BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

160 related articles for article (PubMed ID: 28002960)

  • 1. Characterization of New Cationic N,N-Dimethyl[70]fulleropyrrolidinium Iodide Derivatives as Potent HIV-1 Maturation Inhibitors.
    Castro E; Martinez ZS; Seong CS; Cabrera-Espinoza A; Ruiz M; Hernandez Garcia A; Valdez F; Llano M; Echegoyen L
    J Med Chem; 2016 Dec; 59(24):10963-10973. PubMed ID: 28002960
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Fullerene Derivatives Strongly Inhibit HIV-1 Replication by Affecting Virus Maturation without Impairing Protease Activity.
    Martinez ZS; Castro E; Seong CS; Cerón MR; Echegoyen L; Llano M
    Antimicrob Agents Chemother; 2016 Oct; 60(10):5731-41. PubMed ID: 27431232
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Fullerene derivatives as dual inhibitors of HIV-1 reverse transcriptase and protease.
    Yasuno T; Ohe T; Kataoka H; Hashimoto K; Ishikawa Y; Furukawa K; Tateishi Y; Kobayashi T; Takahashi K; Nakamura S; Mashino T
    Bioorg Med Chem Lett; 2021 Jan; 31():127675. PubMed ID: 33161121
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Insights into the activity of maturation inhibitor PF-46396 on HIV-1 clade C.
    Ghimire D; Timilsina U; Srivastava TP; Gaur R
    Sci Rep; 2017 Mar; 7():43711. PubMed ID: 28252110
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Fullerene Derivatives Prevent Packaging of Viral Genomic RNA into HIV-1 Particles by Binding Nucleocapsid Protein.
    Křížová I; Dostálková A; Castro E; Prchal J; Hadravová R; Kaufman F; Hrabal R; Ruml T; Llano M; Echegoyen L; Rumlová M
    Viruses; 2021 Dec; 13(12):. PubMed ID: 34960720
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Novel pyridinium-type fullerene derivatives as multitargeting inhibitors of HIV-1 reverse transcriptase, HIV-1 protease, and HCV NS5B polymerase.
    Kobayashi T; Yasuno T; Takahashi K; Nakamura S; Mashino T; Ohe T
    Bioorg Med Chem Lett; 2021 Oct; 49():128267. PubMed ID: 34271071
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis, stability, antiviral activity, and protease-bound structures of substrate-mimicking constrained macrocyclic inhibitors of HIV-1 protease.
    Tyndall JD; Reid RC; Tyssen DP; Jardine DK; Todd B; Passmore M; March DR; Pattenden LK; Bergman DA; Alewood D; Hu SH; Alewood PF; Birch CJ; Martin JL; Fairlie DP
    J Med Chem; 2000 Sep; 43(19):3495-504. PubMed ID: 11000004
    [TBL] [Abstract][Full Text] [Related]  

  • 8. New anti-HIV derivatives: synthesis and antiviral evaluation.
    De Michelis C; Rocheblave L; Priem G; Chermann JC; Kraus JL
    Bioorg Med Chem; 2000 Jun; 8(6):1253-62. PubMed ID: 10896105
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design, synthesis and biological evaluation of novel HIV-1 protease inhibitors with pentacyclic triterpenoids as P2-ligands.
    Zhu M; Du XN; Li YG; Zhang GN; Wang JX; Wang YC
    Bioorg Med Chem Lett; 2019 Feb; 29(3):357-361. PubMed ID: 30580917
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Alkyl Amine Bevirimat Derivatives Are Potent and Broadly Active HIV-1 Maturation Inhibitors.
    Urano E; Ablan SD; Mandt R; Pauly GT; Sigano DM; Schneider JP; Martin DE; Nitz TJ; Wild CT; Freed EO
    Antimicrob Agents Chemother; 2016 Jan; 60(1):190-7. PubMed ID: 26482309
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis, properties and photodynamic inactivation of Escherichia coli by novel cationic fullerene C60 derivatives.
    Spesia MB; Milanesio ME; Durantini EN
    Eur J Med Chem; 2008 Apr; 43(4):853-61. PubMed ID: 17706838
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and antiviral activity of new anti-HIV amprenavir bioisosteres.
    Rocheblave L; Bihel F; De Michelis C; Priem G; Courcambeck J; Bonnet B; Chermann JC; Kraus JL
    J Med Chem; 2002 Jul; 45(15):3321-4. PubMed ID: 12109915
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Human immunodeficiency virus type 1 Vif-derived peptides inhibit the viral protease and arrest virus production.
    Baraz L; Friedler A; Blumenzweig I; Nussinuv O; Chen N; Steinitz M; Gilon C; Kotler M
    FEBS Lett; 1998 Dec; 441(3):419-26. PubMed ID: 9891983
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design and evaluation of novel piperidine HIV-1 protease inhibitors with potency against DRV-resistant variants.
    Zhu M; Zhou H; Ma L; Dong B; Zhou J; Zhang G; Wang M; Wang J; Cen S; Wang Y
    Eur J Med Chem; 2021 Aug; 220():113450. PubMed ID: 33906049
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Reviewing HIV-1 Gag Mutations in Protease Inhibitors Resistance: Insights for Possible Novel Gag Inhibitor Designs.
    Su CT; Koh DW; Gan SK
    Molecules; 2019 Sep; 24(18):. PubMed ID: 31489889
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Enhanced replication of R5 HIV-1 isolates in vitro by a small-molecule reagent targeting HIV-1 protease.
    Wardle NJ; Hudson HR; Matthews RW; Nunn CM; Vella C; Bligh SW
    ChemMedChem; 2013 May; 8(5):719-21. PubMed ID: 23509042
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and anti-HIV activity of new C2 symmetric derivatives designed as HIV-1 protease inhibitors.
    Peçanha EP; Figueiredo LJ; Brindeiro RM; Tanuri A; Calazans AR; Antunes OA
    Farmaco; 2003 Feb; 58(2):149-57. PubMed ID: 12581781
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Advances in non-peptidomimetic HIV protease inhibitors.
    Pang X; Liu Z; Zhai G
    Curr Med Chem; 2014 Jun; 21(17):1997-2011. PubMed ID: 24533811
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Molecular Dynamics Simulation Study of the HIV-1 Protease Inhibit ion Using Fullerene and New Fullerene Derivatives of Carbon Nanostructures.
    Barzegar A; Naghizadeh E; Zakariazadeh M; Azamat J
    Mini Rev Med Chem; 2017; 17(7):633-647. PubMed ID: 27292780
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Structure-Activity Relationships of the Human Immunodeficiency Virus Type 1 Maturation Inhibitor PF-46396.
    Murgatroyd C; Pirrie L; Tran F; Smith TK; Westwood NJ; Adamson CS
    J Virol; 2016 Sep; 90(18):8181-97. PubMed ID: 27384665
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.