tonelli M; Espinoza S; Gerasimov AS; Gainetdinov RR; Cichero E
    Eur J Med Chem; 2018 Feb; 146():171-184. PubMed ID: 29407948
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Vasodilator Effect of Trace Amines, 3-Iodothyronamine, and RO5263397 in the Rat Perfused Kidney: Comparison with Tryptamine.
    Jragh D; Chandrasekhar B; Yousif MHM; Oriowo MA
    Pharmacology; 2023; 108(4):368-378. PubMed ID: 37245501
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Exploring the determinants of trace amine-associated receptor 1's functional selectivity for the stereoisomers of amphetamine and methamphetamine.
    Reese EA; Norimatsu Y; Grandy MS; Suchland KL; Bunzow JR; Grandy DK
    J Med Chem; 2014 Jan; 57(2):378-90. PubMed ID: 24354319
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Insights into the structure and pharmacology of the human trace amine-associated receptor 1 (hTAAR1): homology modelling and docking studies.
    Cichero E; Espinoza S; Gainetdinov RR; Brasili L; Fossa P
    Chem Biol Drug Des; 2013 Apr; 81(4):509-16. PubMed ID: 22883051
    [TBL] [Abstract][Full Text] [Related]  

  • 25. Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling.
    Grossi G; Scarano N; Musumeci F; Tonelli M; Kanov E; Carbone A; Fossa P; Gainetdinov RR; Cichero E; Schenone S
    Molecules; 2024 Apr; 29(8):. PubMed ID: 38675561
    [TBL] [Abstract][Full Text] [Related]  

  • 26. New diphenylmethane derivatives as peroxisome proliferator-activated receptor alpha/gamma dual agonists endowed with anti-proliferative effects and mitochondrial activity.
    Piemontese L; Cerchia C; Laghezza A; Ziccardi P; Sblano S; Tortorella P; Iacobazzi V; Infantino V; Convertini P; Dal Piaz F; Lupo A; Colantuoni V; Lavecchia A; Loiodice F
    Eur J Med Chem; 2017 Feb; 127():379-397. PubMed ID: 28076827
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Discovery of potential TAAR1 agonist targeting neurological and psychiatric disorders: An in silico approach.
    Garisetti V; Dhanabalan AK; Dasararaju G
    Int J Biol Macromol; 2024 Apr; 264(Pt 2):130528. PubMed ID: 38431013
    [TBL] [Abstract][Full Text] [Related]  

  • 28. 3-Iodothyronamine and Derivatives: New Allies Against Metabolic Syndrome?
    Rutigliano G; Bandini L; Sestito S; Chiellini G
    Int J Mol Sci; 2020 Mar; 21(6):. PubMed ID: 32183490
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Trace Amine-Associated Receptor 1 Agonists as Narcolepsy Therapeutics.
    Black SW; Schwartz MD; Chen TM; Hoener MC; Kilduff TS
    Biol Psychiatry; 2017 Nov; 82(9):623-633. PubMed ID: 27919403
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Selective antagonists of mouse trace amine-associated receptor 1 (mTAAR1): discovery of EPPTB (RO5212773).
    Stalder H; Hoener MC; Norcross RD
    Bioorg Med Chem Lett; 2011 Feb; 21(4):1227-31. PubMed ID: 21237643
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Efficient synthesis of a multi-substituted diphenylmethane skeleton as a steroid mimetic.
    Misawa T; Tanaka K; Demizu Y; Kurihara M
    Bioorg Med Chem Lett; 2017 Jun; 27(11):2590-2593. PubMed ID: 28400239
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Design, synthesis and biological evaluation of a novel class of potent TGR5 agonists based on a 4-phenyl pyridine scaffold.
    Zhu J; Ning M; Guo C; Zhang L; Pan G; Leng Y; Shen J
    Eur J Med Chem; 2013 Nov; 69():55-68. PubMed ID: 24007860
    [TBL] [Abstract][Full Text] [Related]  

  • 33. Further structurally constrained analogues of cis-(6-benzhydrylpiperidin-3-yl)benzylamine with elucidation of bioactive conformation: discovery of 1,4-diazabicyclo[3.3.1]nonane derivatives and evaluation of their biological properties for the monoamine transporters.
    Kolhatkar R; Cook CD; Ghorai SK; Deschamps J; Beardsley PM; Reith ME; Dutta AK
    J Med Chem; 2004 Oct; 47(21):5101-13. PubMed ID: 15456254
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Trace amine-associated receptor 1 activation silences GSK3β signaling of TAAR1 and D2R heteromers.
    Harmeier A; Obermueller S; Meyer CA; Revel FG; Buchy D; Chaboz S; Dernick G; Wettstein JG; Iglesias A; Rolink A; Bettler B; Hoener MC
    Eur Neuropsychopharmacol; 2015 Nov; 25(11):2049-61. PubMed ID: 26372541
    [TBL] [Abstract][Full Text] [Related]  

  • 35. Design, synthesis, and evaluation of phenylglycinols and phenyl amines as agonists of GPR88.
    Dzierba CD; Bi Y; Dasgupta B; Hartz RA; Ahuja V; Cianchetta G; Kumi G; Dong L; Aleem S; Fink C; Garcia Y; Green M; Han J; Kwon S; Qiao Y; Wang J; Zhang Y; Liu Y; Zipp G; Liang Z; Burford N; Ferrante M; Bertekap R; Lewis M; Cacace A; Grace J; Wilson A; Nouraldeen A; Westphal R; Kimball D; Carson K; Bronson JJ; Macor JE
    Bioorg Med Chem Lett; 2015 Apr; 25(7):1448-52. PubMed ID: 25690789
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Design, synthesis, and biological evaluation of novel pan agonists of FFA1, PPARγ and PPARδ.
    Li Z; Zhou Z; Deng F; Li Y; Zhang D; Zhang L
    Eur J Med Chem; 2018 Nov; 159():267-276. PubMed ID: 30296685
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Continued SAR exploration of 1,2,4-thiadiazole-containing scaffolds in the design of free fatty acid receptor 1 (GPR40) agonists.
    Krasavin M; Lukin A; Bakholdina A; Zhurilo N; Onopchenko O; Borysko P; Zozulya S; Moore D; Tikhonova IG
    Eur J Med Chem; 2017 Nov; 140():229-238. PubMed ID: 28938138
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Biogenic amines activate blood leukocytes via trace amine-associated receptors TAAR1 and TAAR2.
    Babusyte A; Kotthoff M; Fiedler J; Krautwurst D
    J Leukoc Biol; 2013 Mar; 93(3):387-94. PubMed ID: 23315425
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Ligand recognition and G-protein coupling of trace amine receptor TAAR1.
    Xu Z; Guo L; Yu J; Shen S; Wu C; Zhang W; Zhao C; Deng Y; Tian X; Feng Y; Hou H; Su L; Wang H; Guo S; Wang H; Wang K; Chen P; Zhao J; Zhang X; Yong X; Cheng L; Liu L; Yang S; Yang F; Wang X; Yu X; Xu Y; Sun JP; Yan W; Shao Z
    Nature; 2023 Dec; 624(7992):672-681. PubMed ID: 37935376
    [TBL] [Abstract][Full Text] [Related]  

  • 40. In-vivo pharmacology of Trace-Amine Associated Receptor 1.
    Lam VM; Espinoza S; Gerasimov AS; Gainetdinov RR; Salahpour A
    Eur J Pharmacol; 2015 Sep; 763(Pt B):136-42. PubMed ID: 26093041
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 8.