139 related articles for article (PubMed ID: 2795598)
1. Enantioselectivity of muscarinic antagonists. Isomeric 2-cyclohexyl-2-phenyl-5-[(dimethylamino)methyl]-1,3-oxathiolane 3-oxide methiodides.
Romanelli MN; Gualtieri F; Angeli P; Picchio MT
J Med Chem; 1989 Oct; 32(10):2269-73. PubMed ID: 2795598
[TBL] [Abstract][Full Text] [Related]
2. Enantioselectivity of muscarinic antagonists. Isomeric 2-cyclohexyl-2-phenyl-5-[(dimethylamino)methyl]-1,3-oxathiolane methiodides.
Romanelli MN; Gualtieri F; Valle G; Brasili L; Angeli P
J Med Chem; 1988 Sep; 31(9):1703-8. PubMed ID: 3411599
[TBL] [Abstract][Full Text] [Related]
3. Enantioselectivity of muscarinic antagonists. 2,2-Dicyclohexyl-5-[(dimethylamino)methyl]-1,3-oxathiolane methiodides and related 3-oxides.
Romanelli MN; Teodori E; Gualtieri F; Angeli P; Brasili L
J Med Chem; 1988 Sep; 31(9):1698-702. PubMed ID: 3411598
[TBL] [Abstract][Full Text] [Related]
4. Resolution, absolute configuration, and cholinergic enantioselectivity of (+)- and (-)-cis-2-methyl-5-[(dimethylamino)methyl]-1,3-oxathiolane methiodide.
Teodori E; Gualtieri F; Angeli P; Brasili L; Giannella M; Pigini M
J Med Chem; 1986 Sep; 29(9):1610-5. PubMed ID: 3746812
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and calcium channel-modulating effects of alkyl (or cycloalkyl) 1,4-dihydro-2,6-dimethyl-3-nitro-4-pyridyl-5-pyridinecarboxylate racemates and enantiomers.
Ramesh M; Matowe WC; Akula MR; Vo D; Dagnino L; Li-Kwong-Ken MC; Wolowyk MW; Knaus EE
J Med Chem; 1998 Feb; 41(4):509-14. PubMed ID: 9484501
[TBL] [Abstract][Full Text] [Related]
6. Chiral muscarinic agonists possessing a 1,3-oxathiolane nucleus: enantio- and tissue-selectivity on isolated preparations of guinea-pig ileum and atria and of rat urinary bladder.
Angeli P; Brasili L; Giannella M; Gualtieri F; Picchio MT; Teodori E
Naunyn Schmiedebergs Arch Pharmacol; 1988 Mar; 337(3):241-5. PubMed ID: 3393229
[TBL] [Abstract][Full Text] [Related]
7. Molecular requirements for antimuscarinic activity in 1,3-oxathiolanes.
Angeli P; Bacchiocchi D; Giannella M; Pigini M; Romanelli MN
Drug Des Deliv; 1988 May; 2(4):263-72. PubMed ID: 3255319
[TBL] [Abstract][Full Text] [Related]
8. Resolution, absolute configuration, and cholinergic enantioselectivity of (-)- and (+)-c-2-methyl-r-5-[(dimethylamino)methyl]-1,3-oxathiolane t-3-oxide methiodide and related sulfones.
Teodori E; Gualtieri F; Angeli P; Brasili L; Giannella M
J Med Chem; 1987 Oct; 30(10):1934-8. PubMed ID: 3656366
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and muscarinic receptors affinity of a series of antagonist bivalent ligands.
Piergentili A; Quaglia W; Tayebati SK; Paparelli F; Malmusi L; Brasili L
Farmaco; 1994 Feb; 49(2):83-7. PubMed ID: 7516166
[TBL] [Abstract][Full Text] [Related]
10. New analogues of oxotremorine and oxotremorine-M: estimation of their in vitro affinity and efficacy at muscarinic receptor subtypes.
Barocelli E; Ballabeni V; Bertoni S; Dallanoce C; De Amici M; De Micheli C; Impicciatore M
Life Sci; 2000 Jun; 67(6):717-23. PubMed ID: 12659177
[TBL] [Abstract][Full Text] [Related]
11. Nitrile oxides in medicinal chemistry. 3. Synthesis and bioenantioselectivity of (+)- and (-)-2-methyl-5-[(dimethylamino)-methyl]-3-oxo-isoxazolidine methiodide.
De Amici M; De Micheli C; Grana E; Lucchelli A; Zonta F
Farmaco; 1990 Jul; 45(7-8):859-66. PubMed ID: 2282119
[TBL] [Abstract][Full Text] [Related]
12. Synthesis, affinity profile, and functional activity of muscarinic antagonists with a 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl)pyrrolidine structure.
Dei S; Bellucci C; Buccioni M; Ferraroni M; Guandalini L; Manetti D; Martini E; Marucci G; Matucci R; Nesi M; Romanelli MN; Scapecchi S; Teodori E
J Med Chem; 2007 Mar; 50(6):1409-13. PubMed ID: 17305327
[TBL] [Abstract][Full Text] [Related]
13. Cholinergic agents structurally related to furtrethonium. 2. Synthesis and antimuscarinic activity of a series of N-[5-[(1'-substituted-acetoxy) methyl]-2-furfuryl]dialkylamines.
Feriani A; Gaviraghi G; Toson G; Mor M; Barbieri A; Grana E; Boselli C; Guarneri M; Simoni D; Manfredini S
J Med Chem; 1994 Dec; 37(25):4278-87. PubMed ID: 7996539
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and pharmacological evaluation of enantiomerically pure 4-deoxy-4-fluoromuscarines.
Bravo P; Resnati G; Angeli P; Frigerio M; Viani F; Arnone A; Marucci G; Cantalamessa F
J Med Chem; 1992 Aug; 35(17):3102-10. PubMed ID: 1507199
[TBL] [Abstract][Full Text] [Related]
15. In vitro and in vivo antimuscarinic effects of (-)cis 2,3-dihydro-3-(4-methylpiperazinylmethyl)-2-phenyl-1,5 benzothiazepin-4-(5H)one HCl (BTM-1086) in guinea pig peripheral tissues.
Noronha-Blob L; Sturm BL; Lowe VC; Jackson KN; Kachur JF
Life Sci; 1990; 46(17):1223-31. PubMed ID: 2338887
[TBL] [Abstract][Full Text] [Related]
16. Pharmacological characteristics of liriodenine, isolated from Fissistigma glaucescens, a novel muscarinic receptor antagonist in guinea-pigs.
Lin CH; Chang GJ; Su MJ; Wu YC; Teng CM; Ko FN
Br J Pharmacol; 1994 Sep; 113(1):275-81. PubMed ID: 7812621
[TBL] [Abstract][Full Text] [Related]
17. Muscarinic receptor subtype specificity of (N,N-dialkylamino)alkyl 2-cyclohexyl-2-phenylpropionates: cylexphenes (cyclohexyl-substituted aprophen analogues).
Leader H; Gordon RK; Baumgold J; Boyd VL; Newman AH; Smejkal RM; Chiang PK
J Med Chem; 1992 Apr; 35(7):1290-5. PubMed ID: 1560441
[TBL] [Abstract][Full Text] [Related]
18. Distinct functional muscarinic receptors in guinea-pig gallbladder, ileum and atria.
Karaalp A; Akici A; Akbulut H; Ulusoy NB; Oktay S
Pharmacol Res; 1999 May; 39(5):389-95. PubMed ID: 10328997
[TBL] [Abstract][Full Text] [Related]
19. Selective inactivation of muscarinic M2 and M3 receptors in guinea-pig ileum and atria in vitro.
Eglen RM; Harris GC
Br J Pharmacol; 1993 Aug; 109(4):946-52. PubMed ID: 8401947
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and antagonistic activity at muscarinic receptor subtypes of some derivatives of diphenidol.
Varoli L; Angeli P; Buccioni M; Burnelli S; Cavalli A; Marucci G; Recanatini M
Farmaco; 2003 Sep; 58(9):651-7. PubMed ID: 13679157
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]