167 related articles for article (PubMed ID: 27809515)
1. Structure-Cytotoxicity Relationships of Analogues of N
Toader D; Wang F; Gingipalli L; Vasbinder M; Roth M; Mao S; Block M; Harper J; Thota S; Su M; Ma J; Bedian V; Kamal A
J Med Chem; 2016 Dec; 59(23):10781-10787. PubMed ID: 27809515
[TBL] [Abstract][Full Text] [Related]
2. Cytotoxic simplified tubulysin analogues.
Raghavan B; Balasubramanian R; Steele JC; Sackett DL; Fecik RA
J Med Chem; 2008 Mar; 51(6):1530-3. PubMed ID: 18314944
[TBL] [Abstract][Full Text] [Related]
3. Structure-activity relationships of tubulysin analogues.
Courter JR; Hamilton JZ; Hendrick NR; Zaval M; Waight AB; Lyon RP; Senter PD; Jeffrey SC; Burke PJ
Bioorg Med Chem Lett; 2020 Jul; 30(14):127241. PubMed ID: 32527543
[TBL] [Abstract][Full Text] [Related]
4. Total Synthesis and Biological Evaluation of Tubulysin Analogues.
Colombo R; Wang Z; Han J; Balachandran R; Daghestani HN; Camarco DP; Vogt A; Day BW; Mendel D; Wipf P
J Org Chem; 2016 Nov; 81(21):10302-10320. PubMed ID: 27447195
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and antiproliferative activity of C- and N-terminal analogues of culicinin D.
Li FF; Stubbing LA; Kavianinia I; Abbattista MR; Harris PWR; Smaill JB; Patterson AV; Brimble MA
Bioorg Med Chem Lett; 2020 Aug; 30(16):127331. PubMed ID: 32631536
[TBL] [Abstract][Full Text] [Related]
6. Synthesis of novel peptides through Ugi-ligation and their anti-cancer activities.
Tahoori F; Sheikhnejad R; Balalaie S; Sadjadi M
Amino Acids; 2013 Oct; 45(4):975-81. PubMed ID: 23864432
[TBL] [Abstract][Full Text] [Related]
7. Total Synthesis and Biological Evaluation of Natural and Designed Tubulysins.
Nicolaou KC; Yin J; Mandal D; Erande RD; Klahn P; Jin M; Aujay M; Sandoval J; Gavrilyuk J; Vourloumis D
J Am Chem Soc; 2016 Feb; 138(5):1698-708. PubMed ID: 26829208
[TBL] [Abstract][Full Text] [Related]
8. Exploration of the carmaphycins as payloads in antibody drug conjugate anticancer agents.
Almaliti J; Miller B; Pietraszkiewicz H; Glukhov E; Naman CB; Kline T; Hanson J; Li X; Zhou S; Valeriote FA; Gerwick WH
Eur J Med Chem; 2019 Jan; 161():416-432. PubMed ID: 30384045
[TBL] [Abstract][Full Text] [Related]
9. Aromatic oligopeptides with chlorambucil moiety--synthesis and biological evaluation.
Bartulewicz D
Acta Pol Pharm; 2005; 62(6):451-5. PubMed ID: 16583984
[TBL] [Abstract][Full Text] [Related]
10. Pretubulysin, a potent and chemically accessible tubulysin precursor from Angiococcus disciformis.
Ullrich A; Chai Y; Pistorius D; Elnakady YA; Herrmann JE; Weissman KJ; Kazmaier U; Müller R
Angew Chem Int Ed Engl; 2009; 48(24):4422-5. PubMed ID: 19431172
[TBL] [Abstract][Full Text] [Related]
11. Total synthesis of the putative structure of lucentamycin A.
Pal U; Ranatunga S; Ariyarathna Y; Del Valle JR
Org Lett; 2009 Nov; 11(22):5298-301. PubMed ID: 19863114
[TBL] [Abstract][Full Text] [Related]
12. Minimal C-terminal modification boosts peptide self-assembling ability for necroptosis of cancer cells.
Feng Z; Wang H; Du X; Shi J; Li J; Xu B
Chem Commun (Camb); 2016 May; 52(37):6332-5. PubMed ID: 27087169
[TBL] [Abstract][Full Text] [Related]
13. Pentapeptides for the treatment of small cell lung cancer: Optimisation by N
Haitham Abusara O; Freeman S; Aojula HS
Eur J Med Chem; 2017 Sep; 137():221-232. PubMed ID: 28595067
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and antimitotic/cytotoxic activity of hemiasterlin analogues.
Nieman JA; Coleman JE; Wallace DJ; Piers E; Lim LY; Roberge M; Andersen RJ
J Nat Prod; 2003 Feb; 66(2):183-99. PubMed ID: 12608848
[TBL] [Abstract][Full Text] [Related]
15. Toward Angiogenesis Inhibitors Based on the Conjugation of Organometallic Platinum(II) Complexes to RGD Peptides.
Zamora A; Gandioso A; Massaguer A; Buenestado S; Calvis C; Hernández JL; Mitjans F; Rodríguez V; Ruiz J; Marchán V
ChemMedChem; 2018 Sep; 13(17):1755-1762. PubMed ID: 29932312
[TBL] [Abstract][Full Text] [Related]
16. Total synthesis of tubulysin U and its C-4 epimer.
Yang XD; Dong CM; Chen J; Ding YH; Liu Q; Ma XY; Zhang Q; Chen Y
Chem Asian J; 2013 Jun; 8(6):1213-22. PubMed ID: 23576385
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and structure-activity relationship studies of novel tubulysin U analogues--effect on cytotoxicity of structural variations in the tubuvaline fragment.
Shankar SP; Jagodzinska M; Malpezzi L; Lazzari P; Manca I; Greig IR; Sani M; Zanda M
Org Biomol Chem; 2013 Apr; 11(14):2273-87. PubMed ID: 23411563
[TBL] [Abstract][Full Text] [Related]
18. Improved Total Synthesis of Tubulysins and Design, Synthesis, and Biological Evaluation of New Tubulysins with Highly Potent Cytotoxicities against Cancer Cells as Potential Payloads for Antibody-Drug Conjugates.
Nicolaou KC; Erande RD; Yin J; Vourloumis D; Aujay M; Sandoval J; Munneke S; Gavrilyuk J
J Am Chem Soc; 2018 Mar; 140(10):3690-3711. PubMed ID: 29381062
[TBL] [Abstract][Full Text] [Related]
19. β-Glucuronidase triggers extracellular MMAE release from an integrin-targeted conjugate.
López Rivas P; Müller C; Breunig C; Hechler T; Pahl A; Arosio D; Belvisi L; Pignataro L; Dal Corso A; Gennari C
Org Biomol Chem; 2019 May; 17(19):4705-4710. PubMed ID: 31020985
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and anticancer evaluation of spermatinamine analogues.
Moosa BA; Sagar S; Li S; Esau L; Kaur M; Khashab NM
Bioorg Med Chem Lett; 2016 Mar; 26(6):1629-1632. PubMed ID: 26874403
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]